NO20004350D0 - Preparat med vedvarende frigivinng av AII-antagonist, fremstilling og anvendelse herav - Google Patents

Preparat med vedvarende frigivinng av AII-antagonist, fremstilling og anvendelse herav

Info

Publication number: NO20004350D0
Authority: NO; Norway
Prior art keywords: preparation; sustained release; aii antagonist; angiotensin; antagonistic activity
Prior art date: 1998-03-04

Application number

NO20004350A

Other languages

English (en)

Other versions

NO20004350L (no

Inventor

Yasutaka Igari

Akira Saikawa

Yoshiyuki Inada

Shigeru Kamei

Original Assignee

Takeda Chemical Industries Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1998-03-04

Filing date

2000-09-01

Publication date

2000-09-01

2000-09-01 Application filed by Takeda Chemical Industries Ltd filed Critical Takeda Chemical Industries Ltd

2000-09-01 Publication of NO20004350D0 publication Critical patent/NO20004350D0/no

2000-10-03 Publication of NO20004350L publication Critical patent/NO20004350L/no

Links

239000005557 antagonist Substances 0.000 title 1
238000013268 sustained release Methods 0.000 title 1
239000012730 sustained-release form Substances 0.000 title 1
102000005862 Angiotensin II Human genes 0.000 abstract 2
101800000733 Angiotensin-2 Proteins 0.000 abstract 2
CZGUSIXMZVURDU-JZXHSEFVSA-N Ile(5)-angiotensin II Chemical compound C([C@@H](C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CC=1NC=NC=1)C(=O)N1[C@@H](CCC1)C(=O)N[C@@H](CC=1C=CC=CC=1)C([O-])=O)NC(=O)[C@@H](NC(=O)[C@H](CCCNC(N)=[NH2+])NC(=O)[C@@H]([NH3+])CC([O-])=O)C(C)C)C1=CC=C(O)C=C1 CZGUSIXMZVURDU-JZXHSEFVSA-N 0.000 abstract 2
229950006323 angiotensin ii Drugs 0.000 abstract 2
230000003042 antagnostic effect Effects 0.000 abstract 2
229920002988 biodegradable polymer Polymers 0.000 abstract 1
239000004621 biodegradable polymer Substances 0.000 abstract 1
230000036772 blood pressure Effects 0.000 abstract 1
230000027288 circadian rhythm Effects 0.000 abstract 1
150000001875 compounds Chemical class 0.000 abstract 1
239000003405 delayed action preparation Substances 0.000 abstract 1
239000002184 metal Substances 0.000 abstract 1
229940002612 prodrug Drugs 0.000 abstract 1
239000000651 prodrug Substances 0.000 abstract 1
150000003839 salts Chemical class 0.000 abstract 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4184—1,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1611—Inorganic compounds
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1629—Organic macromolecular compounds
- A61K9/1641—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, poloxamers
- A61K9/1647—Polyesters, e.g. poly(lactide-co-glycolide)
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Epidemiology (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Inorganic Chemistry (AREA)
Heart & Thoracic Surgery (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Organic Chemistry (AREA)
Cardiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Medicinal Preparation (AREA)
Plural Heterocyclic Compounds (AREA)
Preparation Of Compounds By Using Micro-Organisms (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

NO20004350A 1998-03-04 2000-09-01 Preparat med vedvarende frigivinng av AII-antagonist, fremstilling og anvendelse herav NO20004350L (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
JP5236698		1998-03-04
PCT/JP1999/001011 WO1999044590A1 (en)	1998-03-04	1999-03-03	Sustained-release preparation for aii antagonist, production and use thereof

Publications (2)

Publication Number	Publication Date
NO20004350D0 true NO20004350D0 (no)	2000-09-01
NO20004350L NO20004350L (no)	2000-10-03

Family

ID=12912818

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO20004350A NO20004350L (no)	1998-03-04	2000-09-01	Preparat med vedvarende frigivinng av AII-antagonist, fremstilling og anvendelse herav

Country Status (21)

Country	Link
US (2)	US6589547B1 (no)
EP (1)	EP1058541B1 (no)
KR (1)	KR20010086245A (no)
CN (1)	CN1291888A (no)
AT (1)	ATE258430T1 (no)
AU (1)	AU2745199A (no)
BR (1)	BR9908474A (no)
CA (1)	CA2318446C (no)
DE (1)	DE69914460T2 (no)
EE (1)	EE200000499A (no)
ES (1)	ES2214013T3 (no)
HU (1)	HUP0101439A3 (no)
ID (1)	ID25640A (no)
IL (1)	IL137979A0 (no)
LT (1)	LT4800B (no)
LV (1)	LV12585B (no)
NO (1)	NO20004350L (no)
PL (1)	PL342684A1 (no)
SK (1)	SK11902000A3 (no)
WO (1)	WO1999044590A1 (no)
ZA (1)	ZA991706B (no)

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US20030187038A1 (en) *	2000-08-25	2003-10-02	Yoshimi Imura	Fibrinogen-lowering agents
AU2002210925A1 (en) *	2000-10-25	2002-05-06	Takeda Chemical Industries Ltd.	Preventives/remedies for portal hypertension
US20040121008A1 (en) *	2001-03-16	2004-06-24	Keiko Shiraishi	Process for producing sustained release preparation
EP1413315A4 (en) *	2001-08-03	2006-08-16	Takeda Pharmaceutical	DRUGS WITH CONTINUOUS RELEASE
BRPI0105509B8 (pt) *	2001-11-05	2021-05-25	Univ Minas Gerais	formulações do peptídeo angiotensina-(1-7) usando as ciclodextrinas, lipossomas e o polímero plga
EP1444988A4 (en) *	2001-11-13	2007-04-25	Takeda Pharmaceutical	CANCER AGENT
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US7407778B2 (en) *	2002-02-07	2008-08-05	Pettegrew Jay W	Compounds, compositions and methods for treating neuropsychiatric disorders
US7700074B2 (en) *	2002-02-07	2010-04-20	Pettegrew Jay W	Method and system for diagnosis of neuropsychiatric disorders including chronic alcoholism
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US7815894B2 (en) *	2003-05-29	2010-10-19	Jay W. Pettegrew	Compounds, compositions and methods for medical imaging of neuropsychiatric disorders
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EP1806137A4 (en) *	2004-10-29	2011-03-30	Kowa Co	THERAPEUTIC AGENT FOR THE TREATMENT OF GLOMERULAR DISEASE
CA2598410A1 (fr) *	2005-02-21	2006-08-24	Flamel Technologies	Forme pharmaceutique orale de losartan
AR055755A1 (es) *	2005-03-30	2007-09-05	Takeda Pharmaceutical	Derivado de bencimidazol, procesos de obtencion, composiciones farmaceuticas y usos.
DE602006008962D1 (de) *	2005-08-22	2010-07-08	Alembic Ltd	Verfahren zur herstellung von valsartan
CN102813635A (zh) *	2006-08-10	2012-12-12	武田药品工业株式会社	药物组合物
EP1897537A1 (en) *	2006-09-04	2008-03-12	Novartis AG	Composition comprising an angiotensin II receptor antagonist
PE20081364A1 (es) *	2006-09-04	2008-12-04	Novartis Ag	Composicion farmaceutica que comprende valsartan
EP1908469A1 (en)	2006-10-06	2008-04-09	Boehringer Ingelheim Vetmedica Gmbh	Angiotensin II receptor antagonist for the treatment of systemic diseases in cats
MY148370A (en)	2006-12-18	2013-04-15	Takeda Pharmaceutical	Sustained-release composition and method for producing the same
CN101011393B (zh) *	2007-02-16	2010-10-06	广州柏赛罗药业有限公司	厄贝沙坦胃内滞留型缓释药物组合物
TWI415634B (zh) *	2007-03-28	2013-11-21	Takeda Pharmaceutical	固態醫藥組成物
KR101209319B1 (ko) *	2008-04-29	2012-12-06	한올바이오파마주식회사	안지오텐신-ⅱ-수용체 차단제를 포함하는 약제학적 제제
AU2010251194B2 (en)	2009-05-20	2016-02-25	Boehringer Ingelheim Vetmedica Gmbh	Pharmaceutical oral telmisartan solution
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WO1999044590A1 (en) *	1998-03-04	1999-09-10	Takeda Chemical Industries, Ltd.	Sustained-release preparation for aii antagonist, production and use thereof

1999
- 1999-03-03 WO PCT/JP1999/001011 patent/WO1999044590A1/en not_active Ceased
- 1999-03-03 IL IL13797999A patent/IL137979A0/xx unknown
- 1999-03-03 AU AU27451/99A patent/AU2745199A/en not_active Abandoned
- 1999-03-03 HU HU0101439A patent/HUP0101439A3/hu unknown
- 1999-03-03 SK SK1190-2000A patent/SK11902000A3/sk unknown
- 1999-03-03 DE DE69914460T patent/DE69914460T2/de not_active Expired - Lifetime
- 1999-03-03 CN CN99803444A patent/CN1291888A/zh active Pending
- 1999-03-03 EE EEP200000499A patent/EE200000499A/xx unknown
- 1999-03-03 AT AT99907846T patent/ATE258430T1/de not_active IP Right Cessation
- 1999-03-03 PL PL99342684A patent/PL342684A1/xx unknown
- 1999-03-03 BR BR9908474-0A patent/BR9908474A/pt not_active IP Right Cessation
- 1999-03-03 KR KR1020007008919A patent/KR20010086245A/ko not_active Abandoned
- 1999-03-03 EP EP99907846A patent/EP1058541B1/en not_active Expired - Lifetime
- 1999-03-03 ID IDW20001680A patent/ID25640A/id unknown
- 1999-03-03 ES ES99907846T patent/ES2214013T3/es not_active Expired - Lifetime
- 1999-03-03 ZA ZA9901706A patent/ZA991706B/xx unknown
- 1999-03-03 CA CA002318446A patent/CA2318446C/en not_active Expired - Fee Related
- 1999-03-09 US US09/601,986 patent/US6589547B1/en not_active Expired - Fee Related
2000
- 2000-08-16 LV LVP-00-110A patent/LV12585B/en unknown
- 2000-08-31 LT LT2000082A patent/LT4800B/lt not_active IP Right Cessation
- 2000-09-01 NO NO20004350A patent/NO20004350L/no unknown
2003
- 2003-05-22 US US10/443,308 patent/US7294344B2/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
KR20010086245A (ko)	2001-09-10
US6589547B1 (en)	2003-07-08
CA2318446C (en)	2008-09-23
DE69914460D1 (de)	2004-03-04
EP1058541B1 (en)	2004-01-28
HUP0101439A2 (hu)	2001-10-28
LV12585A (en)	2000-12-20
AU2745199A (en)	1999-09-20
LV12585B (en)	2001-03-20
ZA991706B (en)	2000-10-03
HUP0101439A3 (en)	2002-09-30
ID25640A (id)	2000-10-19
WO1999044590A1 (en)	1999-09-10
PL342684A1 (en)	2001-07-02
US7294344B2 (en)	2007-11-13
LT4800B (lt)	2001-06-25
ES2214013T3 (es)	2004-09-01
US20030198676A1 (en)	2003-10-23
LT2000082A (en)	2001-03-26
BR9908474A (pt)	2000-12-05
CA2318446A1 (en)	1999-09-10
EE200000499A (et)	2002-02-15
EP1058541A1 (en)	2000-12-13
CN1291888A (zh)	2001-04-18
DE69914460T2 (de)	2004-10-28
NO20004350L (no)	2000-10-03
IL137979A0 (en)	2001-10-31
ATE258430T1 (de)	2004-02-15
SK11902000A3 (sk)	2001-02-12

Publication	Publication Date	Title
ID25640A (id)	2000-10-19	Preparat pelepasan terus menerus untuk antagonistik aii, produksi dan penggunaannya
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