NO20002834D0 - S-oksyd og S,S-dioksyd-tetrahydrothiopyran- fenyloksazolidinoner - Google Patents
S-oksyd og S,S-dioksyd-tetrahydrothiopyran- fenyloksazolidinonerInfo
- Publication number
- NO20002834D0 NO20002834D0 NO20002834A NO20002834A NO20002834D0 NO 20002834 D0 NO20002834 D0 NO 20002834D0 NO 20002834 A NO20002834 A NO 20002834A NO 20002834 A NO20002834 A NO 20002834A NO 20002834 D0 NO20002834 D0 NO 20002834D0
- Authority
- NO
- Norway
- Prior art keywords
- phenyloxazolidinones
- tetrahydrothiopyran
- dioxide
- oxide
- dichloromethyl
- Prior art date
Links
- RCCPEORTSYDPMB-UHFFFAOYSA-N hydroxy benzenecarboximidothioate Chemical compound OSC(=N)C1=CC=CC=C1 RCCPEORTSYDPMB-UHFFFAOYSA-N 0.000 title 1
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 1
- 239000004599 antimicrobial Substances 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 125000004772 dichloromethyl group Chemical group [H]C(Cl)(Cl)* 0.000 abstract 1
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 abstract 1
- 125000001153 fluoro group Chemical group F* 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D263/18—Oxygen atoms
- C07D263/20—Oxygen atoms attached in position 2
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Plural Heterocyclic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Catalysts (AREA)
- Solid-Sorbent Or Filter-Aiding Compositions (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US6783097P | 1997-12-05 | 1997-12-05 | |
| US8949898P | 1998-06-16 | 1998-06-16 | |
| US10018598P | 1998-09-14 | 1998-09-14 | |
| PCT/US1998/024526 WO1999029688A1 (en) | 1997-12-05 | 1998-11-23 | S-oxide and s,s-dioxide tetrahydrothiopyran phenyloxazolidinones |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO20002834D0 true NO20002834D0 (no) | 2000-06-02 |
| NO20002834L NO20002834L (no) | 2000-07-21 |
| NO316447B1 NO316447B1 (no) | 2004-01-26 |
Family
ID=27371238
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20002834A NO316447B1 (no) | 1997-12-05 | 2000-06-02 | S-oksidtetrahydrotiopyran-fenyloksazolidinoner og anvendelse derav |
Country Status (21)
| Country | Link |
|---|---|
| US (2) | US6083967A (no) |
| EP (2) | EP1036074B1 (no) |
| JP (1) | JP2001525408A (no) |
| KR (1) | KR20010032782A (no) |
| CN (2) | CN1532535A (no) |
| AT (1) | ATE231859T1 (no) |
| AU (2) | AU752454B2 (no) |
| BR (1) | BR9814897A (no) |
| CA (1) | CA2309026A1 (no) |
| DE (1) | DE69811117T2 (no) |
| DK (1) | DK1036074T3 (no) |
| ES (1) | ES2191985T3 (no) |
| HU (1) | HUP0100558A3 (no) |
| ID (1) | ID21450A (no) |
| NO (1) | NO316447B1 (no) |
| NZ (1) | NZ504930A (no) |
| PL (1) | PL340835A1 (no) |
| SI (1) | SI1036074T1 (no) |
| SK (1) | SK7692000A3 (no) |
| TW (2) | TW553942B (no) |
| WO (1) | WO1999029688A1 (no) |
Families Citing this family (22)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6511468B1 (en) | 1997-10-17 | 2003-01-28 | Micro Therapeutics, Inc. | Device and method for controlling injection of liquid embolic composition |
| TR200003595T2 (tr) | 1998-06-05 | 2001-07-23 | Astrazeneca Ab | Kimyasal bileşikler |
| MY120189A (en) * | 1999-11-04 | 2005-09-30 | Upjohn Co | Sultam and sultone derived oxazolidinones |
| GB9928568D0 (en) | 1999-12-03 | 2000-02-02 | Zeneca Ltd | Chemical compounds |
| DE19962924A1 (de) | 1999-12-24 | 2001-07-05 | Bayer Ag | Substituierte Oxazolidinone und ihre Verwendung |
| GB0009803D0 (en) | 2000-04-25 | 2000-06-07 | Astrazeneca Ab | Chemical compounds |
| DE10129725A1 (de) | 2001-06-20 | 2003-01-02 | Bayer Ag | Kombinationstherapie substituierter Oxazolidinone |
| US7141588B2 (en) | 2002-02-25 | 2006-11-28 | Pfizer, Inc. | N-aryl-2-oxazolidinone-5-carboxamides and their derivatives |
| AR038536A1 (es) | 2002-02-25 | 2005-01-19 | Upjohn Co | N-aril-2-oxazolidinona-5- carboxamidas y sus derivados |
| ES2258234T3 (es) | 2002-08-12 | 2006-08-16 | PHARMACIA & UPJOHN COMPANY LLC | N-aril-2-oxazolidinonas y sus derivados. |
| JP2006509035A (ja) | 2002-11-21 | 2006-03-16 | ファルマシア・アンド・アップジョン・カンパニー・エルエルシー | 抗菌剤としてのｎ−（４−（ピペラジン−１−イル）−フェニル−２−オキサゾリジノン−５−カルボキサミド誘導体および関連化合物 |
| DE10300111A1 (de) | 2003-01-07 | 2004-07-15 | Bayer Healthcare Ag | Verfahren zur Herstellung von 5-Chlor-N-({(5S)-2-oxo-3-[4-(3-oxo-4-morpholinyl)-phenyl]-1,3-oxazolidin-5-yl}-methyl)-2-thiophencarboxamid |
| US7304050B2 (en) | 2003-09-16 | 2007-12-04 | Pfizer Inc. | Antibacterial agents |
| DE10355461A1 (de) | 2003-11-27 | 2005-06-23 | Bayer Healthcare Ag | Verfahren zur Herstellung einer festen, oral applizierbaren pharmazeutischen Zusammensetzung |
| DE102004062475A1 (de) * | 2004-12-24 | 2006-07-06 | Bayer Healthcare Ag | Feste, oral applizierbare pharmazeutische Darreichungsformen mit modifizierter Freisetzung |
| EP1685841A1 (en) | 2005-01-31 | 2006-08-02 | Bayer Health Care Aktiengesellschaft | Prevention and treatment of thromboembolic disorders |
| DE102005045518A1 (de) | 2005-09-23 | 2007-03-29 | Bayer Healthcare Ag | 2-Aminoethoxyessigsäure-Derivate und ihre Verwendung |
| US8188270B2 (en) | 2005-10-04 | 2012-05-29 | Bayer Schering Pharma Aktiengesellschaft | Polymorphous form of 5-chloro-N-({(5S)-2-oxo-3[4-(3-oxo-4-morpholinyl)-phenyl]-1,3-oxazolidine-5-yl}-methyl)-2-thiophene carboxamide |
| DE102005047561A1 (de) | 2005-10-04 | 2007-04-05 | Bayer Healthcare Ag | Feste, oral applizierbare pharmazeutische Darreichungsformen mit schneller Wirkstofffreisetzung |
| DE102005047558A1 (de) * | 2005-10-04 | 2008-02-07 | Bayer Healthcare Ag | Kombinationstherapie substituierter Oxazolidinone zur Prophylaxe und Behandlung von cerebralen Durchblutungsstörungen |
| CN102262066A (zh) * | 2011-06-16 | 2011-11-30 | 董理 | 一种检测单胺氧化酶含量的方法和试剂盒 |
| CN104610479B (zh) * | 2013-11-05 | 2017-03-29 | 中国石油化工股份有限公司 | 用于乙烯聚合的负载化茂金属催化剂及其制备方法和应用 |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4897409A (en) * | 1986-09-03 | 1990-01-30 | Delalande S.A. | 5-aminoethyloxazolidin-2-one derivatives |
| US4885154A (en) * | 1988-03-01 | 1989-12-05 | Alza Corporation | Method for reducing sensitization or irritation in transdermal drug delivery and means therefor |
| US5254577A (en) * | 1988-07-29 | 1993-10-19 | The Du Pont Merck Pharmaceutical Company | Aminomethyloxooxazolidinyl arylbenzene derivatives useful as antibacterial agents |
| US5130316A (en) * | 1988-07-29 | 1992-07-14 | Du Pont Merck Pharmaceutical Company | Aminomethyloxooxazlidinyl arylbenzene derivatives useful as antibacterial agents |
| US4948801A (en) * | 1988-07-29 | 1990-08-14 | E. I. Du Pont De Nemours And Company | Aminomethyloxooxazolidinyl arylbenzene derivatives useful as antibacterial agents |
| JP2669579B2 (ja) * | 1991-10-23 | 1997-10-29 | エーザイ株式会社 | オキサゾリドン誘導体 |
| ATE146783T1 (de) * | 1991-11-01 | 1997-01-15 | Upjohn Co | Substituierte aryl- und heteroaryl- phenyloxazolidinone |
| EP0673370B1 (en) * | 1992-12-08 | 1998-01-07 | PHARMACIA & UPJOHN COMPANY | Tropone-substituted phenyloxazolidinone antibacterial agents |
| RU2175324C2 (ru) * | 1995-09-01 | 2001-10-27 | Фармация Энд Апджон Компани | Фенилоксазолидиноны, имеющие с-с-связь с 4-8-членными гетероциклическими кольцами |
| GB9702213D0 (en) * | 1996-02-24 | 1997-03-26 | Zeneca Ltd | Chemical compounds |
-
1998
- 1998-11-20 US US09/196,890 patent/US6083967A/en not_active Expired - Fee Related
- 1998-11-23 EP EP98962811A patent/EP1036074B1/en not_active Expired - Lifetime
- 1998-11-23 BR BR9814897-4A patent/BR9814897A/pt not_active Application Discontinuation
- 1998-11-23 NZ NZ504930A patent/NZ504930A/en unknown
- 1998-11-23 KR KR1020007006081A patent/KR20010032782A/ko not_active Ceased
- 1998-11-23 CN CNA2004100328277A patent/CN1532535A/zh active Pending
- 1998-11-23 JP JP2000524282A patent/JP2001525408A/ja active Pending
- 1998-11-23 SK SK769-2000A patent/SK7692000A3/sk unknown
- 1998-11-23 DK DK98962811T patent/DK1036074T3/da active
- 1998-11-23 DE DE69811117T patent/DE69811117T2/de not_active Expired - Fee Related
- 1998-11-23 AU AU17968/99A patent/AU752454B2/en not_active Ceased
- 1998-11-23 WO PCT/US1998/024526 patent/WO1999029688A1/en not_active Ceased
- 1998-11-23 ES ES98962811T patent/ES2191985T3/es not_active Expired - Lifetime
- 1998-11-23 AT AT98962811T patent/ATE231859T1/de not_active IP Right Cessation
- 1998-11-23 SI SI9830371T patent/SI1036074T1/xx unknown
- 1998-11-23 EP EP02015566A patent/EP1254906A1/en not_active Withdrawn
- 1998-11-23 HU HU0100558A patent/HUP0100558A3/hu unknown
- 1998-11-23 CN CNB988110695A patent/CN1154645C/zh not_active Expired - Fee Related
- 1998-11-23 CA CA002309026A patent/CA2309026A1/en not_active Abandoned
- 1998-11-23 PL PL98340835A patent/PL340835A1/xx unknown
- 1998-11-26 ID IDP981545A patent/ID21450A/id unknown
- 1998-12-04 TW TW087120185A patent/TW553942B/zh not_active IP Right Cessation
- 1998-12-04 TW TW092121194A patent/TWI239331B/zh not_active IP Right Cessation
-
1999
- 1999-11-05 US US09/434,911 patent/US6265178B1/en not_active Expired - Fee Related
-
2000
- 2000-06-02 NO NO20002834A patent/NO316447B1/no unknown
-
2002
- 2002-09-16 AU AU2002301031A patent/AU2002301031B2/en not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| NO316447B1 (no) | 2004-01-26 |
| NO20002834L (no) | 2000-07-21 |
| TWI239331B (en) | 2005-09-11 |
| AU752454B2 (en) | 2002-09-19 |
| ID21450A (id) | 1999-06-10 |
| SK7692000A3 (en) | 2001-03-12 |
| CN1532535A (zh) | 2004-09-29 |
| EP1036074A1 (en) | 2000-09-20 |
| ATE231859T1 (de) | 2003-02-15 |
| CA2309026A1 (en) | 1999-06-17 |
| AU1796899A (en) | 1999-06-28 |
| CN1278817A (zh) | 2001-01-03 |
| DE69811117D1 (de) | 2003-03-06 |
| AU2002301031B2 (en) | 2005-08-25 |
| TW200307673A (en) | 2003-12-16 |
| HUP0100558A3 (en) | 2002-08-28 |
| DE69811117T2 (de) | 2003-07-17 |
| US6083967A (en) | 2000-07-04 |
| EP1254906A1 (en) | 2002-11-06 |
| ES2191985T3 (es) | 2003-09-16 |
| DK1036074T3 (da) | 2003-06-23 |
| NZ504930A (en) | 2002-05-31 |
| JP2001525408A (ja) | 2001-12-11 |
| US6265178B1 (en) | 2001-07-24 |
| SI1036074T1 (en) | 2003-08-31 |
| KR20010032782A (ko) | 2001-04-25 |
| PL340835A1 (en) | 2001-02-26 |
| WO1999029688A1 (en) | 1999-06-17 |
| CN1154645C (zh) | 2004-06-23 |
| HUP0100558A2 (hu) | 2002-05-29 |
| EP1036074B1 (en) | 2003-01-29 |
| HK1032970A1 (en) | 2001-08-10 |
| TW553942B (en) | 2003-09-21 |
| BR9814897A (pt) | 2000-10-03 |
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