NO20084418L - Azolopyridin-3-on derivater som inhibitorer av endoteliallipase - Google Patents

Azolopyridin-3-on derivater som inhibitorer av endoteliallipase

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Publication number
NO20084418L
NO20084418L NO20084418A NO20084418A NO20084418L NO 20084418 L NO20084418 L NO 20084418L NO 20084418 A NO20084418 A NO 20084418A NO 20084418 A NO20084418 A NO 20084418A NO 20084418 L NO20084418 L NO 20084418L
Authority
NO
Norway
Prior art keywords
inhibitors
derivatives
azolopyridin
endothelial lipase
lipase
Prior art date
Application number
NO20084418A
Other languages
English (en)
Inventor
Gerhard Zoller
Stefan Petry
Gunter Muller
Norbert Tennagels
Original Assignee
Sanofi Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38190768&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20084418(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of NO20084418L publication Critical patent/NO20084418L/no

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    • C—CHEMISTRY; METALLURGY
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    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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Abstract

Foreliggende oppfinnelse angår azlopyridin-3-on derivater med generell formel (1) med betydningene indikert i beskrivelsen, dens farmasøytiske anvendelige salter og deres anvendelse som medisinske substanser. Forbindelsene er inhibitorer av endotel lipase.
NO20084418A 2006-03-28 2008-10-21 Azolopyridin-3-on derivater som inhibitorer av endoteliallipase NO20084418L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102006014688A DE102006014688A1 (de) 2006-03-28 2006-03-28 Azolopyridin-3-on-derivate als Inhibitoren von Lipasen und Phospholipasen
PCT/EP2007/002649 WO2007110216A1 (en) 2006-03-28 2007-03-26 Azolopyridin-3-one derivatives as inhibitors of endothelial lipase

Publications (1)

Publication Number Publication Date
NO20084418L true NO20084418L (no) 2008-12-23

Family

ID=38190768

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20084418A NO20084418L (no) 2006-03-28 2008-10-21 Azolopyridin-3-on derivater som inhibitorer av endoteliallipase

Country Status (17)

Country Link
US (1) US8148395B2 (no)
EP (1) EP2001879B1 (no)
JP (1) JP2009531357A (no)
KR (1) KR20080104032A (no)
CN (1) CN101415706A (no)
AR (1) AR060158A1 (no)
AU (1) AU2007229709A1 (no)
BR (1) BRPI0709217A2 (no)
CA (1) CA2647425A1 (no)
DE (1) DE102006014688A1 (no)
MA (1) MA30291B1 (no)
MX (1) MX2008012127A (no)
NO (1) NO20084418L (no)
RU (1) RU2008142535A (no)
TW (1) TW200813049A (no)
WO (1) WO2007110216A1 (no)
ZA (1) ZA200807135B (no)

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RU2008142535A (ru) 2010-05-10
AU2007229709A1 (en) 2007-10-04
EP2001879B1 (en) 2013-08-21
US20090054478A1 (en) 2009-02-26
AR060158A1 (es) 2008-05-28
TW200813049A (en) 2008-03-16
WO2007110216A1 (en) 2007-10-04
EP2001879A1 (en) 2008-12-17
BRPI0709217A2 (pt) 2011-07-12
CA2647425A1 (en) 2007-10-04
MX2008012127A (es) 2008-10-03
JP2009531357A (ja) 2009-09-03
ZA200807135B (en) 2009-05-27
US8148395B2 (en) 2012-04-03
KR20080104032A (ko) 2008-11-28
CN101415706A (zh) 2009-04-22
MA30291B1 (fr) 2009-03-02
DE102006014688A1 (de) 2007-10-04

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