NO20031588L - Substituerte 3,4-dihydro-pyrimido(1,2-a)pyrimidiner og 3,4- dihydropyrazino(1,2-a)pyrimidiner - Google Patents

Substituerte 3,4-dihydro-pyrimido(1,2-a)pyrimidiner og 3,4- dihydropyrazino(1,2-a)pyrimidiner

Info

Publication number: NO20031588L
Authority: NO; Norway
Prior art keywords: pyrimidines; dihydropyrazino; pyrimido; dihydro; substituted
Prior art date: 2000-10-13

Application number

NO20031588A

Other languages

English (en)

Other versions

NO20031588D0 (no

Inventor

Matthias Gerlach

Corinna Maul

Utz-Peter Jagusch

Original Assignee

Gruenenthal Gmbh

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-10-13

Filing date

2003-04-08

Publication date

2003-04-08

2003-04-08 Application filed by Gruenenthal Gmbh filed Critical Gruenenthal Gmbh

2003-04-08 Publication of NO20031588L publication Critical patent/NO20031588L/no

2003-04-08 Publication of NO20031588D0 publication Critical patent/NO20031588D0/no

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/12—Antidiarrhoeals
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/04—Antipruritics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/16—Otologicals
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/08—Bridged systems
- C—CHEMISTRY; METALLURGY
- C40—COMBINATORIAL TECHNOLOGY
- C40B—COMBINATORIAL CHEMISTRY; LIBRARIES, e.g. CHEMICAL LIBRARIES
- C40B40/00—Libraries per se, e.g. arrays, mixtures

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Pain & Pain Management (AREA)
Urology & Nephrology (AREA)
Rheumatology (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Dermatology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

NO20031588A 2000-10-13 2003-04-08 Substituerte 3,4-dihydro-pyrimido(1,2-a)pyrimidiner og 3,4- dihydropyrazino(1,2-a)pyrimidiner NO20031588D0 (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
DE10050661A DE10050661A1 (de)	2000-10-13	2000-10-13	Substituierte 3,4-Dihydro-pyrimido[1,2-a]pyrimidine und 3,4-Dihydro-pyrazino[1,2-a]pyrimidine
PCT/EP2001/011702 WO2002030934A1 (de)	2000-10-13	2001-10-10	Substituierte 3,4-dihydro-pyrimido[1,2-a]pyrimidine und 3,4-dihydropyrazino[1,2-a]pyrimidine

Publications (2)

Publication Number	Publication Date
NO20031588L true NO20031588L (no)	2003-04-08
NO20031588D0 NO20031588D0 (no)	2003-04-08

Family

ID=7659596

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO20031588A NO20031588D0 (no)	2000-10-13	2003-04-08	Substituerte 3,4-dihydro-pyrimido(1,2-a)pyrimidiner og 3,4- dihydropyrazino(1,2-a)pyrimidiner

Country Status (25)

Country	Link
US (1)	US7226924B2 (no)
EP (1)	EP1325010B1 (no)
JP (1)	JP2004511485A (no)
KR (1)	KR20030036923A (no)
CN (1)	CN1243753C (no)
AR (1)	AR035496A1 (no)
AT (1)	ATE294180T1 (no)
AU (1)	AU2002214007A1 (no)
BR (1)	BR0114735A (no)
CA (1)	CA2425685A1 (no)
DE (2)	DE10050661A1 (no)
EC (1)	ECSP034554A (no)
ES (1)	ES2239168T3 (no)
HU (1)	HUP0302606A3 (no)
IL (1)	IL155379A0 (no)
MX (1)	MXPA03003199A (no)
NO (1)	NO20031588D0 (no)
NZ (1)	NZ525651A (no)
PE (1)	PE20020477A1 (no)
PL (1)	PL361777A1 (no)
PT (1)	PT1325010E (no)
RU (1)	RU2003113965A (no)
SK (1)	SK4152003A3 (no)
WO (1)	WO2002030934A1 (no)
ZA (1)	ZA200303634B (no)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
EP1828186A1 (en)	2004-12-13	2007-09-05	Sunesis Pharmaceuticals, Inc.	Pyrido pyrimidinones, dihydro pyrimido pyrimidinones and pteridinones useful as raf kinase inhibitors
US20070155738A1 (en)	2005-05-20	2007-07-05	Alantos Pharmaceuticals, Inc.	Heterobicyclic metalloprotease inhibitors

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3558618A (en) *	1968-04-01	1971-01-26	Dow Chemical Co	Novel 4h-pyrazino(1,2-a)pyrimidine-4-ones
GB1347493A (en) *	1971-02-11	1974-02-27	Aspro Nicholas Ltd	Benzazine derivatives
HU178910B (en) *	1977-08-19	1982-07-28	Chinoin Gyogyszer Es Vegyeszet	Process for preparing 2,3-disubstituted-4-oxo-4h-pyrido/1,2-a/-pyrimidines
JP2668259B2 (ja) *	1988-02-18	1997-10-27	塩野義製薬株式会社	複素環化合物および抗潰瘍剤
FI94531C (fi) *	1990-03-13	1995-09-25	Ime Intermed Enterpris Sa	Menetelmä farmaseuttisesti aktiivisen 1,3,4,6,7,8-heksahydro-2H-pyrimido-(1,2-a)-pyrimidiinijohdannaisen valmistamiseksi
IT1263804B (it) *	1993-01-22	1996-09-03	Luso Farmaco Inst	Derivati pirimidinonici fusi con eterocicli azotati ad attivita' a ii antagonista
AU707530B2 (en) *	1995-09-28	1999-07-15	Otsuka Pharmaceutical Factory, Inc.	Analgesic composition

2000
- 2000-10-13 DE DE10050661A patent/DE10050661A1/de not_active Withdrawn
2001
- 2001-10-09 AR ARP010104730A patent/AR035496A1/es not_active Application Discontinuation
- 2001-10-10 KR KR10-2003-7005149A patent/KR20030036923A/ko not_active Withdrawn
- 2001-10-10 CN CNB018171591A patent/CN1243753C/zh not_active Expired - Fee Related
- 2001-10-10 CA CA002425685A patent/CA2425685A1/en not_active Abandoned
- 2001-10-10 WO PCT/EP2001/011702 patent/WO2002030934A1/de not_active Ceased
- 2001-10-10 AT AT01982417T patent/ATE294180T1/de active
- 2001-10-10 BR BR0114735-8A patent/BR0114735A/pt not_active IP Right Cessation
- 2001-10-10 MX MXPA03003199A patent/MXPA03003199A/es active IP Right Grant
- 2001-10-10 RU RU2003113965/04A patent/RU2003113965A/ru not_active Application Discontinuation
- 2001-10-10 PL PL01361777A patent/PL361777A1/xx not_active Application Discontinuation
- 2001-10-10 EP EP01982417A patent/EP1325010B1/de not_active Expired - Lifetime
- 2001-10-10 AU AU2002214007A patent/AU2002214007A1/en not_active Abandoned
- 2001-10-10 IL IL15537901A patent/IL155379A0/xx unknown
- 2001-10-10 PT PT01982417T patent/PT1325010E/pt unknown
- 2001-10-10 ES ES01982417T patent/ES2239168T3/es not_active Expired - Lifetime
- 2001-10-10 NZ NZ525651A patent/NZ525651A/en unknown
- 2001-10-10 HU HU0302606A patent/HUP0302606A3/hu unknown
- 2001-10-10 JP JP2002534320A patent/JP2004511485A/ja not_active Withdrawn
- 2001-10-10 DE DE50106048T patent/DE50106048D1/de not_active Expired - Lifetime
- 2001-10-10 SK SK415-2003A patent/SK4152003A3/sk unknown
- 2001-10-12 PE PE2001001013A patent/PE20020477A1/es not_active Application Discontinuation
2003
- 2003-04-08 NO NO20031588A patent/NO20031588D0/no unknown
- 2003-04-09 US US10/409,614 patent/US7226924B2/en not_active Expired - Fee Related
- 2003-04-11 EC EC2003004554A patent/ECSP034554A/es unknown
- 2003-05-12 ZA ZA200303634A patent/ZA200303634B/en unknown

Also Published As

Publication number	Publication date
ATE294180T1 (de)	2005-05-15
CN1243753C (zh)	2006-03-01
HK1056558A1 (en)	2004-02-20
HUP0302606A3 (en)	2007-03-28
DE10050661A1 (de)	2002-04-18
NZ525651A (en)	2004-10-29
KR20030036923A (ko)	2003-05-09
EP1325010A1 (de)	2003-07-09
WO2002030934A1 (de)	2002-04-18
CN1469879A (zh)	2004-01-21
AR035496A1 (es)	2004-06-02
EP1325010B1 (de)	2005-04-27
CA2425685A1 (en)	2003-04-11
AU2002214007A1 (en)	2002-04-22
DE50106048D1 (de)	2005-06-02
ZA200303634B (en)	2004-08-12
MXPA03003199A (es)	2004-03-18
BR0114735A (pt)	2003-10-14
IL155379A0 (en)	2003-11-23
PE20020477A1 (es)	2002-06-29
US7226924B2 (en)	2007-06-05
RU2003113965A (ru)	2004-12-10
ES2239168T3 (es)	2005-09-16
US20030220322A1 (en)	2003-11-27
PT1325010E (pt)	2005-08-31
SK4152003A3 (en)	2003-10-07
HUP0302606A2 (hu)	2004-07-28
PL361777A1 (en)	2004-10-04
ECSP034554A (es)	2003-05-26
NO20031588D0 (no)	2003-04-08
JP2004511485A (ja)	2004-04-15

Publication	Publication Date	Title
NO20021356D0 (no)	2002-03-19	Alkylendiamin-substituerte pyrazolo[1,5,-a]-1,5-pyrimidiner og pyrazolo[1,5-a]-1,3,5-triaziner
DK1278750T3 (da)	2004-11-22	Imidazopyrimidinderivater og triazolopyrimidinderivater
IS7283A (is)	2004-05-21	3-ß-D-ríbófúranósýlþíasól[4,5-d]pýridímín kirnisleifar og notkun þeirra
NO20006090L (no)	2001-01-31	Pyrrolo(2,3d)pyrimidin sammensetninger og anvendelse herav
ATE261970T1 (de)	2004-04-15	Triazolo(4,5-d)pyrimidin-derivate
ATE251623T1 (de)	2003-10-15	Imidazo(1,2-a)pyridin- und pyrazolo(2,3- a)pyridinderivate
NO20022738D0 (no)	2002-06-07	Pyrrolo(2,3-d)pyrimidinforbindelser
NO20006454L (no)	2001-02-15	Pyrrolo(2,3-d)pyrimidinforbindelser
NO20006453L (no)	2001-02-05	Pyrrolo(2,3-d)pyrimidinforbindelser
NO20041142L (no)	2004-06-21	Subsitituerte 2-pyrimidinyl-6,7,8,9-tetrahydropyrimido[1,2-A]pyrimidin-4-on og 7-pyrimidinyl-2,3-dihydroimidazo[1,2-A]pyrimidin-5(1H)on-derivater for neurodegenerative lidelser
NO20030033L (no)	2003-01-03	Pyrido[2,3-D]pyrimidin- og pyrimido[4,5-D]pyrimidin- nukleosider
NO991150L (no)	1999-09-13	Pyrazolopyrimidiner og pyrazolotriaziner
IL160402A0 (en)	2004-07-25	Substituted 2-pyridinyl-6,7,8,9-tetrahydropyrimido {1,2-a} pyrimidin-4-one and 7-pyridinyl-2,3-dihydroimidazo{1,2-pyrimidin-5 (1h) one derivatives
DK1315731T3 (da)	2004-10-11	2-pyridinyl-6,7,8,9-tetrahydropyrimido[1,2-a]pyrimidin-4-on og 7-pyridinyl-2,3-dihydroimidazo[1,2-a]pyrimidin-5(1H)on-derivater
DE50208341D1 (de)	2006-11-16	Triazolopyrimidine
NO20031588D0 (no)	2003-04-08	Substituerte 3,4-dihydro-pyrimido(1,2-a)pyrimidiner og 3,4- dihydropyrazino(1,2-a)pyrimidiner
DK1325010T3 (da)	2005-05-17	Substituerede 3,4-dihydro-pyrimido[1,2-a]pyrimidiner og 3,4-dihydro-pyrazino[1,2-a]pyrimidiner
PT1326866E (pt)	2005-08-31	3,4-di-hidropirido[1,2-a]pirimidinas substituidas
SI1325010T1 (en)	2005-10-31	Substituted 3.4-dihydro-pyrimido (1,2-a)pyrimidines and 3.4-dihydropyrazino (1,2-a)pyrimidines
SI1368355T1 (sl)	2006-12-31	Substituirani pirazolo- in tiazolopirimidini kot analgetiki
DK1326866T3 (da)	2005-08-01	Substituerede 3,4-dihydro-pyrido[1,2-a]pyrimidiner