MA39421A - Peptides dérivés de l'ezrine et compositions pharmaceutiques correspondantes - Google Patents

Peptides dérivés de l'ezrine et compositions pharmaceutiques correspondantes

Info

Publication number
MA39421A
MA39421A MA039421A MA39421A MA39421A MA 39421 A MA39421 A MA 39421A MA 039421 A MA039421 A MA 039421A MA 39421 A MA39421 A MA 39421A MA 39421 A MA39421 A MA 39421A
Authority
MA
Morocco
Prior art keywords
sub
relates
peptides
gastrointestinal tract
pharmaceutical compositions
Prior art date
Application number
MA039421A
Other languages
English (en)
Inventor
Ravshan Ataullakhanov
Rustam Ataullakhanov
Rupert Holms
Khachik Sayadyan
Original Assignee
Nearmedic International Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Nearmedic International Ltd filed Critical Nearmedic International Ltd
Publication of MA39421A publication Critical patent/MA39421A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K14/00Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/46Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates
    • C07K14/47Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates from mammals
    • C07K14/4701Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates from mammals not used
    • C07K14/4735Villin
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04Linear peptides containing only normal peptide links
    • C07K7/08Linear peptides containing only normal peptide links having 12 to 20 amino acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K39/00Medicinal preparations containing antigens or antibodies
    • A61K39/39Medicinal preparations containing antigens or antibodies characterised by the immunostimulating additives, e.g. chemical adjuvants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/08Peptides having 5 to 11 amino acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/10Peptides having 12 to 20 amino acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/04Immunostimulants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K39/00Medicinal preparations containing antigens or antibodies
    • A61K2039/555Medicinal preparations containing antigens or antibodies characterised by a specific combination antigen/adjuvant
    • A61K2039/55511Organic adjuvants
    • A61K2039/55516Proteins; Peptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K39/00Medicinal preparations containing antigens or antibodies
    • A61K2039/57Medicinal preparations containing antigens or antibodies characterised by the type of response, e.g. Th1, Th2
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K14/00Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/46Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates
    • C07K14/47Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates from mammals
    • C07K14/4701Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates from mammals not used
    • C07K14/4713Autoimmune diseases, e.g. Insulin-dependent diabetes mellitus, multiple sclerosis, rheumathoid arthritis, systemic lupus erythematosus; Autoantigens

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Immunology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Epidemiology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Rheumatology (AREA)
  • Zoology (AREA)
  • Toxicology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Rehabilitation Therapy (AREA)
  • Mycology (AREA)
  • Microbiology (AREA)
  • Pulmonology (AREA)
  • Pain & Pain Management (AREA)
  • Virology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)

Abstract

<!--startfragment-->la présente invention concerne le domaine de la médecine, en particulier le domaine de l'industrie chimique et pharmaceutique et concerne des peptides dérivés de l'ezrine, en particulier un peptide comprenant une séquence d'acides aminés de formule générale (i) x<sub>1</sub> ekkrretvere x<sub>2</sub>x<sub>3</sub>, dans laquelle chaque x représente un résidu d'acide aminé non polaire. L'invention concerne l'utilisation de ces peptides en tant qu'agents immunostimulants et, plus spécifiquement, pour une utilisation dans le traitement et la prévention d'infections antivirales, antibactériennes et antifongiques et le traitement de maladies du tractus gastro-intestinal, en particulier les troubles ulcératifs du tractus gastro-intestinal. La présente invention concerne également des compositions pharmaceutiques comprenant les peptides. En outre, l'invention concerne des procédés de traitement d'une infection et de maladies ulcératives du tractus gastro-intestinal, consistant à administrer les peptides à des patients qui en ont besoin.<!--endfragment-->
MA039421A 2015-06-01 2016-06-01 Peptides dérivés de l'ezrine et compositions pharmaceutiques correspondantes MA39421A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
RU2015120667 2015-06-01

Publications (1)

Publication Number Publication Date
MA39421A true MA39421A (fr) 2017-07-19

Family

ID=56117690

Family Applications (1)

Application Number Title Priority Date Filing Date
MA039421A MA39421A (fr) 2015-06-01 2016-06-01 Peptides dérivés de l'ezrine et compositions pharmaceutiques correspondantes

Country Status (26)

Country Link
US (1) US9682140B2 (fr)
EP (1) EP3191504B1 (fr)
JP (1) JP6721419B2 (fr)
KR (1) KR101842978B1 (fr)
CN (1) CN106188267B (fr)
AU (1) AU2016203656B2 (fr)
CA (1) CA2931875C (fr)
CY (1) CY1120501T1 (fr)
DK (1) DK3191504T3 (fr)
ES (1) ES2660894T3 (fr)
GB (1) GB2546439B (fr)
HR (1) HRP20180560T1 (fr)
HU (1) HUE038737T2 (fr)
LT (1) LT3191504T (fr)
MA (1) MA39421A (fr)
MD (1) MD3191504T2 (fr)
ME (1) ME03033B (fr)
MX (1) MX377333B (fr)
PL (1) PL3191504T3 (fr)
PT (1) PT3191504T (fr)
RS (1) RS57067B1 (fr)
SG (1) SG10201604401UA (fr)
SI (1) SI3191504T1 (fr)
SM (1) SMT201800190T1 (fr)
WO (1) WO2016193285A1 (fr)
ZA (1) ZA201603723B (fr)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US11174288B2 (en) 2016-12-06 2021-11-16 Northeastern University Heparin-binding cationic peptide self-assembling peptide amphiphiles useful against drug-resistant bacteria
CN106596977B (zh) * 2017-02-08 2018-06-08 南京医科大学第一附属医院 ezrin在制备哮喘诊断试剂中的应用
WO2021198346A2 (fr) 2020-04-01 2021-10-07 Dr. Nesselhut Besitzgesellschaft Mbh Peptide ezrine 1 destiné à être utilisé dans un procédé de traitement de la covid-19
EP4125996B1 (fr) * 2020-04-01 2024-08-28 Pantapharm AG Peptide ezrine 1 destiné à être utilisé dans un procédé de traitement de la covid-19
AU2022247001A1 (en) 2021-03-31 2023-10-05 Pantapharm Ag Ezrin peptide 1 for use in a method of treating post covid-19

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2290293A (en) 1994-06-08 1995-12-20 Rupert Donald Holms Preparation which inhibits the autoimmune response in HIV, or SLE, patients
GB2354241A (en) * 1999-09-17 2001-03-21 Rupert Donald Holms Regulatory/unfolding peptides of ezrin
GB0301879D0 (en) 2003-01-27 2003-02-26 Regent Res Llp HCV combination therapy
WO2007060440A2 (fr) 2005-11-23 2007-05-31 Regent Research L.L.P. Utilisation de peptides dans une thérapie anti-ulcère

Also Published As

Publication number Publication date
WO2016193285A1 (fr) 2016-12-08
ME03033B (fr) 2018-10-20
GB2546439B (en) 2020-08-26
JP6721419B2 (ja) 2020-07-15
JP2017025055A (ja) 2017-02-02
CA2931875A1 (fr) 2016-12-01
MX2016007122A (es) 2017-01-25
US9682140B2 (en) 2017-06-20
PL3191504T3 (pl) 2018-08-31
ES2660894T3 (es) 2018-03-26
EP3191504B1 (fr) 2018-01-17
GB201705990D0 (en) 2017-05-31
ZA201603723B (en) 2019-03-27
SG10201604401UA (en) 2017-01-27
HRP20180560T1 (hr) 2018-05-04
DK3191504T3 (en) 2018-04-30
CN106188267A (zh) 2016-12-07
EP3191504A1 (fr) 2017-07-19
MX377333B (es) 2025-03-06
MD3191504T2 (ro) 2018-04-30
CN106188267B (zh) 2020-11-06
RS57067B1 (sr) 2018-06-29
US20160346383A1 (en) 2016-12-01
SMT201800190T1 (it) 2018-05-02
NZ720748A (en) 2023-09-29
AU2016203656B2 (en) 2020-02-06
SI3191504T1 (en) 2018-04-30
CA2931875C (fr) 2022-06-21
GB2546439A (en) 2017-07-19
LT3191504T (lt) 2018-04-10
BR102016012501A2 (pt) 2020-04-28
HUE038737T2 (hu) 2018-11-28
AU2016203656A1 (en) 2016-12-15
KR101842978B1 (ko) 2018-03-29
KR20160141673A (ko) 2016-12-09
CY1120501T1 (el) 2019-07-10
PT3191504T (pt) 2018-04-16

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