MA51738A - Composés pour le traitement de la douleur - Google Patents

Composés pour le traitement de la douleur

Info

Publication number
MA51738A
MA51738A MA051738A MA51738A MA51738A MA 51738 A MA51738 A MA 51738A MA 051738 A MA051738 A MA 051738A MA 51738 A MA51738 A MA 51738A MA 51738 A MA51738 A MA 51738A
Authority
MA
Morocco
Prior art keywords
pain
compounds
treatment
Prior art date
Application number
MA051738A
Other languages
English (en)
Inventor
Juan Alvarez
Markus Haeberlein
Demetri Moustakas
Lewis Pennington
Thomas Wynn
Original Assignee
Alkermes Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Alkermes Inc filed Critical Alkermes Inc
Publication of MA51738A publication Critical patent/MA51738A/fr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/439Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D221/00Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/22Bridged ring systems
    • C07D221/26Benzomorphans
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/04Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/04Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D453/00Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pain & Pain Management (AREA)
  • Engineering & Computer Science (AREA)
  • Biomedical Technology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Epidemiology (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Plural Heterocyclic Compounds (AREA)
MA051738A 2018-02-05 2019-02-04 Composés pour le traitement de la douleur MA51738A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201862626499P 2018-02-05 2018-02-05

Publications (1)

Publication Number Publication Date
MA51738A true MA51738A (fr) 2021-05-12

Family

ID=65444375

Family Applications (1)

Application Number Title Priority Date Filing Date
MA051738A MA51738A (fr) 2018-02-05 2019-02-04 Composés pour le traitement de la douleur

Country Status (14)

Country Link
US (3) US10604489B2 (fr)
EP (1) EP3749667A1 (fr)
JP (1) JP2021512952A (fr)
KR (1) KR20200136384A (fr)
CN (1) CN111989327A (fr)
AU (1) AU2019216522A1 (fr)
BR (1) BR112020015712A2 (fr)
CA (1) CA3090385A1 (fr)
EA (1) EA202091881A1 (fr)
IL (1) IL276482A (fr)
MA (1) MA51738A (fr)
MX (1) MX2020008195A (fr)
SG (1) SG11202007422QA (fr)
WO (1) WO2019152946A1 (fr)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR112020015712A2 (pt) * 2018-02-05 2020-12-08 Alkermes, Inc. Compostos para tratamento de dor
WO2021026377A1 (fr) * 2019-08-07 2021-02-11 Alkermes, Inc. Composés contenant du lactame pour le traitement de la douleur
WO2021026378A1 (fr) * 2019-08-07 2021-02-11 Alkermes, Inc. Composés d'indole pour le traitement de la douleur
WO2021026375A1 (fr) * 2019-08-07 2021-02-11 Alkermes, Inc. Composés bicycliques fusionnés pour le traitement de la douleur
WO2021026380A1 (fr) * 2019-08-07 2021-02-11 Alkermes, Inc. Composés de phényltriazole pour le traitement de la douleur
TW202142537A (zh) 2020-02-04 2021-11-16 美商艾爾凱默斯公司 3-((1R,5S,9r)-9-乙氧基-3-氮雜雙環并[3.3.1]壬烷-9-基)—苯甲醯胺之結晶形式及其鹽形式

Family Cites Families (47)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3167562A (en) 1965-01-26 New j-azabicyclo
GB952137A (en) 1961-03-14 1964-03-11 Sankyo Co New 3-azabicyclo [3.3.1] nonane compounds and a process for preparing these compounds
US3196154A (en) 1962-05-17 1965-07-20 Sterling Drug Inc 3-substituted-9-methyl-3, 9-diazabicyclo [3.3.1] nonanes
US3475439A (en) 1966-05-07 1969-10-28 Sankyo Co 3-azabicyclo(3.3.1)nonane compounds
GB1195746A (en) 1967-06-07 1970-06-24 Yoshitomi Pharmaceutical 3-Azabicyclo [3,3,1] Nonane Derivatives
GB1393253A (en) 1971-09-10 1975-05-07 Wyeth John & Brother Ltd 3-azabicyclo-3,3,1-nonanes
JPS4856680A (fr) 1971-11-18 1973-08-09
JPS4961168A (fr) 1972-10-14 1974-06-13
JPS5592384A (en) * 1978-12-30 1980-07-12 Beecham Group Ltd Compound having pharmacological activity
IL59004A0 (en) * 1978-12-30 1980-03-31 Beecham Group Ltd Substituted benzamides their preparation and pharmaceutical compositions containing them
US5244904A (en) 1990-06-05 1993-09-14 Toray Industries, Inc. Indole derivatives
EP0483403A1 (fr) 1990-10-31 1992-05-06 Hoechst Aktiengesellschaft Dérivés d'amino-acides ayant une activité d'inhibitrice de rénine, leur procédé de préparation et les médicaments les contenant
DE4341403A1 (de) 1993-12-04 1995-06-08 Basf Ag N-substituierte 3-Azabicycloalkan-Derivate, ihre Herstellung und Verwendung
US5541217A (en) 1995-05-17 1996-07-30 Ortho Pharmaceutical Corporation 4-arylcyclopenta[c]pyrrole analgesics
JP2808089B2 (ja) 1995-08-29 1998-10-08 レーザーテクノ株式会社 墨出し用レーザー装置
TWI244481B (en) 1998-12-23 2005-12-01 Pfizer 3-azabicyclo[3.1.0]hexane derivatives useful in therapy
DE19952146A1 (de) 1999-10-29 2001-06-07 Boehringer Ingelheim Pharma Arylalkane, Arylalkene und Aryl-azaalkane, diese Verbindungen enthaltende Arzneimittel und Verfahren zu ihrer Herstellung
JP2005522456A (ja) * 2002-02-15 2005-07-28 ファルマシア・アンド・アップジョン・カンパニー・エルエルシー Cns関連障害治療のためのアザビシクロ置換ベンゾイルアミドおよびチオアミド
US7056930B2 (en) 2003-04-14 2006-06-06 Pfizer Inc. 2-Azabicyclo[3.3.1]nonane derivatives
MXPA05011070A (es) * 2003-04-14 2005-12-12 Pfizer Prod Inc Derivados de 3-azabiciclo [3.2.1] octano.
US20050043327A1 (en) * 2003-08-21 2005-02-24 Pfizer Inc Pharmaceutical composition for the prevention and treatment of addiction in a mammal
EP1678172B1 (fr) 2003-10-15 2009-12-09 Targacept, Inc. Compositions pharmaceutiques et methodes destinees au soulagement de la douleur et au traitement de troubles du systeme nerveux central
US7750158B2 (en) 2004-06-22 2010-07-06 Schering Corporation Cannabinoid receptor ligands
WO2007029156A2 (fr) 2005-09-05 2007-03-15 Ranbaxy Laboratories Limited Derives d'isoindoledione comme antagonistes de recepteurs adrenergiques
US7538110B2 (en) 2005-10-27 2009-05-26 Adolor Corporation Opioid antagonists
US7488726B2 (en) 2005-11-03 2009-02-10 Activbiotics Pharma, Llc Rifamycin analogs and uses thereof
MY145633A (en) 2006-03-01 2012-03-15 Theravance Inc 8-azabicyclo[3.2.1]octane compounds as mu opioid receptor antagonists
FR2918986B1 (fr) 2007-07-19 2009-09-04 Sanofi Aventis Sa Derives de 6-cycloamino-3-(pyridazin-4-yl)imidazo[1,2-b]- pyridazine, leur preparation et leur application en therapeutique
TWI423801B (zh) 2007-08-27 2014-01-21 Theravance Inc 作為μ類鴉片受體拮抗劑之8-氮雜雙環〔3.2.1〕辛基-2-羥基苯甲醯胺化合物
US8048895B2 (en) 2008-04-18 2011-11-01 Research Triangle Institute Kappa opioid receptor ligands
GB0815947D0 (en) 2008-09-02 2008-10-08 Univ Dundee Compounds
EP2485735B1 (fr) 2009-10-08 2015-07-29 Merck Sharp & Dohme Corp. Inhibiteurs de protéines de liaison aux acides gras (fabp)
FR2953839A1 (fr) 2009-12-14 2011-06-17 Sanofi Aventis Nouveaux derives d'(heterocycle-piperidine condensee)-(piperazinyl)-1alcanone ou d'(heterocycle-pyrrolidine condensee)-(piperazinyl)-1alcanone et leur utilisation comme inhibiteurs de p75
TW201209054A (en) 2010-05-28 2012-03-01 Prosidion Ltd Novel compounds
US8354420B2 (en) 2010-06-04 2013-01-15 Genentech, Inc. Aminopyrimidine derivatives as LRRK2 inhibitors
WO2012075232A1 (fr) 2010-12-04 2012-06-07 Trevena, Inc. Ligands de récepteurs opioïdes et procédés d'utilisation et de fabrication de ceux-ci
SMT201700325T1 (it) 2011-03-23 2017-09-07 Trevena Inc Ligandi del recettore degli oppioidi e metodi per l’uso e la produzione dei medesimi
JP2014237589A (ja) 2011-09-28 2014-12-18 日本曹達株式会社 環状アミン化合物および有害生物防除剤
GB2498976A (en) 2012-02-01 2013-08-07 Prosidion Ltd GPR119 agonists useful in the treatment of type II diabetes
JP2015083543A (ja) 2012-02-14 2015-04-30 大日本住友製薬株式会社 新規縮環ピロリジン誘導体
EP2716291B1 (fr) * 2012-10-08 2019-11-27 Universität Ulm Combinaison d'opioïdes et médicaments anticancéreux pour le traitement du cancer
WO2014194519A1 (fr) 2013-06-07 2014-12-11 Merck Sharp & Dohme Corp. Dérivés imidazole et leurs procédés d'utilisation pour l'amélioration des propriétés pharmacocinétiques d'un médicament
WO2015091931A1 (fr) 2013-12-20 2015-06-25 AbbVie Deutschland GmbH & Co. KG Dérivés d'oxindole à substituant azétidinyl substitué par pipéridyl, et leur utilisation pour le traitement de maladies liées à la vasopressine
NO2721710T3 (fr) 2014-08-21 2018-03-31
US10683283B2 (en) 2016-09-01 2020-06-16 Mebias Discovery, Inc. Substituted ureas and methods of making and using same
WO2018136546A1 (fr) 2017-01-17 2018-07-26 Mebias Discovery Llc 3-dialkylaminométhyl-pipéridine-4-yl-benzamides substitués et leur procédés de préparation et d'utilisation
BR112020015712A2 (pt) * 2018-02-05 2020-12-08 Alkermes, Inc. Compostos para tratamento de dor

Also Published As

Publication number Publication date
WO2019152946A1 (fr) 2019-08-08
IL276482A (en) 2020-09-30
MX2020008195A (es) 2020-11-24
US11180455B2 (en) 2021-11-23
EP3749667A1 (fr) 2020-12-16
US20220033394A1 (en) 2022-02-03
JP2021512952A (ja) 2021-05-20
CA3090385A1 (fr) 2019-08-08
BR112020015712A2 (pt) 2020-12-08
US10604489B2 (en) 2020-03-31
US20190241524A1 (en) 2019-08-08
AU2019216522A1 (en) 2020-08-27
US20200255383A1 (en) 2020-08-13
EA202091881A1 (ru) 2020-11-10
SG11202007422QA (en) 2020-09-29
CN111989327A (zh) 2020-11-24
KR20200136384A (ko) 2020-12-07

Similar Documents

Publication Publication Date Title
EP3935050A4 (fr) Composés hétérocycliques pour traitement médical
EP3893940A4 (fr) Polythérapie pour le traitement de la dystrophie musculaire
EP3728271A4 (fr) Composés macrocycliques pour le traitement de maladie
EP3968996A4 (fr) Composés triaryles pour le traitement de maladies pd-l1
MA55325A (fr) Composés pour le traitement de maladies pd-l1
EP3704108A4 (fr) Composés et compositions pour le traitement de troubles hématologiques
MA47719A (fr) Esketamine pour le traitement de la dépression
MA44083A (fr) Composés de biarylmonobactame pour le traitement d'infections bactériennes
EP3621973A4 (fr) Composés pour la prévention et le traitement de maladies et leur utilisation
EP3852745A4 (fr) Composés destinés au traitement de certaines leucémies
EP3883554A4 (fr) Composés d'aryl-aniline et d'hétéroaryl-aniline pour le traitement de marques de naissance
EP3317274A4 (fr) Utilisation de composés de chloroquine et de clémizole pour le traitement d'états pathologiques inflammatoires et cancéreux
MA55218A (fr) Eskétamine pour le traitement de la dépression
EP3352749A4 (fr) Composés et compositions pour le traitement de troubles oculaires
MA55143A (fr) Composés aryl-aniline et hétéroaryl-aniline pour le traitement de cancers de la peau
MA51672A (fr) Composés destinés au traitement des troubles kinases-dépendants
EP3898991A4 (fr) Administration périnéale de résinifératoxine pour le traitement de la douleur maladaptative
EP3805216A4 (fr) Composés pour le traitement ou la prévention de maladies hépatiques
MA49140A (fr) Composés hétéroaromatiques-aniline fusionnés pour le traitement de troubles dermiques
EP3877382A4 (fr) Nouveaux composés pour le traitement de maladies respiratoires
SG11202007422QA (en) Compounds for the treatment of pain
EP3373931A4 (fr) Composés hétérocycliques pour le traitement de maladies
EP3413898A4 (fr) Utilisation de tréhalose pour le traitement de maladies neurologiques
MA55141A (fr) Composés cyanoaryl-aniline pour le traitement d'affections de la peau
EP3990458A4 (fr) Composés pour le traitement du cancer