MA49140A - Composés hétéroaromatiques-aniline fusionnés pour le traitement de troubles dermiques - Google Patents

Composés hétéroaromatiques-aniline fusionnés pour le traitement de troubles dermiques

Info

Publication number
MA49140A
MA49140A MA049140A MA49140A MA49140A MA 49140 A MA49140 A MA 49140A MA 049140 A MA049140 A MA 049140A MA 49140 A MA49140 A MA 49140A MA 49140 A MA49140 A MA 49140A
Authority
MA
Morocco
Prior art keywords
heteroaromatic
merged
treatment
aniline compounds
dermal disorders
Prior art date
Application number
MA049140A
Other languages
English (en)
Inventor
Matthew Duncton
John Kincaid
Original Assignee
Nflection Therapeutics Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Nflection Therapeutics Inc filed Critical Nflection Therapeutics Inc
Publication of MA49140A publication Critical patent/MA49140A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4355Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having oxygen as a ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4365Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system having sulfur as a ring hetero atom, e.g. ticlopidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Dermatology (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pyridine Compounds (AREA)
MA049140A 2017-05-19 2018-05-18 Composés hétéroaromatiques-aniline fusionnés pour le traitement de troubles dermiques MA49140A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201762508997P 2017-05-19 2017-05-19

Publications (1)

Publication Number Publication Date
MA49140A true MA49140A (fr) 2020-03-25

Family

ID=62620965

Family Applications (1)

Application Number Title Priority Date Filing Date
MA049140A MA49140A (fr) 2017-05-19 2018-05-18 Composés hétéroaromatiques-aniline fusionnés pour le traitement de troubles dermiques

Country Status (13)

Country Link
US (2) US10988483B2 (fr)
EP (1) EP3624795B1 (fr)
JP (1) JP7237941B2 (fr)
KR (1) KR102659322B1 (fr)
CN (1) CN111093658B (fr)
AU (1) AU2018270292B2 (fr)
CA (1) CA3063535A1 (fr)
DK (1) DK3624795T3 (fr)
ES (1) ES2913213T3 (fr)
IL (1) IL270576B (fr)
MA (1) MA49140A (fr)
MX (1) MX2019013562A (fr)
WO (1) WO2018213807A1 (fr)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP7237941B2 (ja) * 2017-05-19 2023-03-13 エヌフレクション セラピューティクス インコーポレイテッド 皮膚障害の処置用の融合複素環式芳香族アニリン化合物
CA3120351A1 (fr) * 2018-11-20 2020-05-28 Nflection Therapeutics, Inc. Composes aryl-aniline et heteroaryl-aniline pour le traitement de cancers de la peau
WO2020106308A1 (fr) 2018-11-20 2020-05-28 Nflection Therapeutics, Inc. Composés naphthyridinone-aniline destinés au traitement d'affections de la peau
WO2020106306A1 (fr) 2018-11-20 2020-05-28 Nflection Therapeutics, Inc. Composés cyanoaryl-aniline pour le traitement d'affections de la peau
WO2020106305A1 (fr) 2018-11-20 2020-05-28 Nflection Therapeutics, Inc. Composés thiényl-aniline destinés au traitement d'affections de la peau
EP4233834A3 (fr) * 2018-11-20 2023-10-25 NFlection Therapeutics, Inc. Composés d'aryl-aniline et d'hétéroaryl-aniline pour le traitement de marques de naissance

Family Cites Families (53)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3536809A (en) 1969-02-17 1970-10-27 Alza Corp Medication method
US3598123A (en) 1969-04-01 1971-08-10 Alza Corp Bandage for administering drugs
US3845770A (en) 1972-06-05 1974-11-05 Alza Corp Osmatic dispensing device for releasing beneficial agent
US3916899A (en) 1973-04-25 1975-11-04 Alza Corp Osmotic dispensing device with maximum and minimum sizes for the passageway
US4008719A (en) 1976-02-02 1977-02-22 Alza Corporation Osmotic system having laminar arrangement for programming delivery of active agent
HU196714B (en) 1984-10-04 1989-01-30 Monsanto Co Process for producing non-aqueous composition comprising somatotropin
IE58110B1 (en) 1984-10-30 1993-07-14 Elan Corp Plc Controlled release powder and process for its preparation
US5073543A (en) 1988-07-21 1991-12-17 G. D. Searle & Co. Controlled release formulations of trophic factors in ganglioside-lipsome vehicle
IT1229203B (it) 1989-03-22 1991-07-25 Bioresearch Spa Impiego di acido 5 metiltetraidrofolico, di acido 5 formiltetraidrofolico e dei loro sali farmaceuticamente accettabili per la preparazione di composizioni farmaceutiche in forma a rilascio controllato attive nella terapia dei disturbi mentali organici e composizioni farmaceutiche relative.
PH30995A (en) 1989-07-07 1997-12-23 Novartis Inc Sustained release formulations of water soluble peptides.
US5120548A (en) 1989-11-07 1992-06-09 Merck & Co., Inc. Swelling modulated polymeric drug delivery device
US5733566A (en) 1990-05-15 1998-03-31 Alkermes Controlled Therapeutics Inc. Ii Controlled release of antiparasitic agents in animals
US5580578A (en) 1992-01-27 1996-12-03 Euro-Celtique, S.A. Controlled release formulations coated with aqueous dispersions of acrylic polymers
TW333456B (en) 1992-12-07 1998-06-11 Takeda Pharm Ind Co Ltd A pharmaceutical composition of sustained-release preparation the invention relates to a pharmaceutical composition of sustained-release preparation which comprises a physiologically active peptide.
US5591767A (en) 1993-01-25 1997-01-07 Pharmetrix Corporation Liquid reservoir transdermal patch for the administration of ketorolac
US6087324A (en) 1993-06-24 2000-07-11 Takeda Chemical Industries, Ltd. Sustained-release preparation
IT1270594B (it) 1994-07-07 1997-05-07 Recordati Chem Pharm Composizione farmaceutica a rilascio controllato di moguisteina in sospensione liquida
AU6242096A (en) 1995-06-27 1997-01-30 Takeda Chemical Industries Ltd. Method of producing sustained-release preparation
TW448055B (en) 1995-09-04 2001-08-01 Takeda Chemical Industries Ltd Method of production of sustained-release preparation
JP2909418B2 (ja) 1995-09-18 1999-06-23 株式会社資生堂 薬物の遅延放出型マイクロスフイア
US5980945A (en) 1996-01-16 1999-11-09 Societe De Conseils De Recherches Et D'applications Scientifique S.A. Sustained release drug formulations
US6264970B1 (en) 1996-06-26 2001-07-24 Takeda Chemical Industries, Ltd. Sustained-release preparation
US6419961B1 (en) 1996-08-29 2002-07-16 Takeda Chemical Industries, Ltd. Sustained release microcapsules of a bioactive substance and a biodegradable polymer
CA2217134A1 (fr) 1996-10-09 1998-04-09 Sumitomo Pharmaceuticals Co., Ltd. Formulation a liberation-retard
PT839525E (pt) 1996-10-31 2004-10-29 Takeda Chemical Industries Ltd Preparacao de libertacao prolongada
WO1998027980A2 (fr) 1996-12-20 1998-07-02 Takeda Chemical Industries, Ltd. Procede de production d'une preparation a liberation prolongee
US5891474A (en) 1997-01-29 1999-04-06 Poli Industria Chimica, S.P.A. Time-specific controlled release dosage formulations and method of preparing same
US6613358B2 (en) 1998-03-18 2003-09-02 Theodore W. Randolph Sustained-release composition including amorphous polymer
KR19990085365A (ko) 1998-05-16 1999-12-06 허영섭 지속적으로 약물 조절방출이 가능한 생분해성 고분자 미립구 및그 제조방법
US6248363B1 (en) 1999-11-23 2001-06-19 Lipocine, Inc. Solid carriers for improved delivery of active ingredients in pharmaceutical compositions
US7674907B2 (en) 2004-07-23 2010-03-09 Amgen Inc. Furanopyridine derivatives and methods of use
JP5710855B2 (ja) 2005-02-02 2015-04-30 ネクスジェニクス・ファーマシューティカルズ,リミテッド・ライアビリティ・カンパニー 神経線維腫の局所治療
UA95244C2 (ru) 2005-06-22 2011-07-25 Плексикон, Инк. Соединения и способ модулирования активности киназ, и показания для их применения
GB0601962D0 (en) * 2006-01-31 2006-03-15 Ucb Sa Therapeutic agents
GB0616214D0 (en) 2006-08-15 2006-09-27 Ucb Sa Therapeutic Agents
ES2528797T3 (es) * 2006-08-21 2015-02-12 Genentech, Inc. Compuestos de aza-benzotiofenilo y métodos de uso
AU2007286808B2 (en) * 2006-08-21 2012-12-06 Genentech, Inc. Aza-benzofuranyl compounds and methods of use
EP2089359A2 (fr) 2006-10-31 2009-08-19 Takeda Pharmaceutical Company Limited Inhibiteurs de kinase mapk/erk
PE20081354A1 (es) 2006-11-30 2008-11-14 Genentech Inc Compuestos de azaindolilo como inhibidores de mek
US20080312307A1 (en) 2007-05-25 2008-12-18 Takeda Pharmaceutical Company Limited Mapk/erk kinase inhibitors
GB0714384D0 (en) * 2007-07-23 2007-09-05 Ucb Pharma Sa theraputic agents
CA2708176A1 (fr) 2007-12-21 2009-07-02 Genentech, Inc. Azaindolizines et procedes d'utilisation
EP2240494B1 (fr) 2008-01-21 2016-03-30 UCB Biopharma SPRL Dérivés de thiénopyridine utilisés comme inhibiteurs de mek
GB0801081D0 (en) 2008-01-21 2008-02-27 Ucb Pharma Sa Therapeutic agents
GB0801080D0 (en) 2008-01-21 2008-02-27 Ucb Pharma Sa Therapeutic agents
GB0811304D0 (en) 2008-06-19 2008-07-30 Ucb Pharma Sa Therapeutic agents
JP2010043019A (ja) 2008-08-12 2010-02-25 Taisho Pharmaceutical Co Ltd ピペリジニルピペラジン化合物
AR082453A1 (es) 2010-04-21 2012-12-12 Novartis Ag Compuestos de furopiridina, composiciones farmaceuticas que los contienen y usos de los mismos
WO2012040636A2 (fr) 2010-09-24 2012-03-29 The Broad Institute, Inc. Composés et méthodes de traitement de maladies à médiation par des récepteurs activés par une protéase
WO2014179785A1 (fr) 2013-05-03 2014-11-06 Inscent, Inc. Répulsifs améliorés contre les abeilles domestiques et leurs utilisations
CN105384754B (zh) 2014-09-02 2018-04-20 上海科州药物研发有限公司 作为蛋白激酶抑制剂的杂环类化合物及其制备方法和用途
PT3624796T (pt) 2017-05-19 2025-06-02 Nflection Therapeutics Inc Compostos de pirrolopiridina-anilina para tratamento de distúrbios dérmicos
JP7237941B2 (ja) 2017-05-19 2023-03-13 エヌフレクション セラピューティクス インコーポレイテッド 皮膚障害の処置用の融合複素環式芳香族アニリン化合物

Also Published As

Publication number Publication date
US11542271B2 (en) 2023-01-03
CA3063535A1 (fr) 2018-11-22
US20210380601A1 (en) 2021-12-09
CN111093658B (zh) 2022-10-14
US10988483B2 (en) 2021-04-27
CN111093658A (zh) 2020-05-01
US20200172550A1 (en) 2020-06-04
EP3624795B1 (fr) 2022-04-20
IL270576B (en) 2022-01-01
EP3624795A1 (fr) 2020-03-25
JP7237941B2 (ja) 2023-03-13
WO2018213807A1 (fr) 2018-11-22
JP2020520994A (ja) 2020-07-16
KR20200026812A (ko) 2020-03-11
MX2019013562A (es) 2020-08-03
DK3624795T3 (da) 2022-05-23
ES2913213T3 (es) 2022-06-01
AU2018270292A1 (en) 2019-12-05
KR102659322B1 (ko) 2024-04-22
AU2018270292B2 (en) 2022-02-10

Similar Documents

Publication Publication Date Title
EP3704108A4 (fr) Composés et compositions pour le traitement de troubles hématologiques
MA47719A (fr) Esketamine pour le traitement de la dépression
EP3340982A4 (fr) Composés pour le traitement de troubles immunitaires et inflammatoires
EP3448398A4 (fr) Compositions et méthodes pour le traitement de troubles cutanés
EP3570844A4 (fr) Azolopyrimidine pour le traitement de troubles liés au cancer
EP3013345A4 (fr) Composés pour le traitement d'une amyotrophie spinale
MA45481A (fr) Utilisation d'exosomes pour le traitement de maladies
EP3352749A4 (fr) Composés et compositions pour le traitement de troubles oculaires
EP3411380A4 (fr) Composés destinés au traitement de troubles ou de maladies oculaires
MA49140A (fr) Composés hétéroaromatiques-aniline fusionnés pour le traitement de troubles dermiques
MA44875A (fr) Compositions pour le traitement de troubles acido-basiques
EP3621973A4 (fr) Composés pour la prévention et le traitement de maladies et leur utilisation
EP3328864A4 (fr) Composés et compositions thérapeutiques pour le traitement de troubles sociaux et de troubles liés à la toxicomanie
MA44737A (fr) Compositions pour le traitement de troubles liés à l'hyperkératose
EP3630102A4 (fr) Formulations pour le traitement d'un trouble de stress post-traumatique
EP3774743C0 (fr) Composés de type promédicaments activés par akr1c3 et leur utilisation pour le traitement de troubles hyperprolifératifs
MA51672A (fr) Composés destinés au traitement des troubles kinases-dépendants
MA47212A (fr) Méthodes de traitement de troubles neurologiques
MA51738A (fr) Composés pour le traitement de la douleur
EP3352755A4 (fr) Nouveaux composés, compositions et méthodes pour le traitement de troubles cutanés
MA55218A (fr) Eskétamine pour le traitement de la dépression
EP3621434A4 (fr) Méthodes de traitement de troubles neuropsychiatriques
MA47207A (fr) Composés utiles pour le traitement de troubles du tractus digestif
EP3606542A4 (fr) Protéines pour le traitement de troubles de la fonction barrière épithéliale
MA46099A (fr) Composés pour le traitement de maladies associées à un dysfonctionnement mitochondrial