MA30576B1 - Formes cristallines de la 4-[2-(4-methylphenylsulfanyl)-phenyl] piperidine avec inhibition de la reabsorption de la serotonine et de la norepinephrine en combinaison pour le traitement de la douleur neuropathique - Google Patents

Formes cristallines de la 4-[2-(4-methylphenylsulfanyl)-phenyl] piperidine avec inhibition de la reabsorption de la serotonine et de la norepinephrine en combinaison pour le traitement de la douleur neuropathique

Info

Publication number
MA30576B1
MA30576B1 MA31551A MA31551A MA30576B1 MA 30576 B1 MA30576 B1 MA 30576B1 MA 31551 A MA31551 A MA 31551A MA 31551 A MA31551 A MA 31551A MA 30576 B1 MA30576 B1 MA 30576B1
Authority
MA
Morocco
Prior art keywords
methylphenylsulfanyl
piperidine
phenyl
treatment
reabsorption
Prior art date
Application number
MA31551A
Other languages
English (en)
Inventor
Benny Bang-Andersen
Andre Faldt
Tine Bryan Stensboel
Silke Miller
De Diego Heidi Lopez
Original Assignee
Lundbeck & Co As H
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38434468&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MA30576(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Lundbeck & Co As H filed Critical Lundbeck & Co As H
Publication of MA30576B1 publication Critical patent/MA30576B1/fr

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    • C—CHEMISTRY; METALLURGY
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
    • C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D211/20—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms
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    • C07C229/02—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C229/04—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated
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  • Psychiatry (AREA)
  • Diabetes (AREA)
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  • Orthopedic Medicine & Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Hematology (AREA)
  • Virology (AREA)
  • Urology & Nephrology (AREA)
  • Hospice & Palliative Care (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Psychology (AREA)
  • Obesity (AREA)
  • Emergency Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
  • Anesthesiology (AREA)
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Abstract

Des formes cristallines de 4-[2-(4-methylphenylsulfanyl)-phényle] pipéridine et leurs sels sont fournies par exemple, pour le traitement de la douleur neuropathique.
MA31551A 2006-06-16 2009-01-06 Formes cristallines de la 4-[2-(4-methylphenylsulfanyl)-phenyl] piperidine avec inhibition de la reabsorption de la serotonine et de la norepinephrine en combinaison pour le traitement de la douleur neuropathique MA30576B1 (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US80500906P 2006-06-16 2006-06-16
DKPA200600816 2006-06-16
DKPA200700423 2007-03-20

Publications (1)

Publication Number Publication Date
MA30576B1 true MA30576B1 (fr) 2009-07-01

Family

ID=38434468

Family Applications (1)

Application Number Title Priority Date Filing Date
MA31551A MA30576B1 (fr) 2006-06-16 2009-01-06 Formes cristallines de la 4-[2-(4-methylphenylsulfanyl)-phenyl] piperidine avec inhibition de la reabsorption de la serotonine et de la norepinephrine en combinaison pour le traitement de la douleur neuropathique

Country Status (14)

Country Link
US (4) US8299095B2 (fr)
EP (1) EP2044020B1 (fr)
JP (2) JP5318757B2 (fr)
AU (1) AU2007260356B2 (fr)
CA (1) CA2656057C (fr)
CY (1) CY1111619T1 (fr)
EA (1) EA016054B1 (fr)
HR (1) HRP20110412T1 (fr)
IL (1) IL195310A (fr)
MA (1) MA30576B1 (fr)
MX (1) MX2008016008A (fr)
NO (1) NO20090250L (fr)
PL (1) PL2044020T3 (fr)
WO (1) WO2007144006A1 (fr)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX2008016008A (es) * 2006-06-16 2009-01-16 Lundbeck & Co As H Formas cristalinas de 4-[2-(4-metilfenilsulfonil)-fenil] piperidina con inhibicion combinada de la recaptacion de serotonina y norepinefrina para el tratamiento del dolor neuropatico.
MY150647A (en) 2006-06-16 2014-02-14 Lundbeck & Co As H 1-[2-(2,4-dimethylphenylsulfanyl)-phenyl] piperazine as a compound with combined serotonin reuptake, 5-ht3 and 5-ht1a activity for the treatment of cognitive impairment
CA2784304A1 (fr) * 2006-06-16 2007-12-21 H. Lundbeck A/S Formes cristallines de la 4-[2-(4-methylphenylsulfanyl)-phenyl] piperidine avec inhibition de la reabsorption de la serotonine et de la norepinephrine en combinaison pour le traitement de la douleur neuropathique
TWI405588B (zh) * 2007-03-20 2013-08-21 Lundbeck & Co As H ４-〔２-（４-甲苯基硫基）-苯基〕哌啶之鹽類的液體調配物
TWI432194B (zh) 2007-03-20 2014-04-01 Lundbeck & Co As H ４-〔２-（４-甲基苯硫基）苯基〕哌啶之新穎治療用途
HRP20140044T1 (hr) 2007-06-15 2014-02-14 H. Lundbeck A/S 4-[2-(4-metilfenilsulfanil)fenil]piperidin za lijeäśenje iritabilnog sindroma crijeva (ibs)
TW200938194A (en) * 2007-12-14 2009-09-16 Lundbeck & Co As H Therapeutic uses of compounds having affinity to the serotonin transporter, serotonin receptors and noradrenalin transporter
UA98698C2 (en) * 2008-03-03 2012-06-11 Х. Луннбек А/С Phenylsulfanylphenyl-piperidines and process for the preparation thereof
TW201033181A (en) * 2009-02-17 2010-09-16 Lundbeck & Co As H Purification of 1-[2-(2,4-dimethylphenylsulfanyl)phenyl]piperazine
RS53539B1 (sr) * 2009-04-24 2015-02-27 H. Lundbeck A/S Tečne formulacije soli 1-[2-(2,4-dimetilfenilsulfanil)fenil] piperazina
MX2011011579A (es) * 2009-04-30 2012-01-27 Supernus Pharmaceuticals Inc Metodo de tratamiento contra la depresion.
JP5787881B2 (ja) * 2010-04-30 2015-09-30 武田薬品工業株式会社 腸溶性錠剤
MA45532A (fr) 2016-07-01 2019-05-08 H Lundbeck As Schémas posologiques de la vortioxétine destinés à une apparition rapide de l'effet antidépresseur
US20200048979A1 (en) 2018-08-13 2020-02-13 Saudi Arabian Oil Company Bottomhole assembly deployment
CN112638526B (zh) * 2018-08-22 2024-01-05 巴斯夫公司 先进的nox还原催化剂
US20210393621A1 (en) 2018-10-26 2021-12-23 The Research Foundation For The State University Of New York Combination serotonin specific reuptake inhibitor and serotonin 1a receptor partial agonist for reducing l-dopa-induced dyskinesia

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WO2007144006A1 (fr) 2007-12-21
CA2656057A1 (fr) 2007-12-21
JP2009539890A (ja) 2009-11-19
PL2044020T3 (pl) 2011-09-30
IL195310A0 (en) 2009-08-03
US20170037006A1 (en) 2017-02-09
NO20090250L (no) 2009-01-16
EP2044020A1 (fr) 2009-04-08
MX2008016008A (es) 2009-01-16
CY1111619T1 (el) 2015-10-07
US20090264465A1 (en) 2009-10-22
EA016054B1 (ru) 2012-01-30
US8299095B2 (en) 2012-10-30
CA2656057C (fr) 2012-10-02
AU2007260356B2 (en) 2013-01-24
HK1134287A1 (en) 2010-04-23
IL195310A (en) 2013-12-31
EA200970019A1 (ru) 2009-08-28
AU2007260356A1 (en) 2007-12-21
US9315459B2 (en) 2016-04-19
US20150073018A1 (en) 2015-03-12
US20130190352A1 (en) 2013-07-25
HRP20110412T1 (hr) 2011-06-30
JP2013216669A (ja) 2013-10-24
JP5318757B2 (ja) 2013-10-16
JP5650280B2 (ja) 2015-01-07

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