MX2014008190A - Composiciones de biguanida y métodos para tratar transtornos metabólicos. - Google Patents

Composiciones de biguanida y métodos para tratar transtornos metabólicos.

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Publication number
MX2014008190A
MX2014008190A MX2014008190A MX2014008190A MX2014008190A MX 2014008190 A MX2014008190 A MX 2014008190A MX 2014008190 A MX2014008190 A MX 2014008190A MX 2014008190 A MX2014008190 A MX 2014008190A MX 2014008190 A MX2014008190 A MX 2014008190A
Authority
MX
Mexico
Prior art keywords
methods
metabolic disorders
biguanide
treating metabolic
compositions
Prior art date
Application number
MX2014008190A
Other languages
English (en)
Inventor
Alain D Baron
Nigel R A Beeley
Mark S Fineman
Original Assignee
Elcelyx Therapeutics Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US13/345,135 external-priority patent/US20120177730A1/en
Application filed by Elcelyx Therapeutics Inc filed Critical Elcelyx Therapeutics Inc
Publication of MX2014008190A publication Critical patent/MX2014008190A/es

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    • A61K31/13Amines
    • A61K31/155Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
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    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
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    • A61K31/34Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
    • A61K31/341Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide not condensed with another ring, e.g. ranitidine, furosemide, bufetolol, muscarine
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Abstract

Se proveen en la presente métodos para tratar ciertas condiciones, incluyendo diabetes, obesidad y otras enfermedades, alteraciones o condiciones metabólicas al administrar una composición que comprende una biguanida o compuesto heterocíclico relacionado, por ejemplo metformina. También se proveen en la presente biguanida o composiciones de compuesto heterocíclico relacionadas y métodos para la preparación de los mismos para uso en los métodos de la presente invención. También se proveen en la presente composiciones que comprenden metformina y sales de la misma y métodos de uso.
MX2014008190A 2012-01-06 2012-07-11 Composiciones de biguanida y métodos para tratar transtornos metabólicos. MX2014008190A (es)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US13/345,135 US20120177730A1 (en) 2011-01-07 2012-01-06 Chemosensory Receptor Ligand-Based Therapies
PCT/US2012/020548 WO2012094636A2 (en) 2011-01-07 2012-01-06 Chemosensory receptor ligand-based therapies
US201261649171P 2012-05-18 2012-05-18
PCT/US2012/046335 WO2013103384A1 (en) 2012-01-06 2012-07-11 Biguanide compositions and methods of treating metabolic disorders

Publications (1)

Publication Number Publication Date
MX2014008190A true MX2014008190A (es) 2015-02-04

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Family Applications (2)

Application Number Title Priority Date Filing Date
MX2014008190A MX2014008190A (es) 2012-01-06 2012-07-11 Composiciones de biguanida y métodos para tratar transtornos metabólicos.
MX2020003112A MX2020003112A (es) 2012-01-06 2014-07-02 Composiciones de biguanida y metodos para tratar trastornos metabolicos.

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MX2020003112A MX2020003112A (es) 2012-01-06 2014-07-02 Composiciones de biguanida y metodos para tratar trastornos metabolicos.

Country Status (15)

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US (2) US10154972B2 (es)
EP (1) EP2800561B1 (es)
JP (4) JP2015503582A (es)
KR (4) KR20190120430A (es)
CN (2) CN110693868A (es)
AU (2) AU2012363873B2 (es)
BR (1) BR112014016808B1 (es)
CA (1) CA2862533C (es)
EA (1) EA201491335A1 (es)
ES (1) ES2832773T3 (es)
IL (1) IL233506B (es)
MX (2) MX2014008190A (es)
SG (2) SG11201403839SA (es)
WO (1) WO2013103384A1 (es)
ZA (1) ZA201405046B (es)

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* Cited by examiner, † Cited by third party
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US9480663B2 (en) 2011-01-07 2016-11-01 Elcelyx Therapeutics, Inc. Biguanide compositions and methods of treating metabolic disorders
US9572784B2 (en) 2011-01-07 2017-02-21 Elcelyx Therapeutics, Inc. Compositions comprising statins, biguanides and further agents for reducing cardiometabolic risk
EP2661266B1 (en) 2011-01-07 2020-09-16 Anji Pharma (US) LLC Chemosensory receptor ligand-based therapies
US9211263B2 (en) 2012-01-06 2015-12-15 Elcelyx Therapeutics, Inc. Compositions and methods of treating metabolic disorders
US11759441B2 (en) 2011-01-07 2023-09-19 Anji Pharmaceuticals Inc. Biguanide compositions and methods of treating metabolic disorders
US8796338B2 (en) 2011-01-07 2014-08-05 Elcelyx Therapeutics, Inc Biguanide compositions and methods of treating metabolic disorders
US11974971B2 (en) 2011-01-07 2024-05-07 Anji Pharmaceuticals Inc. Compositions and methods for treating metabolic disorders
EP2800562A2 (en) 2012-01-06 2014-11-12 Elcelyx Therapeutics, Inc. Compositions and methods for treating metabolic disorders
KR20190120430A (ko) * 2012-01-06 2019-10-23 엘셀릭스 테라퓨틱스 인코포레이티드 바이구아나이드 조성물 및 대사 장애를 치료하는 방법
US20140010783A1 (en) * 2012-07-06 2014-01-09 Hoffmann-La Roche Inc. Antiviral compounds
KR101994145B1 (ko) * 2013-01-28 2019-07-01 한올바이오파마주식회사 Ν1-고리아민-ν5-치환된 바이구아나이드 유도체를 유효성분으로 함유하는 시차증후군의 예방 또는 치료용 약학 조성물
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