MX376876B - Moleculas de anticuerpo de union a trombina y sus usos. - Google Patents

Moleculas de anticuerpo de union a trombina y sus usos.

Info

Publication number
MX376876B
MX376876B MX2018000197A MX2018000197A MX376876B MX 376876 B MX376876 B MX 376876B MX 2018000197 A MX2018000197 A MX 2018000197A MX 2018000197 A MX2018000197 A MX 2018000197A MX 376876 B MX376876 B MX 376876B
Authority
MX
Mexico
Prior art keywords
thrombin
antibody molecules
binding antibody
exosite
recognise
Prior art date
Application number
MX2018000197A
Other languages
English (en)
Inventor
James Andrew Huntington
Jonathan Langdown
Trevor Baglin
Original Assignee
Janssen Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceuticals Inc filed Critical Janssen Pharmaceuticals Inc
Publication of MX376876B publication Critical patent/MX376876B/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K16/00Immunoglobulins [IG], e.g. monoclonal or polyclonal antibodies
    • C07K16/40Immunoglobulins [IG], e.g. monoclonal or polyclonal antibodies against enzymes
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/04Antineoplastic agents specific for metastasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/04Antihaemorrhagics; Procoagulants; Haemostatic agents; Antifibrinolytic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K16/00Immunoglobulins [IG], e.g. monoclonal or polyclonal antibodies
    • C07K16/18Immunoglobulins [IG], e.g. monoclonal or polyclonal antibodies against material from animals or humans
    • C07K16/36Immunoglobulins [IG], e.g. monoclonal or polyclonal antibodies against material from animals or humans against blood coagulation factors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K39/00Medicinal preparations containing antigens or antibodies
    • A61K2039/505Medicinal preparations containing antigens or antibodies comprising antibodies
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/20Immunoglobulins specific features characterized by taxonomic origin
    • C07K2317/21Immunoglobulins specific features characterized by taxonomic origin from primates, e.g. man
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/30Immunoglobulins specific features characterized by aspects of specificity or valency
    • C07K2317/34Identification of a linear epitope shorter than 20 amino acid residues or of a conformational epitope defined by amino acid residues
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/50Immunoglobulins specific features characterized by immunoglobulin fragments
    • C07K2317/55Fab or Fab'
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/50Immunoglobulins specific features characterized by immunoglobulin fragments
    • C07K2317/56Immunoglobulins specific features characterized by immunoglobulin fragments variable (Fv) region, i.e. VH and/or VL
    • C07K2317/565Complementarity determining region [CDR]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/70Immunoglobulins specific features characterized by effect upon binding to a cell or to an antigen
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/70Immunoglobulins specific features characterized by effect upon binding to a cell or to an antigen
    • C07K2317/76Antagonist effect on antigen, e.g. neutralization or inhibition of binding
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/90Immunoglobulins specific features characterized by (pharmaco)kinetic aspects or by stability of the immunoglobulin
    • C07K2317/92Affinity (KD), association rate (Ka), dissociation rate (Kd) or EC50 value

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Biochemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Hematology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Oncology (AREA)
  • Biomedical Technology (AREA)
  • Diabetes (AREA)
  • Communicable Diseases (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

La presente invención se refiere a una molécula de anticuerpo aislada que se une específicamente a la región de exositio 1 de trombina, en donde la molécula de anticuerpo comprende un dominio VH que comprende un HCDR1, HCDR2 y HCDR3 que tienen las secuencias de SEC ID Nos. 3, 4 y 5, respectivamente, y un dominio VL que comprende un LCDR2 y LCDR3 que tienen la secuencia de SEC ID Nos. 8 y 9, respectivamente, y un LCDR1 que tiene la secuencia de SEC ID NO. 7 en la que un sitio de glicosilación es mutado al introducir una sustitución en un residuo de aminoácido correspondiente a N28 en la SEC ID NO. 6.
MX2018000197A 2011-12-14 2012-12-14 Moleculas de anticuerpo de union a trombina y sus usos. MX376876B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB1121513.4A GB201121513D0 (en) 2011-12-14 2011-12-14 Thrombin-binding antibody molecules and uses thereof
PCT/GB2012/053140 WO2013088164A1 (en) 2011-12-14 2012-12-14 Thrombin-binding antibody molecules and uses thereof

Publications (1)

Publication Number Publication Date
MX376876B true MX376876B (es) 2025-03-07

Family

ID=45560465

Family Applications (2)

Application Number Title Priority Date Filing Date
MX2018000197A MX376876B (es) 2011-12-14 2012-12-14 Moleculas de anticuerpo de union a trombina y sus usos.
MX2014007170A MX353281B (es) 2011-12-14 2012-12-14 Moleculas de anticuerpo de union a trombina y sus usos.

Family Applications After (1)

Application Number Title Priority Date Filing Date
MX2014007170A MX353281B (es) 2011-12-14 2012-12-14 Moleculas de anticuerpo de union a trombina y sus usos.

Country Status (34)

Country Link
US (5) US9518129B2 (es)
EP (2) EP2791177B1 (es)
JP (2) JP6216954B2 (es)
KR (1) KR102114506B1 (es)
CN (2) CN107936119B (es)
AU (2) AU2012351858B2 (es)
BR (1) BR112014014605A2 (es)
CA (1) CA2856656C (es)
CO (1) CO7101192A2 (es)
CY (1) CY1119599T1 (es)
DK (1) DK2791177T3 (es)
ES (1) ES2642718T3 (es)
GB (1) GB201121513D0 (es)
HK (1) HK1246326A1 (es)
HR (1) HRP20171775T1 (es)
HU (1) HUE034793T2 (es)
IL (1) IL232797B (es)
LT (1) LT2791177T (es)
ME (1) ME02901B (es)
MX (2) MX376876B (es)
MY (1) MY170980A (es)
NO (1) NO2791177T3 (es)
PE (2) PE20141706A1 (es)
PH (1) PH12014501169A1 (es)
PL (1) PL2791177T3 (es)
PT (1) PT2791177T (es)
RS (1) RS56510B1 (es)
RU (2) RU2642276C2 (es)
SG (1) SG11201402560WA (es)
SI (1) SI2791177T1 (es)
SM (1) SMT201700580T1 (es)
UA (1) UA116531C2 (es)
WO (1) WO2013088164A1 (es)
ZA (1) ZA201403836B (es)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9518128B2 (en) * 2011-12-14 2016-12-13 Janssen Pharmaceuticals, Inc. Thrombin-binding antibody molecules
GB201121513D0 (en) * 2011-12-14 2012-01-25 Cambridge Entpr Ltd Thrombin-binding antibody molecules and uses thereof
GB201310949D0 (en) * 2013-06-19 2013-07-31 Cambridge Entpr Ltd Binding Motif
GB201310948D0 (en) * 2013-06-19 2013-07-31 Cambridge Entpr Ltd Screening methods
CN107043423B (zh) * 2016-02-05 2021-02-26 江苏恒瑞医药股份有限公司 凝血酶抗体、其抗原结合片段及医药用途
CA3013254A1 (en) * 2016-02-05 2017-08-10 Jiangsu Hengrui Medicine Co., Ltd. Thrombin antibody, antigen-binding fragment and pharmaceutical use thereof
WO2018081534A1 (en) * 2016-10-28 2018-05-03 President And Fellows Of Harvard College Assay for exo-site binding molecules
WO2019030706A1 (en) 2017-08-10 2019-02-14 Janssen Pharmaceutica Nv ANTI-THROMBIN ANTIBODY MOLECULES AND METHODS OF USE IN ORTHOPEDIC SURGERY
WO2019035055A1 (en) 2017-08-16 2019-02-21 Janssen Pharmaceutica Nv ANTI-THROMBIN ANTIBODY MOLECULES AND METHODS OF USE WITH PLATELET ANTI-AGGREGATE AGENTS
WO2020003077A1 (en) * 2018-06-25 2020-01-02 Janssen Pharmaceutica Nv Anti-thrombin antibody molecules for use in patients at risk for gastrointestinal (gi) bleeding

Family Cites Families (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE68908175T2 (de) * 1988-05-27 1994-03-03 Centocor Inc Gefriergetrocknete formulierung für antikörperprodukte.
US5530101A (en) 1988-12-28 1996-06-25 Protein Design Labs, Inc. Humanized immunoglobulins
US5196404B1 (en) 1989-08-18 1996-09-10 Biogen Inc Inhibitors of thrombin
US5240913A (en) 1989-08-18 1993-08-31 Biogen, Inc. Inhibitors of thrombin
CA2082643A1 (en) 1990-05-10 1991-11-11 Jan H. Nuijens Inhibitors of factor xii activation and applications thereof
GB9015198D0 (en) 1990-07-10 1990-08-29 Brien Caroline J O Binding substance
US5443827A (en) * 1993-05-03 1995-08-22 President And Fellows Of Harvard College Fibrin-targeted inhibitors of thrombin
CA2180140A1 (en) * 1993-12-27 1995-07-06 Jeffrey I. Weitz Methods and compositions for inhibiting thrombogenesis
GB9613718D0 (en) 1996-06-29 1996-08-28 Thrombosis Res Inst Thrombin inhibitors
US5985833A (en) 1996-09-17 1999-11-16 Wisconsin Alumni Research Foundation Thrombin inhibitor
WO2001000667A2 (en) 1999-06-29 2001-01-04 The Government Of The United States Of America, As Represented By The Secretary, Department Of Health And Human Services Anti-thrombin peptide from anopheles albimanus salivary gland
CA2378473A1 (en) * 1999-07-23 2001-02-01 The Regents Of The University Of California Modulation of platelet activation
KR20070116192A (ko) * 2000-05-15 2007-12-06 스미스클라인 비참 코포레이션 항혈전제
AU2001286900A1 (en) 2000-08-31 2002-03-13 Cor Therapeutics, Inc. Therapeutics and diagnostics based on a novel signal transduction system in platelets
CA2453202C (en) * 2001-07-06 2012-10-16 Oregon Health & Science University Peptides which modulate blood coagulation and methods of use thereof
TWI338009B (en) * 2001-10-29 2011-03-01 Genentech Inc Antibodies for inhibiting blood coagulation and methods of use thereof
MEP0208A (xx) 2005-08-26 2010-02-10 Archemix Corp Aptameri koji vezuje trombin sa visokim afininitetom
US20100158890A1 (en) 2006-03-15 2010-06-24 Kenichi Tanaka Use of thrombin mutants to inhibit the anticoagulation effect of thrombin inhibitors
GB0711779D0 (en) 2007-06-18 2007-07-25 Univ Singapore Thrombin inhibitor
TR201820051T4 (tr) 2008-06-19 2019-01-21 Prothix Bv Anti-faktör XI Antikorlarının Trombüs Oluşumunun Engellenmesi Veya Tedavisi İçin Kullanılması
WO2010033167A2 (en) * 2008-09-18 2010-03-25 Archemix Corp. Anti-thrombin aptamer formulations and methods for use
IL230564B2 (en) 2011-07-22 2023-09-01 Csl Ltd Anticoagulant monoclonal antibodies anti–factor xii/fxiia, a method for their preparation, a pharmaceutical compound containing them and medical uses.
GB201121513D0 (en) * 2011-12-14 2012-01-25 Cambridge Entpr Ltd Thrombin-binding antibody molecules and uses thereof
US9518128B2 (en) * 2011-12-14 2016-12-13 Janssen Pharmaceuticals, Inc. Thrombin-binding antibody molecules

Also Published As

Publication number Publication date
MX353281B (es) 2018-01-08
WO2013088164A1 (en) 2013-06-20
EP2791177A1 (en) 2014-10-22
AU2017268655B2 (en) 2019-05-09
ZA201403836B (en) 2015-12-23
CY1119599T1 (el) 2018-04-04
HUE034793T2 (en) 2018-02-28
US20210371543A1 (en) 2021-12-02
AU2012351858A1 (en) 2014-06-12
GB201121513D0 (en) 2012-01-25
CO7101192A2 (es) 2014-10-31
US20140370008A1 (en) 2014-12-18
JP6705785B2 (ja) 2020-06-03
NO2791177T3 (es) 2018-02-03
DK2791177T3 (en) 2017-12-18
CN104053673B (zh) 2018-01-12
ME02901B (me) 2018-04-20
PT2791177T (pt) 2017-11-29
SG11201402560WA (en) 2014-06-27
SMT201700580T1 (it) 2018-01-11
LT2791177T (lt) 2017-11-27
MY170980A (en) 2019-09-23
EP3275903A1 (en) 2018-01-31
RU2014124985A (ru) 2016-02-10
KR102114506B1 (ko) 2020-05-22
SI2791177T1 (en) 2018-03-30
CN104053673A (zh) 2014-09-17
PH12014501169B1 (en) 2014-09-08
CA2856656A1 (en) 2013-06-20
US20190276558A1 (en) 2019-09-12
ES2642718T3 (es) 2017-11-17
EP2791177B1 (en) 2017-09-06
US20180334511A1 (en) 2018-11-22
IL232797B (en) 2018-07-31
US9988463B2 (en) 2018-06-05
RU2017144629A (ru) 2019-02-18
US10287363B2 (en) 2019-05-14
PE20190171A1 (es) 2019-02-01
JP6216954B2 (ja) 2017-10-25
HRP20171775T1 (hr) 2017-12-29
IL232797A0 (en) 2014-07-31
CA2856656C (en) 2021-01-19
US20170066842A1 (en) 2017-03-09
MX2014007170A (es) 2015-04-17
UA116531C2 (uk) 2018-04-10
RU2642276C2 (ru) 2018-01-24
HK1202564A1 (en) 2015-10-02
RS56510B1 (sr) 2018-02-28
PL2791177T3 (pl) 2018-03-30
PH12014501169A1 (en) 2014-09-08
BR112014014605A2 (pt) 2017-06-13
KR20140105556A (ko) 2014-09-01
CN107936119A (zh) 2018-04-20
CN107936119B (zh) 2021-06-15
NZ625386A (en) 2017-03-31
US9518129B2 (en) 2016-12-13
RU2017144629A3 (es) 2021-04-05
HK1246326A1 (en) 2018-09-07
AU2017268655A1 (en) 2017-12-21
JP2018039798A (ja) 2018-03-15
AU2012351858B2 (en) 2017-10-05
PE20141706A1 (es) 2014-11-13
JP2015501830A (ja) 2015-01-19

Similar Documents

Publication Publication Date Title
MX376876B (es) Moleculas de anticuerpo de union a trombina y sus usos.
CY1121862T1 (el) Αντισωματα anti-phf-tau και χρησεις αυτων
EA201791693A1 (ru) Гетеродимерные иммуноглобулины
EA201791485A1 (ru) Анти-cd47-антитела и их применения
MX381456B (es) Regulador de ph de transduccion.
MX382540B (es) Proteinas de fusion para inhibir la angiogenesis
TR201808169T3 (tr) Rekombinant probiyotik bakteriler .
BR112017001579A2 (pt) anticorpos anti-cd3, anticorpos anti-cd3 ativáveis, anticorpos anti-cd3 multiespecíficos, anticorpos anti-cd3 ativáveis multiespecíficos e métodos de uso dos mesmos
EA201491996A1 (ru) Антагонисты st2l и способы их применения
TN2012000366A1 (en) Anticoagulant antidotes
MY198522A (en) Methods of treating and preventing endothelial dysfunction using bardoxolone methyl or analogs thereof
MX2014000363A (es) Anticuerpos monoclonales inhibidores anti-factor xii-xiia.
UA111098C2 (uk) Проліки адреномедуліну на основі поліетиленгліколю і їх застосування
EA201491286A1 (ru) Способ лечения потери костной массы альвеолярного отростка посредством применения антител к склеростину
MX349514B (es) Agentes de reversion anticoagulante.
WO2014159669A3 (en) Aptamers that bind to il-6 and their use in treating or diagnosing il-6 mediated conditions
EA201792328A1 (ru) Способ очистки белков
TN2013000388A1 (en) Anticoagulant antidotes
JOP20140008B1 (ar) استخدام العوامل المساعدة لمستقبل ألفا 7 أسيتيل كولين نيكوتينية
EA201990181A1 (ru) Получение активированных клостридиальных нейротоксинов
MX2018007221A (es) Moleculas de anticuerpos que se unen al factor de necrosis tumoral alfa (tnf alfa).
EA201501176A1 (ru) Замещенные бензоксазолы
EA201691749A1 (ru) Пептиды и способы применения
UA113260C2 (xx) Біопрепарат для очищення господарсько-побутових відходів
TR201111820U (tr) Işıklandırmalı kostüm eteği.