MA50467A - Potentialisateur d'effet antitumoral utilisant un nouveau composé biphényle - Google Patents

Potentialisateur d'effet antitumoral utilisant un nouveau composé biphényle

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Publication number
MA50467A
MA50467A MA050467A MA50467A MA50467A MA 50467 A MA50467 A MA 50467A MA 050467 A MA050467 A MA 050467A MA 50467 A MA50467 A MA 50467A MA 50467 A MA50467 A MA 50467A
Authority
MA
Morocco
Prior art keywords
potentializer
antitumor effect
biphenyl compound
new biphenyl
new
Prior art date
Application number
MA050467A
Other languages
English (en)
Inventor
Akiko Osada
Original Assignee
Taiho Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Taiho Pharmaceutical Co Ltd filed Critical Taiho Pharmaceutical Co Ltd
Publication of MA50467A publication Critical patent/MA50467A/fr

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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/4025—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil not condensed and containing further heterocyclic rings, e.g. cromakalim
    • A—HUMAN NECESSITIES
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/46—8-Azabicyclo [3.2.1] octane; Derivatives thereof, e.g. atropine, cocaine
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    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/20—Carboxylic acids, e.g. valproic acid having a carboxyl group bound to a chain of seven or more carbon atoms, e.g. stearic, palmitic, arachidic acids
    • A61K31/203—Retinoic acids ; Salts thereof
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    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/337—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • A61K31/416—1,2-Diazoles condensed with carbocyclic ring systems, e.g. indazole
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4184—1,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
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RU2765153C2 (ru) 2022-01-26
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TW201900162A (zh) 2019-01-01
JPWO2018216795A1 (ja) 2019-12-26
WO2018216795A1 (fr) 2018-11-29
EP3632443A4 (fr) 2021-01-27
US20210177826A1 (en) 2021-06-17
AU2018272586A1 (en) 2020-01-16
PT3632443T (pt) 2023-08-31
TWI770925B (zh) 2022-07-11
RU2019142111A3 (fr) 2021-06-28
KR102365342B1 (ko) 2022-02-23
EP3632443B1 (fr) 2023-06-07
PL3632443T3 (pl) 2023-09-18
JP6738962B2 (ja) 2020-08-12
TW202137979A (zh) 2021-10-16
US11510915B2 (en) 2022-11-29
RU2019142111A (ru) 2021-06-28
FI3632443T3 (fi) 2023-08-23
KR20200008611A (ko) 2020-01-28
EP3632443A1 (fr) 2020-04-08
AU2018272586B2 (en) 2021-07-29
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