NO20051289L - Lincomycinderivater som fremviser antibakteriell aktivitet. - Google Patents

Lincomycinderivater som fremviser antibakteriell aktivitet.

Info

Publication number
NO20051289L
NO20051289L NO20051289A NO20051289A NO20051289L NO 20051289 L NO20051289 L NO 20051289L NO 20051289 A NO20051289 A NO 20051289A NO 20051289 A NO20051289 A NO 20051289A NO 20051289 L NO20051289 L NO 20051289L
Authority
NO
Norway
Prior art keywords
antibacterial activity
exhibiting antibacterial
derivatives exhibiting
lincomycin derivatives
linkomycin
Prior art date
Application number
NO20051289A
Other languages
English (en)
Inventor
Dinesh V Patel
Mikhail F Gordeev
Jason Lewis
Sampath K Anandan
Original Assignee
Vicuron Pharm Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Vicuron Pharm Inc filed Critical Vicuron Pharm Inc
Publication of NO20051289L publication Critical patent/NO20051289L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/02—Acyclic radicals, not substituted by cyclic structures
    • C07H15/14—Acyclic radicals, not substituted by cyclic structures attached to a sulfur, selenium or tellurium atom of a saccharide radical
    • C07H15/16—Lincomycin; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biotechnology (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Crystallography & Structural Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)

Abstract

Nye linkomycinderivater er beskrevet. Disse linkomycinderivatene fremviser antibakteriell aktivitet. Idet forbindelsen ifølge oppfinnelsen fremviser potente aktiviteter ovenfor bakterier, som inkluderer gram positive organismer, er de anvendelige antimikrobielle midler. Fremgangsmåte for syntese og anvendelse av forbindelsene er også beskrevet.
NO20051289A 2002-08-15 2005-03-14 Lincomycinderivater som fremviser antibakteriell aktivitet. NO20051289L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US40377002P 2002-08-15 2002-08-15
PCT/US2003/025820 WO2004016632A2 (en) 2002-08-15 2003-08-15 Lincomycin derivatives possessing antibacterial activity

Publications (1)

Publication Number Publication Date
NO20051289L true NO20051289L (no) 2005-05-09

Family

ID=31888275

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20051289A NO20051289L (no) 2002-08-15 2005-03-14 Lincomycinderivater som fremviser antibakteriell aktivitet.

Country Status (15)

Country Link
US (1) US7164011B2 (no)
EP (1) EP1529052A2 (no)
JP (1) JP2006504673A (no)
KR (1) KR20050056195A (no)
CN (1) CN1315859C (no)
AU (1) AU2003265475B2 (no)
BR (1) BR0313725A (no)
CA (1) CA2493799A1 (no)
EA (1) EA200500353A1 (no)
IL (1) IL166476A (no)
MX (1) MXPA05001689A (no)
NO (1) NO20051289L (no)
NZ (1) NZ538141A (no)
WO (1) WO2004016632A2 (no)
ZA (1) ZA200501012B (no)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7199105B2 (en) 2002-08-15 2007-04-03 Vicuron Pharmaceuticals, Inc. Lincomycin derivatives possessing antibacterial activity
EP1529052A2 (en) 2002-08-15 2005-05-11 Vicuron Pharmaceuticals, Inc. Lincomycin derivatives possessing antibacterial activity
RS20050931A (sr) * 2003-06-17 2008-04-04 Vicuron Pharmaceuticals Inc., Novi derivati linkomicina koji poseduju antimikrobnu aktivnost
US7199106B2 (en) 2003-06-17 2007-04-03 Vicuron Pharmaceuticals, Inc. Lincomycin derivatives possessing antimicrobial activity
EP1654268A2 (en) * 2003-06-17 2006-05-10 Vicuron Pharmaceuticals, Inc. Lincomycin derivatives possessing antibacterial activity
US7256177B2 (en) 2003-06-17 2007-08-14 Vicuron Pharmaceuticals, Inc. Lincomycin derivatives possessing antibacterial activity
US7361743B2 (en) 2004-02-11 2008-04-22 Pfizer Inc Lincomycin derivatives possessing antibacterial activity
US7871982B2 (en) * 2005-12-09 2011-01-18 Meiji Seika Kaisha, Ltd. Lincomycin derivatives and antimicrobial agents comprising the same as active ingredient
WO2008146919A1 (ja) * 2007-05-31 2008-12-04 Meiji Seika Kaisha, Ltd. リンコサミド誘導体及びこれを有効成分とする抗菌剤
US7879808B2 (en) * 2007-05-31 2011-02-01 Meiji Seika Kaisha, Ltd. Lincomycin derivatives and antimicrobial agents comprising the same as active ingredient
CN101555223B (zh) * 2009-04-17 2011-06-01 北京化工大学 一种吡利霉素中间体及其制备方法
CA2871766C (en) 2011-12-08 2020-06-16 The Board Of Regents Of The University Of Texas System Piperidine-based small molecule 5-hydroxytryptamine 2c receptor (5-ht2cr) allosteric modulators
CN105566411B (zh) * 2014-11-07 2020-11-13 中国科学院上海有机化学研究所 林可霉素生物合成中间产物及其制法和用途

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EP1529052A2 (en) 2002-08-15 2005-05-11 Vicuron Pharmaceuticals, Inc. Lincomycin derivatives possessing antibacterial activity
RS20050931A (sr) 2003-06-17 2008-04-04 Vicuron Pharmaceuticals Inc., Novi derivati linkomicina koji poseduju antimikrobnu aktivnost
EP1654268A2 (en) 2003-06-17 2006-05-10 Vicuron Pharmaceuticals, Inc. Lincomycin derivatives possessing antibacterial activity

Also Published As

Publication number Publication date
AU2003265475A1 (en) 2004-03-03
CN1315859C (zh) 2007-05-16
MXPA05001689A (es) 2005-05-27
ZA200501012B (en) 2006-10-25
CA2493799A1 (en) 2004-02-26
US7164011B2 (en) 2007-01-16
US20040116690A1 (en) 2004-06-17
WO2004016632A8 (en) 2004-09-30
WO2004016632A3 (en) 2004-06-24
CN1681832A (zh) 2005-10-12
JP2006504673A (ja) 2006-02-09
IL166476A0 (en) 2006-01-15
IL166476A (en) 2010-05-31
AU2003265475B2 (en) 2009-08-27
EA200500353A1 (ru) 2006-06-30
NZ538141A (en) 2007-06-29
BR0313725A (pt) 2006-06-13
EP1529052A2 (en) 2005-05-11
WO2004016632A2 (en) 2004-02-26
KR20050056195A (ko) 2005-06-14
WO2004016632B1 (en) 2004-08-19

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