MA33255B1 - Derives de quinazolinedione, leur preparation et leurs diverses applications therapeutiques - Google Patents

Derives de quinazolinedione, leur preparation et leurs diverses applications therapeutiques

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Publication number
MA33255B1
MA33255B1 MA34323A MA34323A MA33255B1 MA 33255 B1 MA33255 B1 MA 33255B1 MA 34323 A MA34323 A MA 34323A MA 34323 A MA34323 A MA 34323A MA 33255 B1 MA33255 B1 MA 33255B1
Authority
MA
Morocco
Prior art keywords
therapeutic applications
preparation
various therapeutic
quinazolinedione derivatives
nervous system
Prior art date
Application number
MA34323A
Other languages
English (en)
Inventor
Annie Clauss
Christophe Glaess
Gilbert Marciniak
Jean-Francois Nave
Bertrand Vivet
Original Assignee
Sanofi Sa
Abu Ghazaleh Intellectual Prop
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=41226702&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MA33255(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Sanofi Sa, Abu Ghazaleh Intellectual Prop filed Critical Sanofi Sa
Publication of MA33255B1 publication Critical patent/MA33255B1/fr

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    • C07D407/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00
    • C07D407/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings
    • C07D407/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
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Abstract

L'invention a pour objet des dérivés de quinazolinedione de formule (I) avec A un atome de soufre ou d'oxygène ou un groupe sulfoxyde ou sulfone, leurs procédés d'obtention et leurs applications thérapeutiques tels que le cancer le diabète, les maladies musculaires, osseuses, cardiovasculaires, du système nerveux central, du système nerveux périphérique entre autres.
MA34323A 2009-04-09 2010-04-07 Derives de quinazolinedione, leur preparation et leurs diverses applications therapeutiques MA33255B1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0901760A FR2944282B1 (fr) 2009-04-09 2009-04-09 Derives de quinazolinedione, leur preparation et leurs diverses applications therapeutiques
PCT/FR2010/050664 WO2010116088A2 (fr) 2009-04-09 2010-04-07 Dérivés de quinazolinedione, leur préparation et leurs diverses applications thérapeutiques

Publications (1)

Publication Number Publication Date
MA33255B1 true MA33255B1 (fr) 2012-05-02

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KR20160105948A (ko) 2010-11-08 2016-09-07 오메로스 코포레이션 Pde7 억제제를 사용한 중독 및 충동-조절 장애의 치료
RS58381B1 (sr) * 2012-05-07 2019-04-30 Omeros Corp Lečenje zavisnosti i poremećaja kontrole impulsa upotrebom pde7 inhibitora
ITMI20130646A1 (it) * 2013-04-19 2014-10-20 Univ Bologna Alma Mater Composti chinazolindionici con attività inibente sulle sirtuine
CN106146413B (zh) * 2015-04-03 2019-01-18 中南大学 2,4-(1h,3h)-喹唑啉二酮衍生物及其合成方法和用途
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CN119768172A (zh) 2022-08-18 2025-04-04 米托迪治愈有限责任公司 具有磷酸二酯酶-7抑制活性的治疗剂在治疗和预防与慢性疲劳、衰竭和/或劳累不耐受有关的疾病中的用途

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WO2010116088A2 (fr) 2010-10-14
UY32556A (es) 2010-11-30
AU2010233594B2 (en) 2016-07-07
SG175130A1 (en) 2011-11-28
IL215609A0 (en) 2011-12-29
MX2011010639A (es) 2012-01-19
JP2012523397A (ja) 2012-10-04
KR20120028872A (ko) 2012-03-23
JP5564101B2 (ja) 2014-07-30
ZA201107363B (en) 2012-12-27
BRPI1014904A2 (pt) 2016-04-19
AU2010233594A1 (en) 2011-11-03
NZ595768A (en) 2012-12-21
FR2944282B1 (fr) 2013-05-03
CN102459244A (zh) 2012-05-16
FR2944282A1 (fr) 2010-10-15
CN102459244B (zh) 2015-07-08
CL2011002522A1 (es) 2012-02-17
EA021765B1 (ru) 2015-08-31
SG10201401232QA (en) 2014-08-28
CA2758233A1 (fr) 2010-10-14
EP2417130A2 (fr) 2012-02-15
AR076233A1 (es) 2011-05-26
US20120115846A1 (en) 2012-05-10
EA201171228A1 (ru) 2012-05-30
WO2010116088A3 (fr) 2010-12-16
TW201040148A (en) 2010-11-16
CO6440583A2 (es) 2012-05-15
US8722659B2 (en) 2014-05-13

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