MX23672A - Derivados de glicopeptidos y procedimiento para su preparacion. - Google Patents

Derivados de glicopeptidos y procedimiento para su preparacion.

Info

Publication number
MX23672A
MX23672A MX2367290A MX2367290A MX23672A MX 23672 A MX23672 A MX 23672A MX 2367290 A MX2367290 A MX 2367290A MX 2367290 A MX2367290 A MX 2367290A MX 23672 A MX23672 A MX 23672A
Authority
MX
Mexico
Prior art keywords
glycopeptides
derivatives
procedure
preparation
Prior art date
Application number
MX2367290A
Other languages
English (en)
Inventor
Ramakrishnan Nagarajan
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of MX23672A publication Critical patent/MX23672A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K9/00Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K9/00Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
    • C07K9/006Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure
    • C07K9/008Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure directly attached to a hetero atom of the saccharide radical, e.g. actaplanin, avoparcin, ristomycin, vancomycin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
MX2367290A 1989-12-13 1990-12-10 Derivados de glicopeptidos y procedimiento para su preparacion. MX23672A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US44917189A 1989-12-13 1989-12-13

Publications (1)

Publication Number Publication Date
MX23672A true MX23672A (es) 1993-11-01

Family

ID=23783157

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2367290A MX23672A (es) 1989-12-13 1990-12-10 Derivados de glicopeptidos y procedimiento para su preparacion.

Country Status (20)

Country Link
US (1) US5591714A (es)
EP (1) EP0435503B1 (es)
JP (1) JP3590638B2 (es)
KR (1) KR910011896A (es)
CN (1) CN1034506C (es)
CA (1) CA2031803C (es)
DE (1) DE69033087T2 (es)
ES (1) ES2131496T3 (es)
FI (1) FI906083A7 (es)
HU (1) HUT55802A (es)
IE (1) IE904485A1 (es)
IL (1) IL96603A (es)
MX (1) MX23672A (es)
NO (1) NO303692B1 (es)
NZ (1) NZ236393A (es)
PH (1) PH27373A (es)
PT (1) PT96139B (es)
RU (2) RU2041237C1 (es)
YU (1) YU234790A (es)
ZA (1) ZA909847B (es)

Families Citing this family (45)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5721208A (en) * 1991-06-29 1998-02-24 Hoechst Aktiengesellschaft Glycopeptides a process for their preparation and their use
TW213468B (es) * 1991-06-29 1993-09-21 Hoechst Ag
US5840684A (en) * 1994-01-28 1998-11-24 Eli Lilly And Company Glycopeptide antibiotic derivatives
TW457248B (en) * 1994-01-28 2001-10-01 Lilly Co Eli Glycopeptide antibiotic derivatives
DE19512484A1 (de) * 1995-04-04 1996-10-17 Bayer Ag Kohlenhydratmodifizierte Cytostatika
US5919756A (en) * 1996-06-28 1999-07-06 Eli Lilly And Company Amides
US5939382A (en) * 1996-11-21 1999-08-17 Eli Lilly And Company Reducing agent for reductive alkylation of glycopeptide antibiotics
US5952466A (en) * 1997-11-12 1999-09-14 Eli Lilly And Company Reductive alkylation of glycopeptide antibiotics
ID18900A (id) * 1996-11-21 1998-05-20 Lilly Co Eli Alkilasi menurun dari gliko peptida anti biotik
RU2124022C1 (ru) * 1997-04-10 1998-12-27 Институт биоорганической химии им.М.М.Шемякина и Ю.А.Овчинникова РАН Фуллереновое производное гликопептида, обладающее адъювантной активностью
US5919771A (en) * 1997-05-20 1999-07-06 Eli Lilly And Company Urea and thiourea derivatives of glycopeptides
US5977063A (en) * 1997-05-20 1999-11-02 Eli Lilly And Company Alkylated hexapeptides
US5952310A (en) * 1997-05-20 1999-09-14 Eli Lilly And Company Glycopeptide hexapeptides
US5972933A (en) * 1998-01-08 1999-10-26 Ed. Geistlich Sohne Ag Fur Chemische Industrie Method of treating microbial infections
WO1999056760A1 (en) * 1998-05-01 1999-11-11 Eli Lilly And Company N1-modified glycopeptides
DE69934582T2 (de) 1998-06-11 2007-10-04 Pharmacia & Upjohn Co. Llc, Kalamazoo Delavirdin tablettenformulierung
PT1140993E (pt) * 1998-12-23 2003-10-31 Theravance Inc Derivados de glicopeptidos e composicoes farmaceuticas contendo os mesmos
GB9925127D0 (en) * 1999-10-22 1999-12-22 Pharmacia & Upjohn Spa Oral formulations for anti-tumor compounds
US20020004502A1 (en) * 2000-01-05 2002-01-10 Redmond H. Paul Treatment of inflammatory bowel disease
CA2726789A1 (en) * 2000-02-05 2001-11-08 Theravance, Inc. Cyclodextrin containing glycopeptide antibiotic compositions
CA2399640A1 (en) 2000-02-11 2001-08-16 Eli Lilly And Company Selective n-acylation of a82846 glycopeptide analogs
AU2001259298A1 (en) * 2000-05-02 2001-11-12 Advanced Medicine, Inc. Polyacid glycopeptide derivatives
JP4713810B2 (ja) * 2000-05-02 2011-06-29 セラヴァンス, インコーポレーテッド グリコペプチドに対する還元的アルキル化プロセス
DE60040329D1 (de) * 2000-05-09 2008-11-06 Lucent Technologies Inc Verbesserte Steurung der Dienstequalität in einem mobilen Telekommunikationsnetz
UA75083C2 (uk) * 2000-06-22 2006-03-15 Тераванс, Інк. Похідні глікопептидфосфонатів
ES2302733T3 (es) 2000-06-22 2008-08-01 Theravance, Inc. Derivados carboxi-sacaridos de glucopeptido.
US6872804B2 (en) * 2000-06-22 2005-03-29 Theravance, Inc. Glycopeptide disulfide and thioester derivatives
WO2001098329A1 (en) 2000-06-22 2001-12-27 Theravance, Inc. Polyhydroxy glycopeptide derivatives
TWI312785B (en) * 2001-08-24 2009-08-01 Theravance Inc Process for preparing vancomycin derivatives
TWI275594B (en) 2001-08-24 2007-03-11 Theravance Inc Process for preparing vancomycin phosphonate derivatives
WO2004091578A2 (en) 2003-04-09 2004-10-28 Biodelivery Sciences International, Inc. Novel encochleation methods, cochleates and methods of use
US8778874B2 (en) * 2004-11-29 2014-07-15 National University Corporation Nagoya University Glycopeptide antibiotic monomer derivatives
UA90707C2 (en) 2005-04-06 2010-05-25 Астразенека Аб Novel 5-substituted 7-amino-[1,3]thiazolo[4,5-d]pyrimidine derivatives
AR053347A1 (es) 2005-04-06 2007-05-02 Astrazeneca Ab Derivados de [1,3]tiazolo[4,5-d]pirimidin-2(3h)-ona 5,7-sustituidos
CA2623198C (en) 2005-09-22 2014-08-05 Medivas, Llc Bis-(a-amino)-diol-diester-containing poly(ester amide) and poly(ester urethane) compositions and methods of use
JP5178520B2 (ja) 2005-09-22 2013-04-10 メディバス エルエルシー 固体ポリマー送達組成物およびその使用法
TW200808818A (en) 2006-05-26 2008-02-16 Shionogi & Co Glycopeptide antibiotic derivatives
CN101959900A (zh) * 2007-12-26 2011-01-26 盐野义制药株式会社 糖肽类抗生素糖基化衍生物
EP2260060A4 (en) 2008-04-01 2013-01-16 Univ Cornell ORGANIC SOLUBLE CHITOSA SALT AND CHITOSAN DERIVED BIOMATERIALS MANUFACTURED THEREFROM
CN101928331B (zh) * 2009-06-26 2014-05-28 上海来益生物药物研究开发中心有限责任公司 一种化合物及其应用
EP2704688B1 (en) 2011-05-05 2019-07-10 Matinas BioPharma Nanotechnologies, Inc. Cochleate compositions and methods of making and using same
CN107759672A (zh) * 2013-08-19 2018-03-06 南京爱斯药业有限公司 万古霉素衍生物、制备方法及其应用
AU2014322817A1 (en) 2013-09-23 2016-04-21 Jawaharlal Nehru Centre for Advanced Scientific Research (JNCASR) Vancomycin-sugar conjugates and uses thereof
EP3169345B1 (en) * 2014-07-17 2025-01-29 Melinta Therapeutics, LLC High purity oritavancin and method of producing same
CN108409837B (zh) 2018-03-06 2021-09-24 上海来益生物药物研究开发中心有限责任公司 一组具有抗耐药性细菌活性的糖肽类化合物、其制备方法和应用

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4552701A (en) * 1984-04-16 1985-11-12 Eli Lilly And Company Glycopeptide antibiotics and process of preparation
US4698327A (en) * 1985-04-25 1987-10-06 Eli Lilly And Company Novel glycopeptide derivatives
US4639433A (en) * 1985-08-14 1987-01-27 Eli Lilly And Company Glycopeptide derivatives
US4643987A (en) * 1985-08-14 1987-02-17 Eli Lilly And Company Modified glycopeptides
US4946941A (en) * 1986-01-24 1990-08-07 Shionogi & Co., Ltd. Novel glycopeptide antibiotics
EG18377A (en) * 1986-09-19 1993-04-30 Lilly Co Eli Process for preparing glycopeptide antibiotics
GB8701872D0 (en) * 1987-01-28 1987-03-04 Lepetit Spa N15-alkyl & n15,n15-dialkyl derivatives
US5071749A (en) * 1987-04-16 1991-12-10 Shionogi & Co., Ltd. Glycopetide antibiotic pa-45052-b

Also Published As

Publication number Publication date
AU6796490A (en) 1991-06-20
PT96139B (pt) 1998-04-30
ZA909847B (en) 1992-08-26
CN1034506C (zh) 1997-04-09
ES2131496T3 (es) 1999-08-01
AU633165B2 (en) 1993-01-21
EP0435503A1 (en) 1991-07-03
CA2031803A1 (en) 1991-06-14
IL96603A0 (en) 1991-09-16
JP3590638B2 (ja) 2004-11-17
CA2031803C (en) 2001-05-29
RU2041237C1 (ru) 1995-08-09
US5591714A (en) 1997-01-07
DE69033087D1 (de) 1999-06-10
IL96603A (en) 1998-02-08
HUT55802A (en) 1991-06-28
CN1052483A (zh) 1991-06-26
DE69033087T2 (de) 1999-10-14
RU2053240C1 (ru) 1996-01-27
NZ236393A (en) 1992-05-26
NO303692B1 (no) 1998-08-17
NO905354D0 (no) 1990-12-11
IE904485A1 (en) 1991-06-19
JPH04108800A (ja) 1992-04-09
KR910011896A (ko) 1991-08-07
NO905354L (no) 1991-06-14
FI906083A7 (fi) 1991-06-14
PT96139A (pt) 1991-09-30
EP0435503B1 (en) 1999-05-06
YU234790A (sh) 1992-12-21
FI906083A0 (fi) 1990-12-11
PH27373A (en) 1993-06-21

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