NO20040821L - 3-substituerte 6,7-dihydroksytetrahydroisokinolinderivater for andvendelse som antibakterielle midler. - Google Patents

3-substituerte 6,7-dihydroksytetrahydroisokinolinderivater for andvendelse som antibakterielle midler.

Info

Publication number
NO20040821L
NO20040821L NO20040821A NO20040821A NO20040821L NO 20040821 L NO20040821 L NO 20040821L NO 20040821 A NO20040821 A NO 20040821A NO 20040821 A NO20040821 A NO 20040821A NO 20040821 L NO20040821 L NO 20040821L
Authority
NO
Norway
Prior art keywords
derivatives
dihydroxytetrahydroisoquinoline
substituted
antibacterial agents
compounds
Prior art date
Application number
NO20040821A
Other languages
English (en)
Inventor
Kaspar Burri
Khalid Islam
Laurent Schmitt
Original Assignee
Arpida Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Arpida Ag filed Critical Arpida Ag
Publication of NO20040821L publication Critical patent/NO20040821L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
    • C07D217/02—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with only hydrogen atoms or radicals containing only carbon and hydrogen atoms, directly attached to carbon atoms of the nitrogen-containing ring; Alkylene-bis-isoquinolines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
    • C07D217/12—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with radicals, substituted by hetero atoms, attached to carbon atoms of the nitrogen-containing ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
    • C07D217/12—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with radicals, substituted by hetero atoms, attached to carbon atoms of the nitrogen-containing ring
    • C07D217/14—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with radicals, substituted by hetero atoms, attached to carbon atoms of the nitrogen-containing ring other than aralkyl radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
    • C07D217/12—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with radicals, substituted by hetero atoms, attached to carbon atoms of the nitrogen-containing ring
    • C07D217/14—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with radicals, substituted by hetero atoms, attached to carbon atoms of the nitrogen-containing ring other than aralkyl radicals
    • C07D217/16—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with radicals, substituted by hetero atoms, attached to carbon atoms of the nitrogen-containing ring other than aralkyl radicals substituted by oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

Det er beskrevet nye tetrahydroisokinolinderivater og anvendelse derav som aktive ingredienser for fremstilling av farmasøytiske sammensetninger. Oppfinnelsen vedrører også beslektede aspekter inkludert fremgangsmåter for fremstilling av forbindelsene, farmasøytiske sammensetninger inneholdende én eller flere av disse forbindelsene og spesielt anvendelse derav som antiinfeksj onsmidler.
NO20040821A 2001-08-27 2004-02-25 3-substituerte 6,7-dihydroksytetrahydroisokinolinderivater for andvendelse som antibakterielle midler. NO20040821L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP0109846 2001-08-27
PCT/EP2002/008916 WO2003018017A1 (en) 2001-08-27 2002-08-09 3-substituted 6,7-dihydroxytetrahydroisoquinoline derivatives for use as antibacterial agents

Publications (1)

Publication Number Publication Date
NO20040821L true NO20040821L (no) 2004-04-26

Family

ID=8164565

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20040821A NO20040821L (no) 2001-08-27 2004-02-25 3-substituerte 6,7-dihydroksytetrahydroisokinolinderivater for andvendelse som antibakterielle midler.

Country Status (12)

Country Link
US (1) US7371762B2 (no)
EP (1) EP1427417B1 (no)
JP (1) JP4383166B2 (no)
CN (1) CN1549716B (no)
AT (1) ATE386525T1 (no)
CA (1) CA2458477A1 (no)
DE (1) DE60225155T2 (no)
ES (1) ES2301701T3 (no)
MX (1) MXPA04001773A (no)
NO (1) NO20040821L (no)
PT (1) PT1427417E (no)
WO (1) WO2003018017A1 (no)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0419192D0 (en) * 2004-08-27 2004-09-29 Merck Sharp & Dohme Therapeutic agents
CN100386319C (zh) * 2005-12-05 2008-05-07 中国人民解放军第二军医大学 具有抗生育和抗真菌活性的四氢异喹啉类化合物或其盐类
EP2387564A1 (en) 2009-01-15 2011-11-23 Rutgers, The State University of New Jersey Benzo ýc¨phenanthridines as antimicrobial agents
CA2760526A1 (en) 2009-04-30 2010-11-04 Rutgers, The State University Of New Jersey Antimicrobial agents
US8933096B2 (en) 2010-06-09 2015-01-13 Rugers, The State University of New Jersey Antimicrobial agents
CA2803890A1 (en) 2010-06-25 2011-12-29 Rutgers, The State University Of New Jersey Antimicrobial agents
WO2013106756A2 (en) 2012-01-13 2013-07-18 Rutgers, The State University Of New Jersey Antimicrobial agents
EP2828245A1 (en) 2012-03-21 2015-01-28 Rutgers, The State University of New Jersey Antimicrobial agents
CN102731328B (zh) * 2012-06-18 2014-11-05 迪沙药业集团有限公司 一种盐酸安非他酮的制备方法
UA118548C2 (uk) 2012-12-21 2019-02-11 Епізайм, Інк. Тетрагідро- та дигідроізохіноліни як інгібітори prmt5 та їх застосування
US9458150B2 (en) 2013-11-08 2016-10-04 Rutgers, The State University Of New Jersey Antimicrobial agents
US10513528B2 (en) 2016-02-25 2019-12-24 Taxis Pharmaceuticals, Inc. Synthetic processes and intermediates
WO2018183917A1 (en) 2017-03-30 2018-10-04 Taxis Pharmaceuticals, Inc. Synthetic processes and synthetic intermediates

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2351027A1 (de) 1973-10-11 1975-04-24 Boehringer Sohn Ingelheim Propanolderivate
FR2662940B1 (fr) * 1990-06-08 1994-10-14 Roussel Uclaf Utilisation de derives de la tetrahydro isoquinoleine pour la preparation de medicaments anti-tumoraux, application a titre de medicaments de derives de la tetrahydro isoquinoleine et produits derives de cette structure.
US5124337A (en) 1991-05-20 1992-06-23 Schering Corporation N-acyl-tetrahydroisoquinolines as inhibitors of acyl-coenzyme a:cholesterol acyl transferase

Also Published As

Publication number Publication date
JP4383166B2 (ja) 2009-12-16
WO2003018017A1 (en) 2003-03-06
EP1427417B1 (en) 2008-02-20
CN1549716B (zh) 2010-05-26
ES2301701T3 (es) 2008-07-01
EP1427417A1 (en) 2004-06-16
CN1549716A (zh) 2004-11-24
ATE386525T1 (de) 2008-03-15
JP2005503392A (ja) 2005-02-03
PT1427417E (pt) 2008-06-02
US7371762B2 (en) 2008-05-13
MXPA04001773A (es) 2004-05-31
CA2458477A1 (en) 2003-03-06
DE60225155D1 (de) 2008-04-03
DE60225155T2 (de) 2009-03-05
US20040266817A1 (en) 2004-12-30

Similar Documents

Publication Publication Date Title
DE60204452D1 (de) Pyrazolo[1,5]pyridinderivate
BRPI0408681A (pt) compostos, composições farmacêuticas, uso de um derivado da 1,2,3,4-tetraidroisoquinolina, método para tratar ou prevenir doenças, processo para a manufatura de composições farmacêuticas, e, uso de um ou mais compostos
NO20051102L (no) Sulfonylamino-eddiksyre-derivater
IS6658A (is) Ný efnasambönd
ATE286500T1 (de) 1,2,3,4-tetrahydroisochinolin-derivate
NO20032905L (no) Nye benzodiazepiner og beslektede heterocykliske derivater som er anvendelige som orexinreseptorantagonister
ATE301653T1 (de) Pyrazolopyridine
PL372809A1 (en) Substituted 1,3-diphenylprop-2-en-1-one derivatives and preparation and uses thereof
ATE332639T1 (de) Herbizidzusammensetzung,umfassend herbizide verbindung in säureform und ansäuerndes mittel, applizierverfahren und herstellungsverfahren davon
EA200400432A1 (ru) Производные мочевины
ATE300541T1 (de) Pyrazolopyridinderivate
TW200514772A (en) Novel tetrahydropyridine derivatives
NO20040821L (no) 3-substituerte 6,7-dihydroksytetrahydroisokinolinderivater for andvendelse som antibakterielle midler.
NO20005497D0 (no) Heterocykliske derivater som inhiberer faktor Xa
IL160171A0 (en) Depsipeptide derivatives, processes for the preparation thereof and pharmaceutical compositions containing the same
NO20054763L (no) Salter av clopidogrel og fremgangsmate for fremstilling derav
AU3620799A (en) Heterocyclic derivatives which inhibit factor xa
TR200402070T4 (tr) Siklobüten-dion türevleri ve bunların damar sertliği tedavisinde kullanımı
ATE373000T1 (de) Pyrazolopyridin-derivate als antiherpesmittel
ATE274515T1 (de) Pyrazolopyridinderivate
SE0300457D0 (sv) Novel compounds
DE50212538D1 (de) Substituierte 5,6,6a,11b-tetrahydro-7-oxa-5-aza-benzoäcüfluoren-6-carbonsäurederivate als nmda-antagonisten
MXPA04000952A (es) Sales de derivados de acido 1,2,3-4-tetrahidro-isoquinolin-2-carboxilico.
ATE469146T1 (de) Benzofuranderivate und deren verwendung bei der behandlung von mikrobiellen infektionen
WO2004105738A3 (en) Use of tetrahydropyridine derivatives