MA47692A - Inhibiteurs de l'intégrine (alpha-v) (bêta-6) - Google Patents

Inhibiteurs de l'intégrine (alpha-v) (bêta-6)

Info

Publication number
MA47692A
MA47692A MA047692A MA47692A MA47692A MA 47692 A MA47692 A MA 47692A MA 047692 A MA047692 A MA 047692A MA 47692 A MA47692 A MA 47692A MA 47692 A MA47692 A MA 47692A
Authority
MA
Morocco
Prior art keywords
integrin
inhibitors
beta
alpha
Prior art date
Application number
MA047692A
Other languages
English (en)
Inventor
Matthew Gregory Bursavich
Aleksey Lgorevich Gerasyuto
Kristopher Neil Hahn
Bryce Alden Harrison
Kyle David Konze
fu-yang Lin
Blaise Scott Lippa
Alexey Alexandrovich Lugovskoy
Bruce Nelsen Rogers
Mats Ake Svensson
Dawn Marie Troast
Original Assignee
Morphic Therapeutic Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Morphic Therapeutic Inc filed Critical Morphic Therapeutic Inc
Publication of MA47692A publication Critical patent/MA47692A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
MA047692A 2017-02-28 2018-02-27 Inhibiteurs de l'intégrine (alpha-v) (bêta-6) MA47692A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201762465047P 2017-02-28 2017-02-28

Publications (1)

Publication Number Publication Date
MA47692A true MA47692A (fr) 2020-01-08

Family

ID=63371319

Family Applications (2)

Application Number Title Priority Date Filing Date
MA047692A MA47692A (fr) 2017-02-28 2018-02-27 Inhibiteurs de l'intégrine (alpha-v) (bêta-6)
MA052117A MA52117A (fr) 2017-02-28 2018-02-27 Inhibiteurs de l'intégrine (alpha-v) (bêta-6)

Family Applications After (1)

Application Number Title Priority Date Filing Date
MA052117A MA52117A (fr) 2017-02-28 2018-02-27 Inhibiteurs de l'intégrine (alpha-v) (bêta-6)

Country Status (6)

Country Link
US (4) US11046685B2 (fr)
EP (3) EP3760202A1 (fr)
AU (3) AU2018227417B2 (fr)
CA (1) CA3054792A1 (fr)
MA (2) MA47692A (fr)
WO (1) WO2018160522A1 (fr)

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US10604520B2 (en) 2016-09-07 2020-03-31 Pliant Therapeutics, Inc. N-acyl amino acid compounds and methods of use
EP3558303A4 (fr) 2016-12-23 2020-07-29 Pliant Therapeutics, Inc. Composés acides aminés et leurs procédés d'utilisation
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IL316954A (en) 2017-02-28 2025-01-01 Morphic Therapeutic Inc (Alpha-V)(beta-6)integrin inhibitors
EP3760202A1 (fr) 2017-02-28 2021-01-06 Morphic Therapeutic, Inc. Inhibiteurs de l'intégrine (alpha-v) (bêta-6)
DK3761980T3 (da) 2018-03-07 2024-01-29 Pliant Therapeutics Inc Aminosyreforbindelser og fremgangsmåder til anvendelse
TWI841573B (zh) * 2018-06-27 2024-05-11 美商普萊恩醫療公司 具有未分支連接子之胺基酸化合物及使用方法
UY38353A (es) 2018-08-29 2020-03-31 Morphic Therapeutic Inc Inhibición de integrina alfavbeta6
UY38352A (es) 2018-08-29 2020-03-31 Morphic Therapeutic Inc Inhibidores de integrina alfavbeta6
WO2020047208A1 (fr) 2018-08-29 2020-03-05 Morphic Therapeutic, Inc. Inhibiteurs de l'intégrine (alpha-v)(bêta-6)
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JP7189369B2 (ja) 2018-10-30 2022-12-13 ギリアード サイエンシーズ, インコーポレイテッド アルファ4β7インテグリンの阻害のための化合物
CN112996786B (zh) 2018-10-30 2024-08-20 吉利德科学公司 用于抑制α4β7整合素的化合物
EP3873900B1 (fr) 2018-10-30 2025-01-08 Gilead Sciences, Inc. Dérivés de imidazo[1,2-a]pyridine en tant qu'inhibiteurs d'integrin alpha4beta7 pour le traitement de maladies inflammatoires
WO2020210404A1 (fr) 2019-04-08 2020-10-15 Pliant Therapeutics, Inc. Formes posologiques et schémas de traitement pour des composés d'acides aminés
JP7491996B2 (ja) 2019-08-14 2024-05-28 ギリアード サイエンシーズ, インコーポレイテッド α4β7インテグリンの阻害のための化合物
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EP3843728B1 (fr) 2018-08-29 2025-04-30 Morphic Therapeutic, Inc. Inhibiteurs de l'intégrine (alpha-v)(bêta -6)
UY38353A (es) 2018-08-29 2020-03-31 Morphic Therapeutic Inc Inhibición de integrina alfavbeta6
UY38352A (es) 2018-08-29 2020-03-31 Morphic Therapeutic Inc Inhibidores de integrina alfavbeta6
TW202028179A (zh) 2018-10-08 2020-08-01 美商普萊恩醫療公司 胺基酸化合物及使用方法
WO2020210404A1 (fr) 2019-04-08 2020-10-15 Pliant Therapeutics, Inc. Formes posologiques et schémas de traitement pour des composés d'acides aminés

Also Published As

Publication number Publication date
AU2018227417A1 (en) 2019-09-19
EP4147698A1 (fr) 2023-03-15
US12145935B2 (en) 2024-11-19
EP3589285A4 (fr) 2020-08-12
AU2022201929B2 (en) 2024-03-21
US20250223289A1 (en) 2025-07-10
EP3760202A1 (fr) 2021-01-06
MA52117A (fr) 2022-04-06
WO2018160522A1 (fr) 2018-09-07
AU2024202105B2 (en) 2026-01-29
US11795167B2 (en) 2023-10-24
AU2018227417B2 (en) 2021-12-23
US11046685B2 (en) 2021-06-29
US20200002334A1 (en) 2020-01-02
EP3589285A1 (fr) 2020-01-08
AU2022201929A1 (en) 2022-04-14
CA3054792A1 (fr) 2018-09-07
US20210284640A1 (en) 2021-09-16
AU2024202105A1 (en) 2024-05-02
US20240116929A1 (en) 2024-04-11

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