MY197383A - Mono- or di-substituted indole derivatives as dengue viral replication inhibitors - Google Patents

Mono- or di-substituted indole derivatives as dengue viral replication inhibitors

Info

Publication number
MY197383A
MY197383A MYPI2018000381A MYPI2018000381A MY197383A MY 197383 A MY197383 A MY 197383A MY PI2018000381 A MYPI2018000381 A MY PI2018000381A MY PI2018000381 A MYPI2018000381 A MY PI2018000381A MY 197383 A MY197383 A MY 197383A
Authority
MY
Malaysia
Prior art keywords
dengue viral
compounds
mono
substituted indole
viral replication
Prior art date
Application number
MYPI2018000381A
Inventor
Alice Marie-Eve Bardiot Dorothee
Didier M Marchand Arnaud
Rudolf Romanie Kesteleyn Bart
Bonfanti Jean-Francois
Hugo Maria Jonckers Tim
Jean-Marie Bernard Raboisson Pierre
Original Assignee
Univ Leuven Kath
Janssen Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Univ Leuven Kath, Janssen Pharmaceuticals Inc filed Critical Univ Leuven Kath
Priority claimed from PCT/EP2016/071845 external-priority patent/WO2017046255A1/en
Publication of MY197383A publication Critical patent/MY197383A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/12—Radicals substituted by oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

The present invention concerns mono- or di-substituted indole compounds, methods to prevent or treat dengue viral infections by using said compounds and also relates to said compounds for use as a medicine, more preferably for use as a medicine to treat or prevent dengue viral infections. The present invention furthermore relates to pharmaceutical compositions or combination preparations of the compounds, to the compositions or preparations for use as a medicine, more preferably for the prevention or treatment of dengue viral infections. The invention also relates to processes for preparation of the compounds
MYPI2018000381A 2015-09-16 2016-09-15 Mono- or di-substituted indole derivatives as dengue viral replication inhibitors MY197383A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP15185523 2015-09-16
PCT/EP2016/071845 WO2017046255A1 (en) 2015-09-16 2016-09-15 Mono- or di-substituted indole derivatives as dengue viral replication inhibitors

Publications (1)

Publication Number Publication Date
MY197383A true MY197383A (en) 2023-06-15

Family

ID=54207297

Family Applications (1)

Application Number Title Priority Date Filing Date
MYPI2018000381A MY197383A (en) 2015-09-16 2016-09-15 Mono- or di-substituted indole derivatives as dengue viral replication inhibitors

Country Status (2)

Country Link
AR (1) AR106029A1 (en)
MY (1) MY197383A (en)

Also Published As

Publication number Publication date
AR106029A1 (en) 2017-12-06

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