MA30917B1 - Procede pour la sulfinylation d'un derive du pyrazole - Google Patents

Procede pour la sulfinylation d'un derive du pyrazole

Info

Publication number
MA30917B1
MA30917B1 MA31913A MA31913A MA30917B1 MA 30917 B1 MA30917 B1 MA 30917B1 MA 31913 A MA31913 A MA 31913A MA 31913 A MA31913 A MA 31913A MA 30917 B1 MA30917 B1 MA 30917B1
Authority
MA
Morocco
Prior art keywords
acid
sulfinylation
amino
alkaline
pyrazole derivative
Prior art date
Application number
MA31913A
Other languages
English (en)
Inventor
Martin Sukopp
Oliver Kuhn
Carsten Groening
Michael Keil
Jon J Longlet
Original Assignee
Basf Se
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Basf Se filed Critical Basf Se
Publication of MA30917B1 publication Critical patent/MA30917B1/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/44—Oxygen and nitrogen or sulfur and nitrogen atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Communicable Diseases (AREA)
  • Wood Science & Technology (AREA)
  • Oncology (AREA)
  • Epidemiology (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Catalysts (AREA)

Abstract

LA PRÉSENTE INVENTION CONCERNE UN PROCÉDÉ DE SULFINYLATION D'UN DÉRIVÉ PYRAZOLE, CARACTÉRISÉ EN CE QU'ON FAIT RÉAGIR UN 5-AMINO-1-[2,6-DICHLORO-4-(TRIFLUOROMÉTHYL)PHÉNYL]-1H-PYRAZOLE-3- CARBONITRILE (II) AVEC UN AGENT DE SULFINYLATION CHOISI PARMI L'ACIDE TRIFLUOROMÉTHYLSULFINIQUE, L'ANHYDRIDE D'ACIDE TRIFLUOROMÉTHYLSULFINIQUE ET UN SEL DE MÉTAL ALCALIN OU ALCALINO-TERREUX DE TRIFLUOROMÉTHYLSULFINATE AINSI QUE DES MÉLANGES DE L'ACIDE ET/OU DU OU DES SELS, EN PRÉSENCE D'AU MOINS UN COMPLEXE D'ACIDES AMINÉS, LA OU LES AMINES ÉTANT CHOISIES PARMI DES AMINES TERTIAIRES, LE OU LES ACIDES ÉTANT CHOISIS PARMI L'ACIDE FLUORHYDRIQUE, CHLORHYDRIQUE, BROMHYDRIQUE ET IODHYDRIQUE ET DES DÉRIVÉS D'ACIDE SULFONIQUE. LEDIT PROCÉDÉ CONSISTE EN OUTRE À AJOUTER UN AGENT HALOGÉNANT.
MA31913A 2006-11-10 2009-05-25 Procede pour la sulfinylation d'un derive du pyrazole MA30917B1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US86517806P 2006-11-10 2006-11-10
US91361707P 2007-04-24 2007-04-24

Publications (1)

Publication Number Publication Date
MA30917B1 true MA30917B1 (fr) 2009-11-02

Family

ID=39167843

Family Applications (1)

Application Number Title Priority Date Filing Date
MA31913A MA30917B1 (fr) 2006-11-10 2009-05-25 Procede pour la sulfinylation d'un derive du pyrazole

Country Status (22)

Country Link
US (2) US8263783B2 (fr)
EP (1) EP2081908B1 (fr)
JP (1) JP5450077B2 (fr)
KR (1) KR20090083453A (fr)
CN (1) CN102746233A (fr)
AR (1) AR063646A1 (fr)
AU (1) AU2007316718B2 (fr)
BR (1) BRPI0718774A2 (fr)
CA (1) CA2667559A1 (fr)
DK (1) DK2081908T3 (fr)
EA (1) EA200900629A1 (fr)
ES (1) ES2422296T3 (fr)
HR (1) HRP20130582T1 (fr)
IL (1) IL198259A (fr)
MA (1) MA30917B1 (fr)
MX (1) MX2009004262A (fr)
NZ (1) NZ576594A (fr)
PL (1) PL2081908T3 (fr)
PT (1) PT2081908E (fr)
TW (1) TWI413498B (fr)
WO (1) WO2008055877A1 (fr)
ZA (1) ZA200903968B (fr)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2007069254A2 (fr) 2005-12-14 2007-06-21 Makhteshim Chemical Works Ltd. Polymorphes et formes amorphes de 5-amino-1-[2,6-dichloro-4-(trifluoromethyl)phenyl]-4-[(trifluoromethyl)sulfinyl]-1h-pyrazole-3-carbonitrile
AU2007316720B2 (en) 2006-11-10 2013-05-09 Basf Se Process for the sulfinylation of a pyrazole derivative
BRPI0919577A2 (pt) * 2008-10-02 2015-12-08 Basf Se processos para purificar e para preparar ácido trifluorometanossulfínico, e, para preparar fipronila.
EP3412658A1 (fr) * 2017-06-09 2018-12-12 Solvay Sa Procédés pour la préparation de dérivés de pyrazole substitués par un soufre
EP3412659A1 (fr) * 2017-06-09 2018-12-12 Solvay Sa Procédé de fabrication de dérivés pyrazole substitués par du soufre
EP3941907A4 (fr) * 2019-03-19 2023-01-04 Gharda Chemicals Limited Procédé de synthèse de fipronil

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2716453B1 (fr) * 1994-02-22 1996-03-29 Rhone Poulenc Agrochimie Procédé de sulfinylation de composés hétérocycliques.
EP0165136B1 (fr) 1984-05-23 1989-03-01 Rhone-Poulenc Chimie Compositions détergentes comprenant des copolymères à base de polyoxyéthylène et de polyoxyalkylène utilisés comme agents antiredéposants , et leur procédé de preparation
GB8713768D0 (en) 1987-06-12 1987-07-15 May & Baker Ltd Compositions of matter
AU728097B2 (en) 1996-08-01 2001-01-04 Rhodia Chimie Process for grafting a substituted difluoromethyle group
JPH11246555A (ja) * 1997-10-31 1999-09-14 Sumitomo Chem Co Ltd フッ素置換ベンゾヘテロ環化合物
WO1999032439A1 (fr) 1997-12-22 1999-07-01 Minnesota Mining And Manufacturing Company Procede de preparation de sulfinates fluores
DE19853560A1 (de) 1998-11-20 2000-05-25 Bayer Ag Verfahren zur Herstellung von 5-Amino-3-(thio)carbamoylpyrazolen
BR9917518B1 (pt) 1999-10-22 2009-08-11 processos para a preparação de pesticidas 1-arilpirazóis e seus intermediários.
JP2001220386A (ja) * 1999-11-30 2001-08-14 Takeda Chem Ind Ltd オキサジアゾリン誘導体の製造方法
JP2002020364A (ja) 2000-07-06 2002-01-23 Konica Corp スルフィン酸ナトリウム、スルフィン酸カリウムの製造方法およびそれらを用いた写真用カプラーの製造方法
EP1331222A1 (fr) * 2002-01-28 2003-07-30 Virbac S.A. Réactifs écologiques et procédé de halogénoalkylsulfinylation de composés organiques
CN1176078C (zh) 2002-03-27 2004-11-17 江苏省农药研究所 带三氟甲基亚磺酰基的吡唑类化合物的亚磺酰化方法
AU2007316720B2 (en) 2006-11-10 2013-05-09 Basf Se Process for the sulfinylation of a pyrazole derivative
EP2084137B1 (fr) 2006-11-10 2013-04-24 BASF Agro B.V., Arnhem (NL), Zürich Branch Procédé de sulfinylation d'un dérivé pyrazole
FR2924115B1 (fr) 2007-11-27 2010-02-26 Rhodia Operations Procede de preparation d'un acide trifluoromethanesulfinique
BRPI0919577A2 (pt) 2008-10-02 2015-12-08 Basf Se processos para purificar e para preparar ácido trifluorometanossulfínico, e, para preparar fipronila.

Also Published As

Publication number Publication date
IL198259A (en) 2013-10-31
US20120309806A1 (en) 2012-12-06
ES2422296T3 (es) 2013-09-10
WO2008055877A1 (fr) 2008-05-15
US20100137395A1 (en) 2010-06-03
KR20090083453A (ko) 2009-08-03
AR063646A1 (es) 2009-02-04
CA2667559A1 (fr) 2008-05-15
NZ576594A (en) 2011-12-22
EP2081908A1 (fr) 2009-07-29
TWI413498B (zh) 2013-11-01
JP2010509271A (ja) 2010-03-25
BRPI0718774A2 (pt) 2013-12-03
HRP20130582T1 (en) 2013-08-31
CN102746233A (zh) 2012-10-24
US8263783B2 (en) 2012-09-11
JP5450077B2 (ja) 2014-03-26
AU2007316718B2 (en) 2013-03-28
PT2081908E (pt) 2013-06-28
PL2081908T3 (pl) 2013-09-30
IL198259A0 (en) 2009-12-24
DK2081908T3 (da) 2013-07-29
TW200829169A (en) 2008-07-16
EA200900629A1 (ru) 2009-10-30
MX2009004262A (es) 2009-05-05
EP2081908B1 (fr) 2013-04-24
ZA200903968B (en) 2012-02-29
AU2007316718A1 (en) 2008-05-15

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