NO20005551L - 2"-deoksyhygromycinderivater - Google Patents
2"-deoksyhygromycinderivaterInfo
- Publication number
- NO20005551L NO20005551L NO20005551A NO20005551A NO20005551L NO 20005551 L NO20005551 L NO 20005551L NO 20005551 A NO20005551 A NO 20005551A NO 20005551 A NO20005551 A NO 20005551A NO 20005551 L NO20005551 L NO 20005551L
- Authority
- NO
- Norway
- Prior art keywords
- compounds
- formula
- infections
- protozoal infections
- deoksyhygromycinderivater
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 abstract 4
- 206010037075 Protozoal infections Diseases 0.000 abstract 2
- 230000001580 bacterial effect Effects 0.000 abstract 2
- 208000035143 Bacterial infection Diseases 0.000 abstract 1
- 239000003242 anti bacterial agent Substances 0.000 abstract 1
- 230000000844 anti-bacterial effect Effects 0.000 abstract 1
- 239000003904 antiprotozoal agent Substances 0.000 abstract 1
- 208000022362 bacterial infectious disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 208000035475 disorder Diseases 0.000 abstract 1
- 208000015181 infectious disease Diseases 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 239000000651 prodrug Substances 0.000 abstract 1
- 229940002612 prodrug Drugs 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 239000012453 solvate Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/20—Carbocyclic rings
- C07H15/203—Monocyclic carbocyclic rings other than cyclohexane rings; Bicyclic carbocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/26—Acyclic or carbocyclic radicals, substituted by hetero rings
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biotechnology (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Biochemistry (AREA)
- Engineering & Computer Science (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Tropical Medicine & Parasitology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
Abstract
Det er beskrevet forbindelser ifølge formel (I) og farmasøytisk akseptable salter, promedikamenter og solvater derav, hvori Rog R2 er som definert heri. Forbindelser ifølge formel (I) er antibakterielle og antiprotozomidler som kan bli anvendt for å behandle forskjellige bakterielle og protozoinfeksjoner og forstyrrelser relatert til slike infeksjoner. Det er videre beskrevet farmasøytiske sammensetninger inneholdendeforbindelsene ifølge formel (I) og fremgangs-måter for behandling av bakterielle protozoinfeksjoner ved administrering av. " forbindelsene ifølge formel (I).
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US8405898P | 1998-05-04 | 1998-05-04 | |
| PCT/IB1999/000611 WO1999057127A1 (en) | 1998-05-04 | 1999-04-08 | 2'-deoxy hygromycin derivatives |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| NO20005551D0 NO20005551D0 (no) | 2000-11-03 |
| NO20005551L true NO20005551L (no) | 2001-01-02 |
Family
ID=22182624
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20005551A NO20005551L (no) | 1998-05-04 | 2000-11-03 | 2"-deoksyhygromycinderivater |
Country Status (38)
| Country | Link |
|---|---|
| US (1) | US6342497B1 (no) |
| EP (1) | EP1077984B1 (no) |
| JP (1) | JP2002513798A (no) |
| KR (1) | KR100396099B1 (no) |
| CN (1) | CN1299367A (no) |
| AP (1) | AP1069A (no) |
| AR (1) | AR015776A1 (no) |
| AT (1) | ATE243218T1 (no) |
| AU (1) | AU762302B2 (no) |
| BG (1) | BG104995A (no) |
| BR (1) | BR9910232A (no) |
| CA (1) | CA2331261C (no) |
| DE (1) | DE69908936T2 (no) |
| DK (1) | DK1077984T3 (no) |
| DZ (1) | DZ2779A1 (no) |
| EA (1) | EA004374B1 (no) |
| ES (1) | ES2199559T3 (no) |
| GT (1) | GT199900058A (no) |
| HN (1) | HN1999000064A (no) |
| HR (1) | HRP20000748A2 (no) |
| HU (1) | HUP0102412A3 (no) |
| ID (1) | ID26368A (no) |
| IL (1) | IL139020A0 (no) |
| IS (1) | IS5680A (no) |
| MA (1) | MA26626A1 (no) |
| NO (1) | NO20005551L (no) |
| NZ (1) | NZ507450A (no) |
| OA (1) | OA11507A (no) |
| PA (1) | PA8471901A1 (no) |
| PE (1) | PE20000440A1 (no) |
| PL (1) | PL344085A1 (no) |
| PT (1) | PT1077984E (no) |
| SK (1) | SK16442000A3 (no) |
| TN (1) | TNSN99084A1 (no) |
| TR (1) | TR200003249T2 (no) |
| WO (1) | WO1999057127A1 (no) |
| YU (1) | YU64300A (no) |
| ZA (1) | ZA993063B (no) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PL348063A1 (en) * | 1998-12-02 | 2002-05-06 | Pfizer Prod Inc | Hygromycin a derivatives as antibacterial agents |
| GB9923078D0 (en) * | 1999-09-29 | 1999-12-01 | Phytopharm Plc | Sapogenin derivatives and their use |
| CN1432019A (zh) * | 2000-06-02 | 2003-07-23 | 辉瑞产品公司 | 用于治疗细菌和原生动物感染的潮霉素a衍生物 |
| CN102168034B (zh) * | 2010-11-29 | 2012-12-05 | 中国科学院南海海洋研究所 | 一种海洋链霉菌以及利用该菌制备替达霉素a和b的方法 |
| EP3840743A4 (en) | 2018-08-20 | 2022-08-17 | Northeastern University | HYGROMYCIN-A COMPOUNDS AND METHODS OF TREATMENT OF SPIROCHETARY DISEASES |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2832356B2 (ja) * | 1988-03-31 | 1998-12-09 | 武田薬品工業株式会社 | ハイグロマイシン類の合成中間体および製造法 |
-
1999
- 1999-04-08 AT AT99909164T patent/ATE243218T1/de not_active IP Right Cessation
- 1999-04-08 BR BR9910232-3A patent/BR9910232A/pt not_active IP Right Cessation
- 1999-04-08 NZ NZ507450A patent/NZ507450A/en unknown
- 1999-04-08 HU HU0102412A patent/HUP0102412A3/hu unknown
- 1999-04-08 CN CN99805810A patent/CN1299367A/zh active Pending
- 1999-04-08 DK DK99909164T patent/DK1077984T3/da active
- 1999-04-08 KR KR10-2000-7012222A patent/KR100396099B1/ko not_active Expired - Fee Related
- 1999-04-08 WO PCT/IB1999/000611 patent/WO1999057127A1/en not_active Ceased
- 1999-04-08 ES ES99909164T patent/ES2199559T3/es not_active Expired - Lifetime
- 1999-04-08 ID IDW20002256A patent/ID26368A/id unknown
- 1999-04-08 YU YU64300A patent/YU64300A/sh unknown
- 1999-04-08 EA EA200001028A patent/EA004374B1/ru not_active IP Right Cessation
- 1999-04-08 EP EP99909164A patent/EP1077984B1/en not_active Expired - Lifetime
- 1999-04-08 DE DE69908936T patent/DE69908936T2/de not_active Expired - Fee Related
- 1999-04-08 JP JP2000547096A patent/JP2002513798A/ja active Pending
- 1999-04-08 PL PL99344085A patent/PL344085A1/xx unknown
- 1999-04-08 HR HR20000748A patent/HRP20000748A2/hr not_active Application Discontinuation
- 1999-04-08 SK SK1644-2000A patent/SK16442000A3/sk unknown
- 1999-04-08 AU AU28508/99A patent/AU762302B2/en not_active Ceased
- 1999-04-08 US US09/380,718 patent/US6342497B1/en not_active Expired - Fee Related
- 1999-04-08 IL IL13902099A patent/IL139020A0/xx unknown
- 1999-04-08 CA CA002331261A patent/CA2331261C/en not_active Expired - Fee Related
- 1999-04-08 PT PT99909164T patent/PT1077984E/pt unknown
- 1999-04-08 TR TR2000/03249T patent/TR200003249T2/xx unknown
- 1999-04-16 GT GT199900058A patent/GT199900058A/es unknown
- 1999-04-29 PE PE1999000355A patent/PE20000440A1/es not_active Application Discontinuation
- 1999-04-29 AP APAP/P/1999/001525A patent/AP1069A/en active
- 1999-04-30 AR ARP990102023A patent/AR015776A1/es not_active Application Discontinuation
- 1999-05-03 HN HN1999000064A patent/HN1999000064A/es unknown
- 1999-05-03 DZ DZ990079A patent/DZ2779A1/xx active
- 1999-05-03 TN TNTNSN99084A patent/TNSN99084A1/fr unknown
- 1999-05-03 ZA ZA9903063A patent/ZA993063B/xx unknown
- 1999-05-03 MA MA25566A patent/MA26626A1/fr unknown
- 1999-05-04 PA PA19998471901A patent/PA8471901A1/es unknown
-
2000
- 2000-10-24 IS IS5680A patent/IS5680A/is unknown
- 2000-10-27 OA OA1200000298A patent/OA11507A/en unknown
- 2000-11-03 NO NO20005551A patent/NO20005551L/no not_active Application Discontinuation
- 2000-11-28 BG BG104995A patent/BG104995A/bg unknown
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FC2A | Withdrawal, rejection or dismissal of laid open patent application |