NO20041485L - Farmasoytisk formulering omfattende (R)-bicalutamid - Google Patents

Farmasoytisk formulering omfattende (R)-bicalutamid

Info

Publication number
NO20041485L
NO20041485L NO20041485A NO20041485A NO20041485L NO 20041485 L NO20041485 L NO 20041485L NO 20041485 A NO20041485 A NO 20041485A NO 20041485 A NO20041485 A NO 20041485A NO 20041485 L NO20041485 L NO 20041485L
Authority
NO
Norway
Prior art keywords
bicalutamide
pharmaceutical formulation
formulation
pharmaceutical
Prior art date
Application number
NO20041485A
Other languages
English (en)
Inventor
Nicola Frances Bateman
Original Assignee
Astrazeneca Uk Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Uk Ltd filed Critical Astrazeneca Uk Ltd
Publication of NO20041485L publication Critical patent/NO20041485L/no

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/275Nitriles; Isonitriles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/146Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic macromolecular compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
NO20041485A 2001-10-15 2004-04-13 Farmasoytisk formulering omfattende (R)-bicalutamid NO20041485L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
SE0103424A SE0103424D0 (sv) 2001-10-15 2001-10-15 Pharmaceutical formulation
PCT/GB2002/004621 WO2003032950A1 (en) 2001-10-15 2002-10-11 Pharmaceutical formulation comprising (r) -bicalutamide

Publications (1)

Publication Number Publication Date
NO20041485L true NO20041485L (no) 2004-04-13

Family

ID=20285650

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20041485A NO20041485L (no) 2001-10-15 2004-04-13 Farmasoytisk formulering omfattende (R)-bicalutamid

Country Status (19)

Country Link
US (1) US20060058381A1 (no)
EP (1) EP1439823A1 (no)
JP (1) JP3639587B2 (no)
KR (1) KR20050035163A (no)
CN (1) CN1571658A (no)
AR (1) AR036877A1 (no)
BR (1) BR0213248A (no)
CA (1) CA2462219A1 (no)
CO (1) CO5580755A2 (no)
HU (1) HUP0401369A3 (no)
IL (1) IL161306A0 (no)
IS (1) IS7219A (no)
MX (1) MXPA04003520A (no)
NO (1) NO20041485L (no)
PL (1) PL368226A1 (no)
RU (1) RU2004115023A (no)
SE (1) SE0103424D0 (no)
WO (1) WO2003032950A1 (no)
ZA (1) ZA200402729B (no)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE307571T1 (de) * 2001-02-27 2005-11-15 Pharmazeutische formulierung enthaltend bicalutamid
EP3366283B1 (en) 2004-01-20 2021-09-01 Novartis AG Direct compression formulation and process
CN101128195A (zh) * 2005-02-23 2008-02-20 阿斯利康(瑞典)有限公司 用于递送增加的稳态血浆水平的比卡鲁胺
US20080045600A1 (en) * 2006-08-17 2008-02-21 Gawande Rahul S Bicalutamide compositions
US20100048524A1 (en) 2008-03-14 2010-02-25 Angela Brodie Novel C-17-Heteroaryl Steroidal CYP17 Inhibitors/Antiandrogens;Synthesis In Vitro Biological Activities, Pharmacokinetics and Antitumor Activity
WO2010091306A1 (en) 2009-02-05 2010-08-12 Tokai Pharmaceuticals Novel prodrugs of steroidal cyp17 inhibitors/antiandrogens
CN101987086B (zh) * 2009-08-03 2012-07-18 北京化工大学 一种超细比卡鲁胺口服片剂及其制备方法
CN103813794A (zh) * 2011-07-18 2014-05-21 拓凯制药公司 用于治疗前列腺癌的新型组合物及方法
TWI673051B (zh) 2012-09-11 2019-10-01 美商梅維森前列腺療法有限責任公司 恩雜魯它脈(enzalutamide)之調和物
EP2968370A4 (en) 2013-03-14 2016-09-21 Univ Maryland AGENT FOR ANDROGEN RECEPTOR DOWNWARD CONTROL AND USES THEREOF
EP3033088A4 (en) 2013-08-12 2017-03-08 Tokai Pharmaceuticals, Inc. Biomarkers for treatment of neoplastic disorders using androgen-targeted therapies
US10285948B2 (en) 2014-12-05 2019-05-14 Janssen Pharmaceutica Nv Anticancer compositions
EA201791222A1 (ru) * 2014-12-05 2017-09-29 Арагон Фармасьютикалз, Инк. Противораковые композиции

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3629237A (en) * 1968-09-12 1971-12-21 Shinetsu Chemical Co Compositions useful as enteric coatings and method for preparing acid phthalates of cellulose ethers for them
US4309405A (en) * 1979-08-09 1982-01-05 American Home Products Corporation Sustained release pharmaceutical compositions
ATE28864T1 (de) * 1982-07-23 1987-08-15 Ici Plc Amide-derivate.
US4946686A (en) * 1987-09-24 1990-08-07 Merck & Co., Inc. Solubility modulated drug delivery system
AU1537292A (en) * 1991-04-16 1992-11-17 Nippon Shinyaku Co. Ltd. Method of manufacturing solid dispersion
WO1995019770A1 (en) * 1994-01-21 1995-07-27 Sepracor, Inc. Methods and compositions for treating androgen-dependent diseases using optically pure r-(-)-casodex
ATE307571T1 (de) * 2001-02-27 2005-11-15 Pharmazeutische formulierung enthaltend bicalutamid
CA2443040A1 (en) * 2001-04-02 2002-10-17 Nicola Frances Bateman Solid pharmaceutical composition comprising 4 -cyano-trifluoro-3-(4-fluorophenyl-sulphonyl) -2-hydroxy-2-methylpropiono- m toluidide and pvp

Also Published As

Publication number Publication date
JP2004521963A (ja) 2004-07-22
RU2004115023A (ru) 2005-04-10
CN1571658A (zh) 2005-01-26
SE0103424D0 (sv) 2001-10-15
MXPA04003520A (es) 2004-07-23
US20060058381A1 (en) 2006-03-16
AR036877A1 (es) 2004-10-13
IL161306A0 (en) 2004-09-27
BR0213248A (pt) 2004-09-28
HUP0401369A2 (hu) 2004-11-29
JP3639587B2 (ja) 2005-04-20
WO2003032950A1 (en) 2003-04-24
CO5580755A2 (es) 2005-11-30
EP1439823A1 (en) 2004-07-28
HUP0401369A3 (en) 2006-05-29
PL368226A1 (en) 2005-03-21
IS7219A (is) 2004-04-14
CA2462219A1 (en) 2003-04-24
KR20050035163A (ko) 2005-04-15
ZA200402729B (en) 2005-01-13

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Legal Events

Date Code Title Description
FC2A Withdrawal, rejection or dismissal of laid open patent application