PT96139A - Processo para a preparacao de novos derivados de glicopeptido - Google Patents

Processo para a preparacao de novos derivados de glicopeptido

Info

Publication number
PT96139A
PT96139A PT96139A PT9613990A PT96139A PT 96139 A PT96139 A PT 96139A PT 96139 A PT96139 A PT 96139A PT 9613990 A PT9613990 A PT 9613990A PT 96139 A PT96139 A PT 96139A
Authority
PT
Portugal
Prior art keywords
preparing new
glycopeptide derivatives
new glycopeptide
derivatives
preparing
Prior art date
Application number
PT96139A
Other languages
English (en)
Other versions
PT96139B (pt
Inventor
Ramakrishnan Nagarajan
Amelia Apolinaria Schabel
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of PT96139A publication Critical patent/PT96139A/pt
Publication of PT96139B publication Critical patent/PT96139B/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K9/00Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K9/00Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
    • C07K9/006Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure
    • C07K9/008Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure directly attached to a hetero atom of the saccharide radical, e.g. actaplanin, avoparcin, ristomycin, vancomycin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
PT96139A 1989-12-13 1990-12-10 Processo para a preparacao de novos derivados de glicopeptido PT96139B (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US44917189A 1989-12-13 1989-12-13

Publications (2)

Publication Number Publication Date
PT96139A true PT96139A (pt) 1991-09-30
PT96139B PT96139B (pt) 1998-04-30

Family

ID=23783157

Family Applications (1)

Application Number Title Priority Date Filing Date
PT96139A PT96139B (pt) 1989-12-13 1990-12-10 Processo para a preparacao de novos derivados de glicopeptido

Country Status (20)

Country Link
US (1) US5591714A (pt)
EP (1) EP0435503B1 (pt)
JP (1) JP3590638B2 (pt)
KR (1) KR910011896A (pt)
CN (1) CN1034506C (pt)
CA (1) CA2031803C (pt)
DE (1) DE69033087T2 (pt)
ES (1) ES2131496T3 (pt)
FI (1) FI906083A7 (pt)
HU (1) HUT55802A (pt)
IE (1) IE904485A1 (pt)
IL (1) IL96603A (pt)
MX (1) MX23672A (pt)
NO (1) NO303692B1 (pt)
NZ (1) NZ236393A (pt)
PH (1) PH27373A (pt)
PT (1) PT96139B (pt)
RU (2) RU2053240C1 (pt)
YU (1) YU234790A (pt)
ZA (1) ZA909847B (pt)

Families Citing this family (45)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW213468B (pt) * 1991-06-29 1993-09-21 Hoechst Ag
US5721208A (en) * 1991-06-29 1998-02-24 Hoechst Aktiengesellschaft Glycopeptides a process for their preparation and their use
US5840684A (en) * 1994-01-28 1998-11-24 Eli Lilly And Company Glycopeptide antibiotic derivatives
AU703106B2 (en) * 1994-01-28 1999-03-18 Eli Lilly And Company Glycopeptide antibiotic derivatives
DE19512484A1 (de) * 1995-04-04 1996-10-17 Bayer Ag Kohlenhydratmodifizierte Cytostatika
US5919756A (en) * 1996-06-28 1999-07-06 Eli Lilly And Company Amides
US5952466A (en) * 1997-11-12 1999-09-14 Eli Lilly And Company Reductive alkylation of glycopeptide antibiotics
US5939382A (en) * 1996-11-21 1999-08-17 Eli Lilly And Company Reducing agent for reductive alkylation of glycopeptide antibiotics
ID18900A (id) * 1996-11-21 1998-05-20 Lilly Co Eli Alkilasi menurun dari gliko peptida anti biotik
RU2124022C1 (ru) * 1997-04-10 1998-12-27 Институт биоорганической химии им.М.М.Шемякина и Ю.А.Овчинникова РАН Фуллереновое производное гликопептида, обладающее адъювантной активностью
US5977063A (en) * 1997-05-20 1999-11-02 Eli Lilly And Company Alkylated hexapeptides
US5952310A (en) * 1997-05-20 1999-09-14 Eli Lilly And Company Glycopeptide hexapeptides
US5919771A (en) * 1997-05-20 1999-07-06 Eli Lilly And Company Urea and thiourea derivatives of glycopeptides
US5972933A (en) * 1998-01-08 1999-10-26 Ed. Geistlich Sohne Ag Fur Chemische Industrie Method of treating microbial infections
JP4307723B2 (ja) 1998-05-01 2009-08-05 イーライ リリー アンド カンパニー N1−修飾グリコペプチド
DK1083885T3 (da) 1998-06-11 2007-02-26 Pharmacia & Upjohn Co Llc Delavirdintabletformulering
US6392012B1 (en) 1998-12-23 2002-05-21 Advanced Medicine, Inc. Glycopeptide derivatives and pharmaceutical compositions containing the same
GB9925127D0 (en) * 1999-10-22 1999-12-22 Pharmacia & Upjohn Spa Oral formulations for anti-tumor compounds
US20020004502A1 (en) * 2000-01-05 2002-01-10 Redmond H. Paul Treatment of inflammatory bowel disease
US7365053B2 (en) * 2000-02-11 2008-04-29 Eli Lilly And Company Selective N-acylation of A82846 glygopeptides analogs
SI1276759T1 (sl) * 2000-05-02 2008-12-31 Theravance Inc Postopek reduktivnega alkiliranja na glikopeptidih
EP1278549B1 (en) 2000-05-02 2008-12-10 Theravance, Inc. Composition containing a cyclodextrin and a glycopeptide antibiotic
WO2001083520A2 (en) * 2000-05-02 2001-11-08 Theravance,Inc Polyacid glycopeptide derivatives
DE60040329D1 (de) * 2000-05-09 2008-11-06 Lucent Technologies Inc Verbesserte Steurung der Dienstequalität in einem mobilen Telekommunikationsnetz
AU2001259816A1 (en) 2000-06-22 2002-01-02 Advanced Medecine, Inc. Polyhydroxy glycopeptide derivatives
US6872804B2 (en) * 2000-06-22 2005-03-29 Theravance, Inc. Glycopeptide disulfide and thioester derivatives
UA75083C2 (uk) 2000-06-22 2006-03-15 Тераванс, Інк. Похідні глікопептидфосфонатів
WO2001098327A2 (en) * 2000-06-22 2001-12-27 Theravance, Inc. Glycopeptide carboxy-saccharide derivatives
TWI312785B (en) * 2001-08-24 2009-08-01 Theravance Inc Process for preparing vancomycin derivatives
TWI275594B (en) * 2001-08-24 2007-03-11 Theravance Inc Process for preparing vancomycin phosphonate derivatives
EP1624858B1 (en) 2003-04-09 2018-06-06 Rutgers, the State University of New Jersey Novel encochleation methods
JP4330169B2 (ja) * 2004-11-29 2009-09-16 国立大学法人名古屋大学 グリコペプチド抗生物質モノマー誘導体
UA90707C2 (en) 2005-04-06 2010-05-25 Астразенека Аб Novel 5-substituted 7-amino-[1,3]thiazolo[4,5-d]pyrimidine derivatives
AR053347A1 (es) 2005-04-06 2007-05-02 Astrazeneca Ab Derivados de [1,3]tiazolo[4,5-d]pirimidin-2(3h)-ona 5,7-sustituidos
JP5178520B2 (ja) 2005-09-22 2013-04-10 メディバス エルエルシー 固体ポリマー送達組成物およびその使用法
JP5192384B2 (ja) 2005-09-22 2013-05-08 メディバス エルエルシー ビス−(α−アミノ)−ジオール−ジエステル含有ポリ(エステルアミド)およびポリ(エステルウレタン)組成物および使用の方法
TW200808818A (en) 2006-05-26 2008-02-16 Shionogi & Co Glycopeptide antibiotic derivatives
KR20100109934A (ko) 2007-12-26 2010-10-11 시오노기세야쿠 가부시키가이샤 글리코펩티드 항생 물질 배당화 유도체
EP2260060A4 (en) 2008-04-01 2013-01-16 Univ Cornell ORGANIC SOLUBLE CHITOSA SALT AND CHITOSAN DERIVED BIOMATERIALS MANUFACTURED THEREFROM
CN101928331B (zh) * 2009-06-26 2014-05-28 上海来益生物药物研究开发中心有限责任公司 一种化合物及其应用
CA2834788C (en) 2011-05-05 2020-11-17 Coordinated Program Development, Llc Cochleate compositions and methods of making and using same
CN104418941B (zh) * 2013-08-19 2017-11-07 爱斯医药科技(南京)有限公司 万古霉素衍生物、制备方法及其应用
IN2013CH04314A (pt) 2013-09-23 2015-08-28 Jawaharlal Nehru Ct For Advanced Scient Res Jncasr
HUE070928T2 (hu) * 2014-07-17 2025-07-28 Melinta Therapeutics Llc Nagy tisztaságú oritavancin és eljárás annak elõállítására
CN108409837B (zh) 2018-03-06 2021-09-24 上海来益生物药物研究开发中心有限责任公司 一组具有抗耐药性细菌活性的糖肽类化合物、其制备方法和应用

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4552701A (en) * 1984-04-16 1985-11-12 Eli Lilly And Company Glycopeptide antibiotics and process of preparation
US4698327A (en) * 1985-04-25 1987-10-06 Eli Lilly And Company Novel glycopeptide derivatives
US4643987A (en) * 1985-08-14 1987-02-17 Eli Lilly And Company Modified glycopeptides
US4639433A (en) * 1985-08-14 1987-01-27 Eli Lilly And Company Glycopeptide derivatives
US4946941A (en) * 1986-01-24 1990-08-07 Shionogi & Co., Ltd. Novel glycopeptide antibiotics
EG18377A (en) * 1986-09-19 1993-04-30 Lilly Co Eli Process for preparing glycopeptide antibiotics
GB8701872D0 (en) * 1987-01-28 1987-03-04 Lepetit Spa N15-alkyl & n15,n15-dialkyl derivatives
US5071749A (en) * 1987-04-16 1991-12-10 Shionogi & Co., Ltd. Glycopetide antibiotic pa-45052-b

Also Published As

Publication number Publication date
HUT55802A (en) 1991-06-28
JP3590638B2 (ja) 2004-11-17
ZA909847B (en) 1992-08-26
EP0435503A1 (en) 1991-07-03
DE69033087D1 (de) 1999-06-10
RU2053240C1 (ru) 1996-01-27
NO905354D0 (no) 1990-12-11
CA2031803C (en) 2001-05-29
IE904485A1 (en) 1991-06-19
EP0435503B1 (en) 1999-05-06
NO905354L (no) 1991-06-14
JPH04108800A (ja) 1992-04-09
IL96603A (en) 1998-02-08
AU633165B2 (en) 1993-01-21
CN1052483A (zh) 1991-06-26
US5591714A (en) 1997-01-07
NZ236393A (en) 1992-05-26
ES2131496T3 (es) 1999-08-01
DE69033087T2 (de) 1999-10-14
AU6796490A (en) 1991-06-20
FI906083A7 (fi) 1991-06-14
FI906083A0 (fi) 1990-12-11
YU234790A (sh) 1992-12-21
NO303692B1 (no) 1998-08-17
CA2031803A1 (en) 1991-06-14
KR910011896A (ko) 1991-08-07
PT96139B (pt) 1998-04-30
CN1034506C (zh) 1997-04-09
PH27373A (en) 1993-06-21
RU2041237C1 (ru) 1995-08-09
IL96603A0 (en) 1991-09-16
MX23672A (es) 1993-11-01

Similar Documents

Publication Publication Date Title
PT97906A (pt) Processo para a preparacao de novos derivados de tiofeno
PT99409A (pt) Processo para a preparacao de benzimidazois polissubstituidos
PT98638A (pt) Processo para a preparacao de derivados de borsolina
PT93785A (pt) Processo para a preparacao de derivados de 3-substituido-2-oxindole
PT96411A (pt) Processo para a preparacao de derivados de azaoxindole
PT82890B (pt) Processo para a preparacao de novos derivados de n-aralquil-piperidinametanol
BR9306629A (pt) Processo para preparar derivados de triaza-ciclo-nonano
PT94059A (pt) Processo para a preparacao de copolimetros hidrossoluveis, de n-vinilamidas
PT89780A (pt) Processo para a preparacao de derivados da tetrahidroisoquinolina
BR8907013A (pt) Processo para preparacao de uma dimetiltetralina
PT90914A (pt) Processo para a preparacao de derivados de benzazepinae benzotiazapina
BR9007734A (pt) Processo para a obtencao de alquil-polietoxietersulfatos
BR9001481A (pt) Metodo para esmerilhamento de um cilindro
PT93629A (pt) Processo para a preparacao de derivados de tieno-triazolo-diazepina
PT82445B (pt) Processo para a preparacao de novos derivados glicopeptidicos
BR9001503A (pt) Processo para a preparacao de alquil-halogenossilanos
PT94008A (pt) Processo para a preparacao de novos derivados de tieno-triazolo-diazepina
PT89026A (pt) Processo para a preparacao de factor de activacao dos neutrofilos
PT96322A (pt) Processo para a preparacao de derivados de glicerol
PT92539A (pt) Processo para a preparacao de derivados de anfotericina b
BR9004539A (pt) Processo para a obtencao de 1,1,1,2-tetrafluoretano
PT91205A (pt) Processo para a preparacao de 2-aminopurina
BR9004428A (pt) Processo para a obtencao de alquilhalogenossilanos
PT93631A (pt) Processo para a preparacao de derivados de tieno-triazolo-diazepina
BR9003360A (pt) Processo para a obtencao de 1,1,1-trifluor-2-cloroetano

Legal Events

Date Code Title Description
BB1A Laying open of patent application

Effective date: 19910430

FG3A Patent granted, date of granting

Effective date: 19980123

MM3A Annulment or lapse

Free format text: LAPSE DUE TO NON-PAYMENT OF FEES

Effective date: 19990731