MX2020005775A - Uso farmaceutico de pirfenidona para la reduccion de fibrosis cardiaca en pacientes con cardiomiopatia y/o esteatosis cardiaca y/o covid-19. - Google Patents
Uso farmaceutico de pirfenidona para la reduccion de fibrosis cardiaca en pacientes con cardiomiopatia y/o esteatosis cardiaca y/o covid-19.Info
- Publication number
- MX2020005775A MX2020005775A MX2020005775A MX2020005775A MX2020005775A MX 2020005775 A MX2020005775 A MX 2020005775A MX 2020005775 A MX2020005775 A MX 2020005775A MX 2020005775 A MX2020005775 A MX 2020005775A MX 2020005775 A MX2020005775 A MX 2020005775A
- Authority
- MX
- Mexico
- Prior art keywords
- cardiac
- covid
- pirfenidone
- cardiomyopathy
- pharmaceutical use
- Prior art date
Links
- 208000025721 COVID-19 Diseases 0.000 title abstract 2
- 208000031229 Cardiomyopathies Diseases 0.000 title abstract 2
- 230000000747 cardiac effect Effects 0.000 title abstract 2
- 230000009787 cardiac fibrosis Effects 0.000 title abstract 2
- ISWRGOKTTBVCFA-UHFFFAOYSA-N pirfenidone Chemical compound C1=C(C)C=CC(=O)N1C1=CC=CC=C1 ISWRGOKTTBVCFA-UHFFFAOYSA-N 0.000 title abstract 2
- 229960003073 pirfenidone Drugs 0.000 title abstract 2
- 230000007863 steatosis Effects 0.000 title abstract 2
- 231100000240 steatosis hepatitis Toxicity 0.000 title abstract 2
- 102000013394 Troponin I Human genes 0.000 abstract 1
- 108010065729 Troponin I Proteins 0.000 abstract 1
- 239000004480 active ingredient Substances 0.000 abstract 1
- 230000000975 bioactive effect Effects 0.000 abstract 1
- 229940079593 drug Drugs 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- JUJWROOIHBZHMG-UHFFFAOYSA-N pyridine Substances C1=CC=NC=C1 JUJWROOIHBZHMG-UHFFFAOYSA-N 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4412—Non condensed pyridines; Hydrogenated derivatives thereof having oxo groups directly attached to the heterocyclic ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La presente desarrollada, se encuentra relacionada al campo de los medicamentos que reducen la fibrosis cardíaca y también la expresión de la troponina I , concretamente al uso farmacéutico que contiene 5-metil -1-fenil -2-(1H) -piridona (Pirfenidona) como principio activo solo o en combinación con cualquier otra molécula bioactiva, concretamente para el manejo de pacientes con cardiomiopatía y/o esteatosis cardiaca y/o COVID-19.
Priority Applications (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| MX2020005775A MX2020005775A (es) | 2020-07-13 | 2020-07-13 | Uso farmaceutico de pirfenidona para la reduccion de fibrosis cardiaca en pacientes con cardiomiopatia y/o esteatosis cardiaca y/o covid-19. |
| PCT/MX2021/000019 WO2022015141A1 (es) | 2020-07-13 | 2021-06-03 | Uso farmacéutico de pirfenidona para la reducción de fibrosis cardiaca en pacientes con cardiomiopatía y/o esteatosis cardiaca y/o covid-19 |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| MX2020005775A MX2020005775A (es) | 2020-07-13 | 2020-07-13 | Uso farmaceutico de pirfenidona para la reduccion de fibrosis cardiaca en pacientes con cardiomiopatia y/o esteatosis cardiaca y/o covid-19. |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX2020005775A true MX2020005775A (es) | 2022-01-14 |
Family
ID=79554854
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2020005775A MX2020005775A (es) | 2020-07-13 | 2020-07-13 | Uso farmaceutico de pirfenidona para la reduccion de fibrosis cardiaca en pacientes con cardiomiopatia y/o esteatosis cardiaca y/o covid-19. |
Country Status (2)
| Country | Link |
|---|---|
| MX (1) | MX2020005775A (es) |
| WO (1) | WO2022015141A1 (es) |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH02215719A (ja) * | 1989-02-15 | 1990-08-28 | Yamauchi Akitomo | 線維化病変組織の修復並びに線維化病変の阻止剤 |
| CN109475626A (zh) * | 2016-07-14 | 2019-03-15 | 儿童医院医疗中心 | 治疗纤维化的方法 |
| WO2018164098A1 (ja) * | 2017-03-06 | 2018-09-13 | 国立大学法人大阪大学 | 心臓線維化モデルとして用いられる細胞集団、その製造方法、それを利用したスクリーニング方法及び心臓線維化モデルの評価方法、並びに心臓線維化モデルの評価システム |
| CN111481547A (zh) * | 2020-04-16 | 2020-08-04 | 青岛海洋生物医药研究院股份有限公司 | 哌非尼酮或其药学上可接受的盐在制备预防和/或治疗新型冠状病毒炎症药物中的应用 |
-
2020
- 2020-07-13 MX MX2020005775A patent/MX2020005775A/es unknown
-
2021
- 2021-06-03 WO PCT/MX2021/000019 patent/WO2022015141A1/es not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| WO2022015141A1 (es) | 2022-01-20 |
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