MA52896A - Composés inhibiteurs de vmat2, compositions et méthodes associées - Google Patents

Composés inhibiteurs de vmat2, compositions et méthodes associées

Info

Publication number
MA52896A
MA52896A MA052896A MA52896A MA52896A MA 52896 A MA52896 A MA 52896A MA 052896 A MA052896 A MA 052896A MA 52896 A MA52896 A MA 52896A MA 52896 A MA52896 A MA 52896A
Authority
MA
Morocco
Prior art keywords
methods
inhibitor compounds
vmat2 inhibitor
associated compositions
compositions
Prior art date
Application number
MA052896A
Other languages
English (en)
Inventor
Nicole Harriott
Christopher F O'brien
Original Assignee
Neurocrine Biosciences Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Neurocrine Biosciences Inc filed Critical Neurocrine Biosciences Inc
Publication of MA52896A publication Critical patent/MA52896A/fr

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4738—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4745—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems condensed with ring systems having nitrogen as a ring hetero atom, e.g. phenantrolines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Neurosurgery (AREA)
  • General Chemical & Material Sciences (AREA)
  • Psychiatry (AREA)
  • Neurology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)
MA052896A 2018-06-14 2019-06-13 Composés inhibiteurs de vmat2, compositions et méthodes associées MA52896A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201862684935P 2018-06-14 2018-06-14

Publications (1)

Publication Number Publication Date
MA52896A true MA52896A (fr) 2021-04-21

Family

ID=67263041

Family Applications (1)

Application Number Title Priority Date Filing Date
MA052896A MA52896A (fr) 2018-06-14 2019-06-13 Composés inhibiteurs de vmat2, compositions et méthodes associées

Country Status (16)

Country Link
EP (2) EP3806856A1 (fr)
JP (2) JP2021528386A (fr)
KR (1) KR20210021006A (fr)
CN (1) CN112638387A (fr)
AU (1) AU2019287524A1 (fr)
BR (1) BR112020024018A2 (fr)
CA (1) CA3100694A1 (fr)
EA (1) EA202092750A1 (fr)
IL (1) IL278758A (fr)
JO (1) JOP20200298A1 (fr)
MA (1) MA52896A (fr)
MX (1) MX2020013004A (fr)
PH (1) PH12020552088A1 (fr)
SG (1) SG11202011544UA (fr)
TW (1) TW202011963A (fr)
WO (1) WO2019241555A1 (fr)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL284874B2 (en) 2015-10-30 2023-10-01 Neurocrine Biosciences Inc Valbenazine salts and polymorphs thereof
LT3394057T (lt) 2015-12-23 2022-06-27 Neurocrine Biosciences, Inc. Sintezės būdas, skirtas pagaminti (s)-(2r,3r,11br)-3-izobutil-9,10-dimetoksi-2,3,4,6,7,11b-heksahidro-1h-pirido[2,1-a]izochinolin-2-ilo 2-amino-3-metilbutanoato di(4-metilbenzensulfonatą)
KR20230169457A (ko) 2017-01-27 2023-12-15 뉴로크린 바이오사이언시즈 인코퍼레이티드 특정 vmat2 억제제의 투여 방법
RS66714B1 (sr) 2017-09-21 2025-05-30 Neurocrine Biosciences Inc Formulacija visoke doze valbenazina i sastavi, postupci i kompleti povezani sa njim
MX2020003421A (es) 2017-10-10 2020-07-20 Neurocrine Biosciences Inc Metodos para la administracion de ciertos inhibidores del transportador vesicular de monoamina 2 (vmat2).
KR20250070134A (ko) 2017-10-10 2025-05-20 뉴로크린 바이오사이언시즈 인코퍼레이티드 특정 vmat2 억제제의 투여 방법
DK3784237T3 (da) 2018-04-25 2024-01-08 Shinkei Therapeutics Inc Indretning til transdermal levering af tetrabenazin
MA53239A (fr) 2018-08-15 2022-05-04 Neurocrine Biosciences Inc Procédés d'administration de certains inhibiteurs de vmat2
US10940141B1 (en) 2019-08-23 2021-03-09 Neurocrine Biosciences, Inc. Methods for the administration of certain VMAT2 inhibitors
US20250000805A1 (en) * 2021-10-29 2025-01-02 Neurocrine Biosciences, Inc. Valbenazine compositions

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JOP20190239A1 (ar) * 2017-04-19 2019-10-09 Neurocrine Biosciences Inc مركبات مثبطة لـ vmat2 وتركيبات منها
RS66714B1 (sr) * 2017-09-21 2025-05-30 Neurocrine Biosciences Inc Formulacija visoke doze valbenazina i sastavi, postupci i kompleti povezani sa njim

Also Published As

Publication number Publication date
JP2021528386A (ja) 2021-10-21
SG11202011544UA (en) 2020-12-30
PH12020552088A1 (en) 2021-08-02
EP4691560A3 (fr) 2026-04-15
CN112638387A (zh) 2021-04-09
EA202092750A1 (ru) 2021-05-13
JP2024114905A (ja) 2024-08-23
EP4691560A2 (fr) 2026-02-11
MX2020013004A (es) 2021-02-17
KR20210021006A (ko) 2021-02-24
BR112020024018A2 (pt) 2021-02-23
TW202011963A (zh) 2020-04-01
WO2019241555A1 (fr) 2019-12-19
CA3100694A1 (fr) 2019-12-19
JOP20200298A1 (ar) 2020-11-22
AU2019287524A1 (en) 2020-12-24
EP3806856A1 (fr) 2021-04-21
IL278758A (en) 2021-01-31

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