NO20035722D0 - Nye pyrido-pyrido-pyrrolo[3,2-g]pyrrolo[3,4-e]indol- og pyrido-pyrrolo[2,3-a]pyrrolo[3,4-c] karbazolforbindelser, fremgangsmåte for deresfremstilling og farmasöytiske sammensetninger inneholdende dem - Google Patents

Nye pyrido-pyrido-pyrrolo[3,2-g]pyrrolo[3,4-e]indol- og pyrido-pyrrolo[2,3-a]pyrrolo[3,4-c] karbazolforbindelser, fremgangsmåte for deresfremstilling og farmasöytiske sammensetninger inneholdende dem

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Publication number
NO20035722D0
NO20035722D0 NO20035722A NO20035722A NO20035722D0 NO 20035722 D0 NO20035722 D0 NO 20035722D0 NO 20035722 A NO20035722 A NO 20035722A NO 20035722 A NO20035722 A NO 20035722A NO 20035722 D0 NO20035722 D0 NO 20035722D0
Authority
NO
Norway
Prior art keywords
pyrrolo
pyrido
indole
preparation
pharmaceutical compositions
Prior art date
Application number
NO20035722A
Other languages
English (en)
Inventor
Michelle Prudhomme
Christelle Marminon
Sylvain Routier
Gerard Coudert
Jean-Yves Merour
John Hickman
Alain Pierre
Pierre Renard
Bruno Pfeiffer
Original Assignee
Servier Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Servier Lab filed Critical Servier Lab
Publication of NO20035722D0 publication Critical patent/NO20035722D0/no

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/22Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed systems contains four or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20Carbocyclic rings
    • C07H15/24Condensed ring systems having three or more rings
    • C07H15/252Naphthacene radicals, e.g. daunomycins, adriamycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Saccharide Compounds (AREA)
NO20035722A 2001-06-29 2003-12-19 Nye pyrido-pyrido-pyrrolo[3,2-g]pyrrolo[3,4-e]indol- og pyrido-pyrrolo[2,3-a]pyrrolo[3,4-c] karbazolforbindelser, fremgangsmåte for deresfremstilling og farmasöytiske sammensetninger inneholdende dem NO20035722D0 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0108615A FR2826653B1 (fr) 2001-06-29 2001-06-29 Nouveaux derives de pyrido-pyrido-pyrrolo[3,2-g]pyrrolo [3,4-e]-indole et pyrido-pyrrolo[2,3-a]pyrrolo[3,4-c] carbazole, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
PCT/FR2002/002250 WO2003002563A1 (fr) 2001-06-29 2002-06-28 Derives de pyrido-pyrido-pyrrolo pyrrolo-indole et pyrido-pyrrolo pyrrolo carbazole, leur procede de preparation et les compositions pharmaceutiques qui les contiennent

Publications (1)

Publication Number Publication Date
NO20035722D0 true NO20035722D0 (no) 2003-12-19

Family

ID=8864927

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20035722A NO20035722D0 (no) 2001-06-29 2003-12-19 Nye pyrido-pyrido-pyrrolo[3,2-g]pyrrolo[3,4-e]indol- og pyrido-pyrrolo[2,3-a]pyrrolo[3,4-c] karbazolforbindelser, fremgangsmåte for deresfremstilling og farmasöytiske sammensetninger inneholdende dem

Country Status (19)

Country Link
US (1) US7001906B2 (no)
EP (1) EP1409486A1 (no)
JP (1) JP2004535450A (no)
KR (1) KR100577543B1 (no)
CN (1) CN1275966C (no)
AR (1) AR036159A1 (no)
BR (1) BR0210698A (no)
CA (1) CA2452192A1 (no)
CZ (1) CZ2004143A3 (no)
EA (1) EA007221B1 (no)
FR (1) FR2826653B1 (no)
HU (1) HUP0400347A2 (no)
MX (1) MXPA03012011A (no)
NO (1) NO20035722D0 (no)
NZ (1) NZ530322A (no)
PL (1) PL366381A1 (no)
SK (1) SK692004A3 (no)
WO (1) WO2003002563A1 (no)
ZA (1) ZA200309514B (no)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2003095452A1 (en) 2002-05-08 2003-11-20 Janssen Pharmaceutica N.V. Substituted pyrroline kinase inhibitors
CA2520590A1 (en) * 2003-03-27 2004-11-04 Janssen Pharmaceutica, N.V. Substituted pyrroline kinase inhibitors
CA2573573A1 (en) 2004-07-27 2006-02-09 Sgx Pharmaceuticals, Inc. Fused ring heterocycle kinase modulators
WO2006015123A1 (en) 2004-07-27 2006-02-09 Sgx Pharmaceuticals, Inc. Pyrrolo-pyridine kinase modulators
US7361764B2 (en) 2004-07-27 2008-04-22 Sgx Pharmaceuticals, Inc. Pyrrolo-pyridine kinase modulators
US7626021B2 (en) 2004-07-27 2009-12-01 Sgx Pharmaceuticals, Inc. Fused ring heterocycle kinase modulators
WO2006061212A1 (en) * 2004-12-08 2006-06-15 Johannes Gutenberg-Universität Mainz 3-(indolyl)-4-arylmaleimide derivatives and their use as angiogenesis inhibitors
TWI499414B (zh) 2006-09-29 2015-09-11 Lexicon Pharmaceuticals Inc 鈉與葡萄糖第2型共同運輸體(co-transporter 2)的抑制物與其應用方法
US7846945B2 (en) * 2007-03-08 2010-12-07 Lexicon Pharmaceuticals, Inc. Piperdine-based inhibitors of sodium glucose co-transporter 2 and methods of their use
CN101720323A (zh) * 2007-04-11 2010-06-02 三井有限公司 具有抗癌活性的化合物
CN101234112B (zh) * 2008-03-03 2010-10-13 中国科学院化学研究所 阳离子咔唑类化合物的制药用途
CN103934464B (zh) * 2013-12-04 2016-01-20 宁波大学 一种咔唑吡啶银纳米棒及其制备方法
EP3119768B1 (en) 2014-03-16 2019-07-31 Hadasit Medical Research Services And Development Ltd. 3,4-bromo or -sulfonate substituted 1h-pyrrole-2,5-dione derivatives as type iii deiodinase (dio3) inhibitors for treating depressions and cancer
AR107030A1 (es) * 2015-12-09 2018-03-14 Padlock Therapeutics Inc Inhibidores aza-bencimidazol de pad4
EP3706735A1 (en) 2017-11-06 2020-09-16 Snap Bio, Inc. Pim kinase inhibitor compositions, methods, and uses thereof

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2108146A1 (en) * 1991-04-11 1992-10-12 Stuart W. Mccombie Anti-tumor and anti-psoriatic agents
GB9319297D0 (en) * 1993-09-17 1993-11-03 Wellcome Found Indole derivatives
GB9416467D0 (en) * 1994-08-13 1994-10-05 Wellcome Found Compounds for use in medicine
US5705511A (en) * 1994-10-14 1998-01-06 Cephalon, Inc. Fused pyrrolocarbazoles
JP2002523780A (ja) * 1998-08-26 2002-07-30 セフアロン・インコーポレーテツド 多系統キナーゼタンパク質の調節
FR2801054B1 (fr) * 1999-11-17 2003-06-13 Adir Nouveaux derives de 12,13-(pyranosyl)-indolo[2,3-a]pyrrolo [3,4-c]carbazole et 12,13-(pyranosyl)-furo[3,4-c]indolo [2,3-a]carbazole, leur procede de preparation et les compositions pharmaceutiques qui les contiennent

Also Published As

Publication number Publication date
SK692004A3 (en) 2004-07-07
NZ530322A (en) 2005-06-24
US20040152721A1 (en) 2004-08-05
HUP0400347A2 (hu) 2004-09-28
KR20040018397A (ko) 2004-03-03
WO2003002563A1 (fr) 2003-01-09
CZ2004143A3 (cs) 2004-05-12
CN1520415A (zh) 2004-08-11
EA007221B1 (ru) 2006-08-25
FR2826653A1 (fr) 2003-01-03
MXPA03012011A (es) 2004-03-26
FR2826653B1 (fr) 2005-10-14
CN1275966C (zh) 2006-09-20
AR036159A1 (es) 2004-08-18
CA2452192A1 (fr) 2003-01-09
EA200301301A1 (ru) 2004-06-24
KR100577543B1 (ko) 2006-05-10
JP2004535450A (ja) 2004-11-25
EP1409486A1 (fr) 2004-04-21
PL366381A1 (en) 2005-01-24
ZA200309514B (en) 2004-12-08
BR0210698A (pt) 2004-09-21
US7001906B2 (en) 2006-02-21

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