NO20004053D0 - Glukokortikoid-selektive antiinflammatoriske midler - Google Patents
Glukokortikoid-selektive antiinflammatoriske midlerInfo
- Publication number
- NO20004053D0 NO20004053D0 NO20004053A NO20004053A NO20004053D0 NO 20004053 D0 NO20004053 D0 NO 20004053D0 NO 20004053 A NO20004053 A NO 20004053A NO 20004053 A NO20004053 A NO 20004053A NO 20004053 D0 NO20004053 D0 NO 20004053D0
- Authority
- NO
- Norway
- Prior art keywords
- glucocorticoid
- inflammatory agents
- selective anti
- mammal
- compounds
- Prior art date
Links
- 229940121363 anti-inflammatory agent Drugs 0.000 title 1
- 239000002260 anti-inflammatory agent Substances 0.000 title 1
- 239000003862 glucocorticoid Substances 0.000 title 1
- 208000023275 Autoimmune disease Diseases 0.000 abstract 2
- 241000124008 Mammalia Species 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 208000026278 immune system disease Diseases 0.000 abstract 2
- 102000003676 Glucocorticoid Receptors Human genes 0.000 abstract 1
- 108090000079 Glucocorticoid Receptors Proteins 0.000 abstract 1
- 230000003042 antagnostic effect Effects 0.000 abstract 1
- 230000001363 autoimmune Effects 0.000 abstract 1
- 208000027866 inflammatory disease Diseases 0.000 abstract 1
- 230000002401 inhibitory effect Effects 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 230000000754 repressing effect Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Rheumatology (AREA)
- Pain & Pain Management (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Steroid Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US2394798A | 1998-02-13 | 1998-02-13 | |
| US24783199A | 1999-02-10 | 1999-02-10 | |
| PCT/US1999/003127 WO1999041256A1 (en) | 1998-02-13 | 1999-02-12 | Glucocorticoid-selective anti-inflammatory agents |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| NO20004053D0 true NO20004053D0 (no) | 2000-08-11 |
| NO20004053L NO20004053L (no) | 2000-09-11 |
Family
ID=26697833
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20004053A NO20004053L (no) | 1998-02-13 | 2000-08-11 | Glukokortikoid-selektive antiinflammatoriske midler |
Country Status (20)
| Country | Link |
|---|---|
| EP (1) | EP1053239B1 (no) |
| JP (1) | JP2002503665A (no) |
| KR (1) | KR20010040935A (no) |
| CN (1) | CN1119348C (no) |
| AT (1) | ATE230749T1 (no) |
| AU (1) | AU766441B2 (no) |
| BG (1) | BG64317B1 (no) |
| BR (1) | BR9907788A (no) |
| CA (1) | CA2320943A1 (no) |
| DE (1) | DE69904804T2 (no) |
| DK (1) | DK1053239T3 (no) |
| ES (1) | ES2192035T3 (no) |
| HU (1) | HUP0100460A3 (no) |
| IL (1) | IL137508A0 (no) |
| NO (1) | NO20004053L (no) |
| NZ (1) | NZ506013A (no) |
| PL (1) | PL193323B1 (no) |
| SK (1) | SK284689B6 (no) |
| TR (1) | TR200003094T2 (no) |
| WO (1) | WO1999041256A1 (no) |
Families Citing this family (30)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6506766B1 (en) | 1998-02-13 | 2003-01-14 | Abbott Laboratories | Glucocortiocoid-selective antinflammatory agents |
| CO5180649A1 (es) * | 1999-09-01 | 2002-07-30 | Abbott Lab | Antagonistas de los receptores de los glucocorticoides para el tratamiento de la diabetes para el tratamiento de la diabetes |
| US6593480B2 (en) | 1999-09-01 | 2003-07-15 | Abbott Laboratories | Glucocorticoid receptor antagonists for treatment of diabetes |
| US6329534B1 (en) | 1999-09-01 | 2001-12-11 | Abbott Laboratories | Glucocorticoid receptor antagonists for treatment of diabetes |
| US6436986B1 (en) | 1999-09-01 | 2002-08-20 | Abbott Laboratories | Glucocorticoid receptor antagonists for treatment of diabetes |
| ES2246292T3 (es) | 2000-10-30 | 2006-02-16 | Pfizer Products Inc. | Moduladores de receptor glucocorticoide. |
| WO2003002548A1 (en) * | 2001-06-29 | 2003-01-09 | Abbott Laboratories | A process for the preparation of chiral glucocorticoid receptor agents |
| US6608216B2 (en) | 2001-06-29 | 2003-08-19 | Abbott Laboratories | Process for the preparation of chiral glucocorticoid receptor agents |
| US6518430B1 (en) * | 2001-09-21 | 2003-02-11 | Abbott Laboratories | Process for the preparation of 5-(substituted)-10-methoxy-2,2,4-trimethyl-2,5-dihydro-1H-chromeno[3,4-F]quinolines and derivatives thereof |
| AU2003202216A1 (en) | 2002-01-14 | 2003-07-30 | Boehringer Ingelheim Pharmaceuticals, Inc. | Glucocorticoid mimetics, methods of making them, pharmaceutical formulations containing them and uses thereof |
| WO2003082787A1 (en) | 2002-03-26 | 2003-10-09 | Boehringer Ingelheim Pharmaceuticals, Inc. | Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof |
| CA2478156C (en) | 2002-03-26 | 2011-02-15 | Boehringer Ingelheim Pharmaceuticals, Inc. | Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof |
| EP1496892B1 (en) | 2002-04-11 | 2011-01-26 | Merck Sharp & Dohme Corp. | 1h-benzo(f)indazol-5-yl derivatives as selective glucocorticoid receptor modulators |
| US7186864B2 (en) | 2002-05-29 | 2007-03-06 | Boehringer Ingelheim Pharmaceuticals, Inc. | Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof |
| US7074806B2 (en) | 2002-06-06 | 2006-07-11 | Boehringer Ingelheim Pharmaceuticals, Inc. | Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof |
| JP2006504678A (ja) | 2002-08-21 | 2006-02-09 | ベーリンガー インゲルハイム ファーマシューティカルズ インコーポレイテッド | グルココルチコイドミメチックス、その製造方法、その医薬組成物、及び使用 |
| AU2003258050A1 (en) | 2002-10-11 | 2004-05-04 | Ligand Pharmaceuticals Incorporated | 5-cycloalkenyl 5h-chromeno(3,4-f)quinoline derivatives as selective progesterone receptor modulator compounds |
| DE20301728U1 (de) | 2002-10-11 | 2004-03-11 | Ligand Pharmaceuticals, Inc., San Diego | 5-substituierte 7,9-Difluor-5H-Chromeno(3,4-f) -Chinolin-Verbindungen als selektive Progesteronrezeptormodulator-Verbindungen |
| CA2501833A1 (en) | 2002-10-11 | 2004-04-22 | Ligand Pharmaceuticals Incorporated | 5-(1',1'-cycloalkyl/alkenyl)methylidene 1,2-dihydro-5h-chromeno[3,4-f]quinolines as selective progesterone receptor modulator compounds |
| CA2512257A1 (en) | 2003-01-03 | 2004-07-29 | Boehringer Ingelheim Pharmaceuticals, Inc. | 1-propanol and 1-propylamine derivatives and their use as glucocorticoid ligands |
| US20070088042A1 (en) | 2004-09-09 | 2007-04-19 | Meissner Robert S | Fluorinated 4-azasteroid derivatives as androgen receptor modulators |
| US7235662B2 (en) | 2003-06-11 | 2007-06-26 | Bristol-Myers Squibb Company | Modulators of the glucocorticoid receptor and method |
| US8097606B2 (en) | 2003-07-23 | 2012-01-17 | Corcept Therapeutics, Inc. | Antiglucocorticoids for the treatment of catatonia |
| UY28526A1 (es) | 2003-09-24 | 2005-04-29 | Boehringer Ingelheim Pharma | Miméticos de glucocorticoides, métodos de preparación composiciones farmacéuticas y usos de los mismos |
| US7507843B2 (en) | 2003-10-16 | 2009-03-24 | Boehringer Ingelheim Pharmaceuticals, Inc. | Stereoselective synthesis of certain trifluoromethyl-substituted alcohols |
| US7795272B2 (en) | 2004-03-13 | 2010-09-14 | Boehringer Ingelheim Pharmaceutical, Inc. | Glucocorticoid mimetics, methods of making them, pharmaceutical compositions and uses thereof |
| CA2592514A1 (en) | 2004-12-27 | 2006-07-06 | Boehringer Ingelheim Pharmaceuticals, Inc. | Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof |
| PL1944290T3 (pl) * | 2005-09-14 | 2014-07-31 | Ayumi Pharmaceutical Corp | Nowa pochodna 1-2-dihydrochinoliny mająca aktywność wiązania glukokortykoidowego receptora |
| CN102834406A (zh) | 2009-06-16 | 2012-12-19 | 默沙东公司 | 作为糖皮质激素受体激动剂的新的[3.2-c]杂芳基甾体、其组合物和用途 |
| US20120220590A1 (en) | 2009-07-31 | 2012-08-30 | Thombare Pravin S | Novel compounds as modulators of glucocorticoid receptors |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1043325B1 (en) * | 1994-12-22 | 2004-06-16 | Ligand Pharmaceuticals Incorporated | Steroid receptor modulator compounds and methods |
-
1999
- 1999-02-12 BR BR9907788-4A patent/BR9907788A/pt not_active Application Discontinuation
- 1999-02-12 KR KR1020007008850A patent/KR20010040935A/ko not_active Ceased
- 1999-02-12 PL PL343018A patent/PL193323B1/pl not_active IP Right Cessation
- 1999-02-12 HU HU0100460A patent/HUP0100460A3/hu unknown
- 1999-02-12 TR TR2000/03094T patent/TR200003094T2/xx unknown
- 1999-02-12 SK SK1197-2000A patent/SK284689B6/sk unknown
- 1999-02-12 ES ES99906996T patent/ES2192035T3/es not_active Expired - Lifetime
- 1999-02-12 AU AU26773/99A patent/AU766441B2/en not_active Ceased
- 1999-02-12 DE DE69904804T patent/DE69904804T2/de not_active Expired - Lifetime
- 1999-02-12 WO PCT/US1999/003127 patent/WO1999041256A1/en not_active Ceased
- 1999-02-12 CN CN99804902A patent/CN1119348C/zh not_active Expired - Fee Related
- 1999-02-12 DK DK99906996T patent/DK1053239T3/da active
- 1999-02-12 AT AT99906996T patent/ATE230749T1/de active
- 1999-02-12 IL IL13750899A patent/IL137508A0/xx unknown
- 1999-02-12 JP JP2000531449A patent/JP2002503665A/ja active Pending
- 1999-02-12 EP EP99906996A patent/EP1053239B1/en not_active Expired - Lifetime
- 1999-02-12 CA CA002320943A patent/CA2320943A1/en not_active Abandoned
- 1999-02-12 NZ NZ506013A patent/NZ506013A/xx unknown
-
2000
- 2000-08-11 NO NO20004053A patent/NO20004053L/no not_active Application Discontinuation
- 2000-08-28 BG BG104719A patent/BG64317B1/bg unknown
Also Published As
| Publication number | Publication date |
|---|---|
| DK1053239T3 (da) | 2003-04-22 |
| DE69904804D1 (de) | 2003-02-13 |
| HUP0100460A3 (en) | 2003-03-28 |
| HK1033308A1 (en) | 2001-08-24 |
| CN1296486A (zh) | 2001-05-23 |
| TR200003094T2 (tr) | 2001-01-22 |
| SK11972000A3 (sk) | 2001-08-06 |
| BR9907788A (pt) | 2001-10-30 |
| CA2320943A1 (en) | 1999-09-19 |
| IL137508A0 (en) | 2001-07-24 |
| PL193323B1 (pl) | 2007-02-28 |
| SK284689B6 (sk) | 2005-09-08 |
| HUP0100460A2 (hu) | 2001-09-28 |
| CN1119348C (zh) | 2003-08-27 |
| NO20004053L (no) | 2000-09-11 |
| BG64317B1 (bg) | 2004-09-30 |
| AU2677399A (en) | 1999-08-30 |
| EP1053239B1 (en) | 2003-01-08 |
| DE69904804T2 (de) | 2003-11-06 |
| JP2002503665A (ja) | 2002-02-05 |
| NZ506013A (en) | 2003-03-28 |
| EP1053239A1 (en) | 2000-11-22 |
| KR20010040935A (ko) | 2001-05-15 |
| ES2192035T3 (es) | 2003-09-16 |
| ATE230749T1 (de) | 2003-01-15 |
| WO1999041256A1 (en) | 1999-08-19 |
| BG104719A (en) | 2001-05-31 |
| AU766441B2 (en) | 2003-10-16 |
| PL343018A1 (en) | 2001-07-30 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FC2A | Withdrawal, rejection or dismissal of laid open patent application |