MA51020B1 - Composés imidazopyridiniques et leur utilisation comme médicament - Google Patents
Composés imidazopyridiniques et leur utilisation comme médicamentInfo
- Publication number
- MA51020B1 MA51020B1 MA51020A MA51020A MA51020B1 MA 51020 B1 MA51020 B1 MA 51020B1 MA 51020 A MA51020 A MA 51020A MA 51020 A MA51020 A MA 51020A MA 51020 B1 MA51020 B1 MA 51020B1
- Authority
- MA
- Morocco
- Prior art keywords
- medicine
- imidazopyridine compounds
- nr2b
- therapy
- prevention
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/07—Optical isomers
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Epidemiology (AREA)
- Pain & Pain Management (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Medicines Containing Plant Substances (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pyrrole Compounds (AREA)
- Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
- Pyrane Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
La présente invention concerne de nouveaux imidazopyridines de formule générale a, leurs procédés de préparation, des compositions pharmaceutiques les contenant et leur utilisation en thérapie, en particulier dans le traitement ou la prévention d'affections associées à des propriétés de modulation allostériques négatives de nr2b.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP17206152 | 2017-12-08 | ||
| PCT/EP2018/083728 WO2019110703A1 (fr) | 2017-12-08 | 2018-12-06 | Dérivés d'imidazopyridine et leur utilisation en tant que médicament |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| MA51020A MA51020A (fr) | 2021-05-26 |
| MA51020B1 true MA51020B1 (fr) | 2021-10-29 |
Family
ID=60629568
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MA51020A MA51020B1 (fr) | 2017-12-08 | 2018-12-06 | Composés imidazopyridiniques et leur utilisation comme médicament |
Country Status (34)
| Country | Link |
|---|---|
| US (1) | US10849907B2 (fr) |
| EP (1) | EP3720855B1 (fr) |
| JP (1) | JP6941235B2 (fr) |
| KR (1) | KR102728343B1 (fr) |
| CN (1) | CN111344291B (fr) |
| AR (1) | AR113923A1 (fr) |
| AU (1) | AU2018379438B2 (fr) |
| BR (1) | BR112020008583A2 (fr) |
| CA (1) | CA3083331A1 (fr) |
| CL (1) | CL2020001402A1 (fr) |
| CO (1) | CO2020006648A2 (fr) |
| CY (1) | CY1124744T1 (fr) |
| DK (1) | DK3720855T3 (fr) |
| EA (1) | EA202091139A1 (fr) |
| ES (1) | ES2897050T3 (fr) |
| HR (1) | HRP20211726T1 (fr) |
| HU (1) | HUE056667T2 (fr) |
| IL (1) | IL274868B2 (fr) |
| LT (1) | LT3720855T (fr) |
| MA (1) | MA51020B1 (fr) |
| MX (1) | MX2020005869A (fr) |
| MY (1) | MY203080A (fr) |
| NZ (1) | NZ763704A (fr) |
| PE (1) | PE20211454A1 (fr) |
| PH (1) | PH12020550785A1 (fr) |
| PL (1) | PL3720855T3 (fr) |
| PT (1) | PT3720855T (fr) |
| RS (1) | RS62517B1 (fr) |
| SA (1) | SA520412155B1 (fr) |
| SG (1) | SG11202005138TA (fr) |
| SI (1) | SI3720855T1 (fr) |
| TW (1) | TWI809014B (fr) |
| UA (1) | UA126247C2 (fr) |
| WO (1) | WO2019110703A1 (fr) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TW202112378A (zh) * | 2019-06-04 | 2021-04-01 | 德商百靈佳殷格翰國際股份有限公司 | 嘌呤衍生物及其作為藥物之用途 |
| CN113906033B (zh) * | 2019-06-04 | 2024-04-02 | 勃林格殷格翰国际有限公司 | 咪唑并吡嗪衍生物及其作为药剂的用途 |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6495561B2 (en) | 1999-10-29 | 2002-12-17 | Merck & Co., Inc. | 2-cyclohexyl imidazopyridine NMDA/NR2B antagonists |
| TWI225488B (en) * | 1999-12-21 | 2004-12-21 | Janssen Pharmaceutica Nv | Derivatives of homopiperidinyl substituted benzimidazole analogues |
| ES2312603T3 (es) | 2001-07-24 | 2009-03-01 | Richter Gedeon Nyrt | Derivados de piperidina como antagonistas del receptor nmda. |
| CA2567935C (fr) * | 2004-05-27 | 2009-10-27 | Pfizer Limited | Derives d'aminopyridine utilises comme agonistes selectifs de la dopamine d3 |
| US20100055071A1 (en) * | 2006-11-21 | 2010-03-04 | Martin Robert Leivers | Anti-Viral Compounds |
| US20110319416A1 (en) | 2009-01-28 | 2011-12-29 | Emory University | Subunit Selective NMDA Receptor Antagonists For The Treatment Of Neurological Conditions |
| ES2599553T3 (es) | 2012-10-18 | 2017-02-02 | F. Hoffmann-La Roche Ag | Derivados de etinilo como moduladores de la actividad del receptor mGluR5 |
| EP3110794A1 (fr) | 2014-02-27 | 2017-01-04 | Merck Patent GmbH | Composés hétérocycliques en tant qu'inhibiteurs du canal nav, et leurs utilisations |
| EP3152213B1 (fr) * | 2014-06-04 | 2018-10-31 | Rugen Holdings (Cayman) Limited | Dérivés de difluoroéthylpyridine en tant qu'antagonistes des récepteurs nmda sélectifs du site nr2b |
| WO2016029146A1 (fr) * | 2014-08-22 | 2016-02-25 | University Of Washington | Inhibiteurs spécifiques de la méthionyl-tarn synthétase |
| AU2015317886A1 (en) * | 2014-09-15 | 2017-03-09 | Rugen Holdings (Cayman) Limited | Pyrrolopyrimidine derivatives as NR2B NMDA receptor antagonists |
-
2018
- 2018-12-06 ES ES18826510T patent/ES2897050T3/es active Active
- 2018-12-06 DK DK18826510.2T patent/DK3720855T3/da active
- 2018-12-06 EA EA202091139A patent/EA202091139A1/ru unknown
- 2018-12-06 MA MA51020A patent/MA51020B1/fr unknown
- 2018-12-06 PL PL18826510T patent/PL3720855T3/pl unknown
- 2018-12-06 MX MX2020005869A patent/MX2020005869A/es unknown
- 2018-12-06 MY MYPI2020002784A patent/MY203080A/en unknown
- 2018-12-06 PH PH1/2020/550785A patent/PH12020550785A1/en unknown
- 2018-12-06 HR HRP20211726TT patent/HRP20211726T1/hr unknown
- 2018-12-06 CA CA3083331A patent/CA3083331A1/fr active Pending
- 2018-12-06 HU HUE18826510A patent/HUE056667T2/hu unknown
- 2018-12-06 PT PT188265102T patent/PT3720855T/pt unknown
- 2018-12-06 CN CN201880072962.4A patent/CN111344291B/zh active Active
- 2018-12-06 RS RS20211347A patent/RS62517B1/sr unknown
- 2018-12-06 JP JP2020530609A patent/JP6941235B2/ja active Active
- 2018-12-06 IL IL274868A patent/IL274868B2/en unknown
- 2018-12-06 US US16/211,355 patent/US10849907B2/en active Active
- 2018-12-06 SI SI201830440T patent/SI3720855T1/sl unknown
- 2018-12-06 KR KR1020207019541A patent/KR102728343B1/ko active Active
- 2018-12-06 AU AU2018379438A patent/AU2018379438B2/en active Active
- 2018-12-06 PE PE2020000681A patent/PE20211454A1/es unknown
- 2018-12-06 BR BR112020008583-9A patent/BR112020008583A2/pt unknown
- 2018-12-06 UA UAA202003988A patent/UA126247C2/uk unknown
- 2018-12-06 LT LTEPPCT/EP2018/083728T patent/LT3720855T/lt unknown
- 2018-12-06 SG SG11202005138TA patent/SG11202005138TA/en unknown
- 2018-12-06 WO PCT/EP2018/083728 patent/WO2019110703A1/fr not_active Ceased
- 2018-12-06 NZ NZ763704A patent/NZ763704A/en unknown
- 2018-12-06 EP EP18826510.2A patent/EP3720855B1/fr active Active
- 2018-12-07 AR ARP180103599A patent/AR113923A1/es unknown
- 2018-12-07 TW TW107144026A patent/TWI809014B/zh active
-
2020
- 2020-05-27 CL CL2020001402A patent/CL2020001402A1/es unknown
- 2020-05-29 CO CONC2020/0006648A patent/CO2020006648A2/es unknown
- 2020-06-08 SA SA520412155A patent/SA520412155B1/ar unknown
-
2021
- 2021-11-16 CY CY20211100993T patent/CY1124744T1/el unknown
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