MD2861F1 - (µ-Imidazol-N, N?) - bis {4-bromo-2- [2- (oxyethylimino) -methyl] -phenolate (2 -) - copper}, which exhibits antifungal activity - Google Patents
(µ-Imidazol-N, N?) - bis {4-bromo-2- [2- (oxyethylimino) -methyl] -phenolate (2 -) - copper}, which exhibits antifungal activity Download PDFInfo
- Publication number
- MD2861F1 MD2861F1 MDA20040233A MD20040233A MD2861F1 MD 2861 F1 MD2861 F1 MD 2861F1 MD A20040233 A MDA20040233 A MD A20040233A MD 20040233 A MD20040233 A MD 20040233A MD 2861 F1 MD2861 F1 MD 2861F1
- Authority
- MD
- Moldova
- Prior art keywords
- copper
- oxyethylimino
- bromo
- bis
- methyl
- Prior art date
Links
- 229910052802 copper Inorganic materials 0.000 title abstract 3
- 239000010949 copper Substances 0.000 title abstract 3
- 230000000843 anti-fungal effect Effects 0.000 title abstract 2
- 229940031826 phenolate Drugs 0.000 title abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 239000003814 drug Substances 0.000 abstract 2
- 240000004808 Saccharomyces cerevisiae Species 0.000 abstract 1
- 230000001857 anti-mycotic effect Effects 0.000 abstract 1
- 230000015572 biosynthetic process Effects 0.000 abstract 1
- 150000001879 copper Chemical class 0.000 abstract 1
- 230000000694 effects Effects 0.000 abstract 1
- 125000002883 imidazolyl group Chemical group 0.000 abstract 1
- 239000003446 ligand Substances 0.000 abstract 1
- 238000003786 synthesis reaction Methods 0.000 abstract 1
- 229910052723 transition metal Inorganic materials 0.000 abstract 1
- 150000003624 transition metals Chemical class 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Inventia se refera la chimia compusilor coordinativi ai metalelor de tranzitie, complecsilor binucleari ai cuprului din clasa salicilideniminoalcoolatilor cu ligand punte de imidazol si anume la (m-imidazol-N,N?)-bis{4-bromo-2-[2-(oxietilimino)-metil]-fenolato(2-)-cupru}, care poate gasi aplicare in medicina sau in medicina veterinara. Esenta inventiei consta in sinteza (m-imidazol-N,N?)-bis{4-bromo-2-[2-(oxietilimino)-metil]-fenolato(2-)-cupru} cu formula : care manifesta activitate antimicotica. Rezultatul inventiei consta in obtinerea unui compus coordinativ nou, care manifesta activitate antimicotica fata de fungii miceliari si levurici, ce depaseste de 1,2...1,5 ori activitatea analogului.The invention relates to the chemistry of the transition metal coordinating compounds, the binuclear copper complexes of the salicylideniminoalcohol class of imidazole bridging ligands, namely (m-imidazole-N, N?) - bis {4-bromo-2- [2- ( oxyethylimino) -methyl] -phenolate (2 -) - copper}, which can be applied in medicine or veterinary medicine. The essence of the invention consists in the synthesis (m-imidazole-N, N?) - bis {4-bromo-2- [2- (oxyethylimino) -methyl] -phenolato (2 -) - copper} of the formula: which exhibits antimycotic activity. The result of the invention consists in obtaining a new coordinating compound, which manifests antifungal activity against mycelial and yeast fungi, which exceeds 1.2 ... 1.5 times the activity of the analog.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| MDA20040233A MD2861G2 (en) | 2004-09-20 | 2004-09-20 | (µ-Imidazole-N,N')-bis{4-bromo-2-[2-(oxyethylimino)-methyl]-phenolato(2-)-copper}, manifesting antimycotic activity |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| MDA20040233A MD2861G2 (en) | 2004-09-20 | 2004-09-20 | (µ-Imidazole-N,N')-bis{4-bromo-2-[2-(oxyethylimino)-methyl]-phenolato(2-)-copper}, manifesting antimycotic activity |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| MD2861F1 true MD2861F1 (en) | 2005-09-30 |
| MD2861G2 MD2861G2 (en) | 2006-04-30 |
Family
ID=35057547
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MDA20040233A MD2861G2 (en) | 2004-09-20 | 2004-09-20 | (µ-Imidazole-N,N')-bis{4-bromo-2-[2-(oxyethylimino)-methyl]-phenolato(2-)-copper}, manifesting antimycotic activity |
Country Status (1)
| Country | Link |
|---|---|
| MD (1) | MD2861G2 (en) |
Cited By (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8575382B2 (en) | 2009-07-13 | 2013-11-05 | “Ivy Pharm” LLC | Low molecular weight pharmacological activity modulators |
| MD4254C1 (en) * | 2012-11-05 | 2014-05-31 | Институт Микробиологии И Биотехнологии Академии Наук Молдовы | Hexafluorotitanate-bis[(dimethylglyoximato)-di-(thiocarbamide)cobalt(III)] dihydrate and process for cultivation of microalga Porphyridium cruentum with the use thereof |
| MD4253C1 (en) * | 2012-11-05 | 2014-05-31 | Институт Микробиологии И Биотехнологии Академии Наук Молдовы | Sulphato-bis(nicotinoylhydrazone)-2,6-diacetylpyridin-cobalt(II )monomethanol trihydrate and process for cultivation of microalga Porphyridium cruentum with the use thereof |
| MD4255C1 (en) * | 2012-11-05 | 2014-05-31 | Институт Микробиологии И Биотехнологии Академии Наук Молдовы | Tetraisothiocyanatocobaltate of bis(nicotinoylhydrazone)-2,6-diformil-4-methylphenol(methanol)(aqua)cobalt(II) and process for cultivation of microalga Porphyridium cruentum with the use thereof |
| MD4258C1 (en) * | 2012-05-31 | 2014-06-30 | Государственный Университет Молд0 | The use of biologically active coordinative compounds of copper(II) with 4-(methoxyphenyl)thiosemicarbazones of 2-benzoylpyridine as inhibitors of Candida albicans |
| MD4303C1 (en) * | 2013-07-05 | 2015-04-30 | Институт Химии Академии Наук Молдовы | Bis(dimethylglyoximato)chloro(isonicotinoylhydrazone-2-hydroxy-1-naphthaldehyde)cobalt(III) and process for cultivation of Porphyridium cruentum microalga with the use thereof |
| MD4326C1 (en) * | 2013-10-22 | 2015-09-30 | Институт Химии Академии Наук Молдовы | N-(D8,13-Bicyclohomofarnesenoylamino)carbazole compound and process for cultivation of Nostoc linckia cyanobacterium with its use |
| MD4327C1 (en) * | 2013-10-22 | 2015-09-30 | Институт Химии Академии Наук Молдовы | N-(D8,13-Bicyclohomofarnesenoyl)-3-amino-1,2,4-triazole compound and process for cultivation of Nostoc linckia cyanobacterium with its use |
| MD4356C1 (en) * | 2014-07-09 | 2016-02-29 | Институт Химии Академии Наук Молдовы | Bis[N'-(2-hydroxy-kO-benzylidene)pyridine-4-carbohydrazidate(-1)-k2N',O]iron(III) nitrate - water (2/3) and process for cultivation of microalga Porphyridium cruentum with its use |
| MD4365C1 (en) * | 2014-07-09 | 2016-03-31 | Институт Химии Академии Наук Молдовы | Bis[1-phenyl-3-methyl-6-(pyridinium-4-yl)-4,5-diaza-hexa-1,3,5-triene-1,6-diolato-O1,N4,O6]iron(III) nitrate and process for cultivation of microalga Porphyridium cruentum with its use |
| MD4367C1 (en) * | 2014-07-09 | 2016-03-31 | Институт Химии Академии Наук Молдовы | Bis[N'-(2-hydroxy-kO-3-carboxybenzilidene)pyridine-3-carbohydrazidate(-1)-k2N',O]iron(III) perchlorate - water (4/5) and process for cultivation of microalga Porphyridium cruentum with its use |
| MD4366C1 (en) * | 2014-07-09 | 2016-03-31 | Институт Химии Академии Наук Молдовы | Bis[1-phenyl-3-methyl-6-(pyridinium-4-il)-4,5-diaza-hexa-1,3,5-triene-1-hydroxy-6-olato-O1,N4,O6]iron(II)sulphate tetrahydrate and process for cultivation of microalga Porphyridium cruentum with its use |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MD3484G2 (en) * | 2007-02-12 | 2008-08-31 | Государственный Университет Молд0 | Di-{µ-[N-(2-hydroxyethyl)-(5-chlorosalicylideneiminato)(-1))]-(O,N,O,Cl)}-bis-(nitrato-imidazolecopper) manifesting antimycotic activity |
| MD4194C1 (en) * | 2012-01-23 | 2013-08-31 | Государственный Университет Молд0 | Trinuclear coordinative compound tris{µ-[3,5-dibromo-2-hydroxybenzylidene-4′-(pyridin-2-yl)-thiosemicarbazido(2-)]copper}hydrate, exhibiting antifungal activity against Candida albicans |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MD2454G2 (en) * | 2003-02-04 | 2004-11-30 | Государственный Университет Молд0 | Nitrate of catene-µ-{2-hydroxymethyl-2-[(2-hydroxy-5-nitrobenzylidene)amino]-propan-1,3-diolo}aquacopper(II) |
-
2004
- 2004-09-20 MD MDA20040233A patent/MD2861G2/en not_active IP Right Cessation
Cited By (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8575382B2 (en) | 2009-07-13 | 2013-11-05 | “Ivy Pharm” LLC | Low molecular weight pharmacological activity modulators |
| MD4258C1 (en) * | 2012-05-31 | 2014-06-30 | Государственный Университет Молд0 | The use of biologically active coordinative compounds of copper(II) with 4-(methoxyphenyl)thiosemicarbazones of 2-benzoylpyridine as inhibitors of Candida albicans |
| MD4254C1 (en) * | 2012-11-05 | 2014-05-31 | Институт Микробиологии И Биотехнологии Академии Наук Молдовы | Hexafluorotitanate-bis[(dimethylglyoximato)-di-(thiocarbamide)cobalt(III)] dihydrate and process for cultivation of microalga Porphyridium cruentum with the use thereof |
| MD4253C1 (en) * | 2012-11-05 | 2014-05-31 | Институт Микробиологии И Биотехнологии Академии Наук Молдовы | Sulphato-bis(nicotinoylhydrazone)-2,6-diacetylpyridin-cobalt(II )monomethanol trihydrate and process for cultivation of microalga Porphyridium cruentum with the use thereof |
| MD4255C1 (en) * | 2012-11-05 | 2014-05-31 | Институт Микробиологии И Биотехнологии Академии Наук Молдовы | Tetraisothiocyanatocobaltate of bis(nicotinoylhydrazone)-2,6-diformil-4-methylphenol(methanol)(aqua)cobalt(II) and process for cultivation of microalga Porphyridium cruentum with the use thereof |
| MD4303C1 (en) * | 2013-07-05 | 2015-04-30 | Институт Химии Академии Наук Молдовы | Bis(dimethylglyoximato)chloro(isonicotinoylhydrazone-2-hydroxy-1-naphthaldehyde)cobalt(III) and process for cultivation of Porphyridium cruentum microalga with the use thereof |
| MD4326C1 (en) * | 2013-10-22 | 2015-09-30 | Институт Химии Академии Наук Молдовы | N-(D8,13-Bicyclohomofarnesenoylamino)carbazole compound and process for cultivation of Nostoc linckia cyanobacterium with its use |
| MD4327C1 (en) * | 2013-10-22 | 2015-09-30 | Институт Химии Академии Наук Молдовы | N-(D8,13-Bicyclohomofarnesenoyl)-3-amino-1,2,4-triazole compound and process for cultivation of Nostoc linckia cyanobacterium with its use |
| MD4356C1 (en) * | 2014-07-09 | 2016-02-29 | Институт Химии Академии Наук Молдовы | Bis[N'-(2-hydroxy-kO-benzylidene)pyridine-4-carbohydrazidate(-1)-k2N',O]iron(III) nitrate - water (2/3) and process for cultivation of microalga Porphyridium cruentum with its use |
| MD4365C1 (en) * | 2014-07-09 | 2016-03-31 | Институт Химии Академии Наук Молдовы | Bis[1-phenyl-3-methyl-6-(pyridinium-4-yl)-4,5-diaza-hexa-1,3,5-triene-1,6-diolato-O1,N4,O6]iron(III) nitrate and process for cultivation of microalga Porphyridium cruentum with its use |
| MD4367C1 (en) * | 2014-07-09 | 2016-03-31 | Институт Химии Академии Наук Молдовы | Bis[N'-(2-hydroxy-kO-3-carboxybenzilidene)pyridine-3-carbohydrazidate(-1)-k2N',O]iron(III) perchlorate - water (4/5) and process for cultivation of microalga Porphyridium cruentum with its use |
| MD4366C1 (en) * | 2014-07-09 | 2016-03-31 | Институт Химии Академии Наук Молдовы | Bis[1-phenyl-3-methyl-6-(pyridinium-4-il)-4,5-diaza-hexa-1,3,5-triene-1-hydroxy-6-olato-O1,N4,O6]iron(II)sulphate tetrahydrate and process for cultivation of microalga Porphyridium cruentum with its use |
Also Published As
| Publication number | Publication date |
|---|---|
| MD2861G2 (en) | 2006-04-30 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| MD2861F1 (en) | (µ-Imidazol-N, N?) - bis {4-bromo-2- [2- (oxyethylimino) -methyl] -phenolate (2 -) - copper}, which exhibits antifungal activity | |
| Pugh et al. | Metal complexes with ‘pincer’-type ligands incorporating N-heterocyclic carbene functionalities | |
| ATE553111T1 (en) | METAL COMPLEXES OF IMIDAZOÄ1,2-FÜPHENANTHRIDINE LIGANDS AND THEIR USE IN OLED DEVICES | |
| TW200606421A (en) | Mediator-modified redox biomolecules for use in electrochemical determination of analyte | |
| DE60305500D1 (en) | CATALYSTS WITH LATE TRANSITION METALS FOR OLEFIN POLYMERIZATION AND OLIGOMERIZATION | |
| MX2008010070A (en) | USE OF COMPLEX METAL COMPOUNDS AS OXIDATION CATALYSTS. | |
| WO2007130306A3 (en) | Ortho-metallated hafnium complexes of imidazole ligands | |
| Wojcicki | Allenyls and propargyls: versatile ligands in transition-metal chemistry | |
| WO2007105052A3 (en) | Multiple-metal complex-containing compound and metal complex, and manufacture methods therefor, and exhaust gas purification catalyst manufacture method using the same | |
| TN2010000102A1 (en) | Novel fungicides | |
| WO2007130307A3 (en) | Improved hafnium complexes of heterocyclic organic ligands | |
| MD4194B1 (en) | Trinuclear coordinative compound tris{µ-¢3,5-dibromo-2-hydroxybenzylidene-4′-(pyridin-2-yl)-thiosemicarbazido(2-)]copper}hydrate, exhibiting antifungal activity against Candida albicans | |
| EP1840130A4 (en) | METAL COMPLEX COMPRISING A TRIDENTATE LIGAND AND A POLYMERIZATION CATALYST COMPRISING SAME | |
| EP2305275A4 (en) | LIQUID COMPOSITION COMPRISING A COORDINATION COMPOUND OF CISPLATIN | |
| NZ592400A (en) | Transition metal complexes of bis[thiohydrazide amide] compounds | |
| PL1660457T3 (en) | Ionic liquids based on imidazolium salts incorporating a nitrile functionality | |
| PL374113A1 (en) | Use of transition metal complexes with nitrogen-containing polydentate ligands as a bleaching catalyst and bleaching agent composition | |
| WO2004085497A3 (en) | Catalyst composition | |
| WO2009068000A3 (en) | CYCLOPENTADIENYLPHOSPHAZENE COMPLEXES (CpPN COMPLEXES) OF METALS OF THE THIRD AND FOURTH GROUP AND OF THE LANTHANOIDS | |
| MD3484F1 (en) | Di- {µ- [N- (2-hydroxyethyl) - (5-chlorosalicylideneiminate (-1))] - (O, N, O, Cl} -bis- (nitrate-imidazole) exhibiting antifungal activity | |
| EP4050013A4 (en) | LIGAND COMPOUND, TRANSITION METAL COMPOUND AND CATALYST COMPOSITION COMPRISING THEM | |
| Tamgho et al. | The synthesis of a silver hexagon using a diiminoisoindoline-based ligand | |
| PL3872157T3 (en) | Dishwashing compositions containing metal complexes | |
| Riis-Johannessen et al. | Solution and solid-state complexes of the potentially tetradentate pyridyl-thiazole ligand 6, 6′-bis (4-methylthiazol-2-yl)-2, 2′-bipyridine with CoII, NiII, CuII, CdII, HgII, CuI and AgI | |
| MX357104B (en) | Ziegler-natta catalyst systems and polymers formed therefrom. |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| KA4A | Patent for invention lapsed due to non-payment of fees (with right of restoration) | ||
| MM4A | Patent for invention definitely lapsed due to non-payment of fees |