NO20013150L - Fremgangsmate ved fremstilling av 5-cyanftalid - Google Patents

Fremgangsmate ved fremstilling av 5-cyanftalid

Info

Publication number
NO20013150L
NO20013150L NO20013150A NO20013150A NO20013150L NO 20013150 L NO20013150 L NO 20013150L NO 20013150 A NO20013150 A NO 20013150A NO 20013150 A NO20013150 A NO 20013150A NO 20013150 L NO20013150 L NO 20013150L
Authority
NO
Norway
Prior art keywords
cyanophthalide
preparing
Prior art date
Application number
NO20013150A
Other languages
English (en)
Other versions
NO20013150D0 (no
NO326516B1 (no
Inventor
Hans Petersen
Poul Dahlberg Nielsen
Original Assignee
Lundbeck & Co As H
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lundbeck & Co As H filed Critical Lundbeck & Co As H
Publication of NO20013150D0 publication Critical patent/NO20013150D0/no
Publication of NO20013150L publication Critical patent/NO20013150L/no
Publication of NO326516B1 publication Critical patent/NO326516B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/87—Benzo [c] furans; Hydrogenated benzo [c] furans
    • C07D307/88—Benzo [c] furans; Hydrogenated benzo [c] furans with one oxygen atom directly attached in position 1 or 3

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Indole Compounds (AREA)
  • Furan Compounds (AREA)
NO20013150A 1998-12-23 2001-06-22 Fremgangsmate ved fremstilling av 5-cyanftalid NO326516B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DKPA199801718 1998-12-23
PCT/DK1999/000728 WO2000039112A1 (en) 1998-12-23 1999-12-22 Method for the preparation of 5-cyanophthalide

Publications (3)

Publication Number Publication Date
NO20013150D0 NO20013150D0 (no) 2001-06-22
NO20013150L true NO20013150L (no) 2001-08-20
NO326516B1 NO326516B1 (no) 2008-12-22

Family

ID=8107494

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20013150A NO326516B1 (no) 1998-12-23 2001-06-22 Fremgangsmate ved fremstilling av 5-cyanftalid

Country Status (31)

Country Link
US (1) US6392060B2 (no)
EP (1) EP1140886B1 (no)
JP (1) JP2002533450A (no)
KR (1) KR100454008B1 (no)
CN (1) CN1149208C (no)
AR (1) AR019791A1 (no)
AT (1) ATE236145T1 (no)
AU (1) AU764161B2 (no)
BG (1) BG64986B1 (no)
BR (1) BR9916955A (no)
CA (1) CA2356188C (no)
CZ (1) CZ300408B6 (no)
DE (1) DE69906580T2 (no)
DK (1) DK1140886T3 (no)
EA (1) EA003057B1 (no)
ES (1) ES2195644T3 (no)
HK (1) HK1043130B (no)
HU (1) HUP0104856A3 (no)
IL (1) IL143422A0 (no)
IS (1) IS2261B (no)
IT (1) IT1315269B1 (no)
NO (1) NO326516B1 (no)
NZ (1) NZ512073A (no)
PL (1) PL203275B1 (no)
PT (1) PT1140886E (no)
SI (1) SI1140886T1 (no)
SK (1) SK285530B6 (no)
TR (1) TR200101796T2 (no)
UA (1) UA70979C2 (no)
WO (1) WO2000039112A1 (no)
ZA (1) ZA200104262B (no)

Families Citing this family (28)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL199423B1 (pl) 1998-10-20 2008-09-30 Lundbeck & Co As H Sposób wytwarzania citalopramu
CN1149208C (zh) 1998-12-23 2004-05-12 H.隆德贝克有限公司 制备5-氰基2-苯并[c]呋喃酮的方法
AR022329A1 (es) * 1999-01-29 2002-09-04 Lundbeck & Co As H Metodo para la preparacion de 5-cianoftalida
NZ514671A (en) 1999-04-14 2003-10-31 H Method for the preparation of citalopram
ITMI991581A1 (it) * 1999-06-25 2001-01-15 Lundbeck & Co As H Metodo per la preparazione di citalopram
ITMI991579A1 (it) 1999-06-25 2001-01-15 Lundbeck & Co As H Metodo per la preparazione di citalopram
CH692298A5 (de) 1999-10-25 2002-04-30 Lundbeck & Co As H Verfahren zur Herstellung von Zwischenstufen für die Citalopramsynthese sowie zur Herstellung von Escitalopram.
EP1298124B1 (en) 1999-10-25 2007-02-28 H. Lundbeck A/S Method For the Preparation of Citalopram
AR026063A1 (es) 1999-11-01 2002-12-26 Lundbeck & Co As H Metodo para la preparacion de 5-carboxiftalida.
EA004742B1 (ru) 1999-12-28 2004-08-26 Х.Лундбекк А/С Способ получения циталопрама
WO2001049672A1 (en) 1999-12-30 2001-07-12 H. Lundbeck A/S Method for the preparation of citalopram
TR200201783T2 (tr) 2000-01-14 2002-12-23 H. Lundbeck A/S 5-Siyanofatalid hazırlamak için yöntem
NL1017415C1 (nl) 2000-02-24 2001-05-18 Lundbeck & Co As H Werkwijze voor de bereiding van Citalopram.
NL1017417C1 (nl) 2000-03-03 2001-03-16 Lundbeck & Co As H Werkwijze voor de bereiding van Citalopram.
NL1017500C1 (nl) 2000-03-13 2001-04-26 Lundbeck & Co As H Werkwijze voor de bereiding van Citalopram.
CZ20023100A3 (cs) * 2000-03-13 2003-02-12 H. Lundbeck A/S Způsob výroby citalopramu
KR20020080481A (ko) 2000-03-13 2002-10-23 하. 룬트벡 아크티에 셀스카브 시탈로프람의 제조 방법
SK14512002A3 (sk) 2000-03-14 2003-03-04 H. Lundbeck A/S Spôsob výroby citalopramu, medziprodukt a citalopram výrobený týmto spôsobom
EP1274699A1 (en) * 2000-03-16 2003-01-15 H. Lundbeck A/S Method for the preparation of 5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofurans
AR032455A1 (es) 2000-05-12 2003-11-12 Lundbeck & Co As H Metodo para la preparacion de citalopram, un intermediario empleado en el metodo, un metodo para la preparacion del intermediario empleado en el metodo y composicion farmaceutica antidepresiva
IL144817A0 (en) * 2000-08-18 2002-06-30 Lundbeck & Co As H Method for the preparation of citalopram
JP3798982B2 (ja) 2000-12-22 2006-07-19 ハー・ルンドベック・アクチエゼルスカベット 純粋なシタロプラムの製造方法
CA2359810C (en) 2000-12-28 2002-11-05 H. Lundbeck A/S Process for the preparation of pure citalopram
EP1321464A1 (en) * 2001-12-21 2003-06-25 ICROM S.p.A. Process for the preparation of 5-cyanophthalide and intermediates useful therein
CN101362743A (zh) * 2003-03-21 2009-02-11 H.隆德贝克有限公司 用于制备西酞普兰和依他普仑的中间体
TR200504022T1 (tr) * 2003-03-24 2006-08-21 Hetero Drugs Limited (S)-sitalopram oksalatın yeni sıvı kristal formları.
EP1777221A1 (en) 2005-10-14 2007-04-25 Adorkem Technology SpA Process for the preparation of 5-cyanophthalide starting from 5-carboxyphthalide
CN119775242B (zh) * 2024-12-31 2025-08-15 内蒙古源宏精细化工有限公司 合成5-氰基苯酞的方法

Family Cites Families (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1143703A (no) 1965-03-18
GB1526331A (en) 1976-01-14 1978-09-27 Kefalas As Phthalanes
GB8419963D0 (en) 1984-08-06 1984-09-12 Lundbeck & Co As H Intermediate compound and method
GB8814057D0 (en) 1988-06-14 1988-07-20 Lundbeck & Co As H New enantiomers & their isolation
DK213290D0 (da) 1990-09-06 1990-09-06 Lundbeck & Co As H Treatment of cerebrovascular disorders
DE19626659A1 (de) 1996-07-03 1998-01-08 Basf Ag Verfahren zur Herstellung von Phthaliden
DE19627697A1 (de) 1996-07-10 1998-01-15 Basf Ag Verfahren zur Herstellung von Phthaliden
ZA9711376B (en) 1996-12-20 1998-07-21 Lundbeck & Co As H Indole or dihydroindole derivatives
TR200000066T2 (tr) 1997-07-08 2000-11-21 H. Lundbeck A/S Sitalopram hazırlanması için yöntem.
UA62985C2 (en) 1997-11-10 2004-01-15 Lunnbeck As H A method for the preparation of citalopram
ES2149734T3 (es) 1997-11-11 2003-02-16 Lundbeck & Co As H Metodo para la preparacion de citalopram.
PL199423B1 (pl) 1998-10-20 2008-09-30 Lundbeck & Co As H Sposób wytwarzania citalopramu
CN1149208C (zh) 1998-12-23 2004-05-12 H.隆德贝克有限公司 制备5-氰基2-苯并[c]呋喃酮的方法
AR022329A1 (es) 1999-01-29 2002-09-04 Lundbeck & Co As H Metodo para la preparacion de 5-cianoftalida
NZ514671A (en) 1999-04-14 2003-10-31 H Method for the preparation of citalopram
ITMI991579A1 (it) 1999-06-25 2001-01-15 Lundbeck & Co As H Metodo per la preparazione di citalopram
ITMI991581A1 (it) 1999-06-25 2001-01-15 Lundbeck & Co As H Metodo per la preparazione di citalopram
CH692298A5 (de) 1999-10-25 2002-04-30 Lundbeck & Co As H Verfahren zur Herstellung von Zwischenstufen für die Citalopramsynthese sowie zur Herstellung von Escitalopram.
US6310222B1 (en) 1999-11-01 2001-10-30 Sumika Fine Chemicals Co., Ltd. Production method of 5-phthalancarbonitrile compound, intermediate therefor and production method of the intermediate

Also Published As

Publication number Publication date
DE69906580T2 (de) 2004-02-12
BG105655A (en) 2002-01-31
JP2002533450A (ja) 2002-10-08
PT1140886E (pt) 2003-08-29
ES2195644T3 (es) 2003-12-01
PL203275B1 (pl) 2009-09-30
HK1043130B (zh) 2005-03-04
AR019791A1 (es) 2002-03-13
EP1140886A1 (en) 2001-10-10
IT1315269B1 (it) 2003-02-03
IS5952A (is) 2001-05-22
US20020019546A1 (en) 2002-02-14
SI1140886T1 (en) 2003-08-31
BG64986B1 (bg) 2006-11-30
HK1043130A1 (en) 2002-09-06
DK1140886T3 (da) 2003-07-28
ZA200104262B (en) 2001-12-11
CA2356188C (en) 2006-05-23
AU764161B2 (en) 2003-08-14
EP1140886B1 (en) 2003-04-02
CA2356188A1 (en) 2000-07-06
PL348608A1 (en) 2002-06-03
HUP0104856A2 (hu) 2002-04-29
IS2261B (is) 2007-06-15
SK285530B6 (sk) 2007-03-01
CZ20012335A3 (cs) 2001-12-12
NZ512073A (en) 2003-10-31
ITMI992696A1 (it) 2001-06-23
NO20013150D0 (no) 2001-06-22
SK8962001A3 (en) 2003-03-04
CN1331686A (zh) 2002-01-16
TR200101796T2 (tr) 2001-11-21
BR9916955A (pt) 2001-09-11
ITMI992696A0 (it) 1999-12-23
EA200100696A1 (ru) 2001-12-24
WO2000039112A1 (en) 2000-07-06
EA003057B1 (ru) 2002-12-26
KR100454008B1 (ko) 2004-10-20
CZ300408B6 (cs) 2009-05-13
DE69906580D1 (de) 2003-05-08
IL143422A0 (en) 2002-04-21
UA70979C2 (uk) 2004-11-15
KR20010082370A (ko) 2001-08-29
HUP0104856A3 (en) 2003-01-28
US6392060B2 (en) 2002-05-21
NO326516B1 (no) 2008-12-22
AU1774200A (en) 2000-07-31
CN1149208C (zh) 2004-05-12
ATE236145T1 (de) 2003-04-15

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Representative=s name: PLOUGMANN & VINGTOFT, POSTBOKS 1003 SENTRUM, 0104

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