NO20054636L - Fremgangsmate for fremstilling av steroidale karbotiosyrederivater og -intermediater - Google Patents

Fremgangsmate for fremstilling av steroidale karbotiosyrederivater og -intermediater

Info

Publication number
NO20054636L
NO20054636L NO20054636A NO20054636A NO20054636L NO 20054636 L NO20054636 L NO 20054636L NO 20054636 A NO20054636 A NO 20054636A NO 20054636 A NO20054636 A NO 20054636A NO 20054636 L NO20054636 L NO 20054636L
Authority
NO
Norway
Prior art keywords
steroidal
intermediates
preparation
acid derivatives
carbothioic acid
Prior art date
Application number
NO20054636A
Other languages
English (en)
Other versions
NO20054636D0 (no
Inventor
Trond Lovli
Anne-Mette Nygaard
Bjorn Reitstoen
Magny Fivelstad
Original Assignee
Alpharma Aps
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from EP03007756A external-priority patent/EP1466920A1/en
Application filed by Alpharma Aps filed Critical Alpharma Aps
Publication of NO20054636D0 publication Critical patent/NO20054636D0/no
Publication of NO20054636L publication Critical patent/NO20054636L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J3/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom
    • C07J3/005—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom the carbon atom being part of a carboxylic function
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
    • C07J31/006—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring not covered by C07J31/003
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J43/003—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)

Abstract

Fremgangsmåte for konvertering av steroide 17(-karboksylsyrer til en karbotionsyre og estere derav som fluticasonpropionat.
NO20054636A 2003-04-04 2005-10-10 Fremgangsmate for fremstilling av steroidale karbotiosyrederivater og -intermediater NO20054636L (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP03007756A EP1466920A1 (en) 2003-04-04 2003-04-04 Process for the preparation of steroidal 17 beta-carbothioates
DKPA200400449 2004-03-19
PCT/DK2004/000242 WO2004087731A1 (en) 2003-04-04 2004-04-02 Process for the preparation of steroidal carbothioic acid derivatives and intermediates

Publications (2)

Publication Number Publication Date
NO20054636D0 NO20054636D0 (no) 2005-10-10
NO20054636L true NO20054636L (no) 2005-12-27

Family

ID=33132910

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20054636A NO20054636L (no) 2003-04-04 2005-10-10 Fremgangsmate for fremstilling av steroidale karbotiosyrederivater og -intermediater

Country Status (7)

Country Link
US (1) US20070270584A1 (no)
EP (1) EP1611149A1 (no)
JP (1) JP2006522028A (no)
AU (1) AU2004226318B2 (no)
CA (1) CA2530680A1 (no)
NO (1) NO20054636L (no)
WO (1) WO2004087731A1 (no)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9303060B1 (en) 2014-10-03 2016-04-05 Amphaster Pharmaceuticals, Inc. Methods of preparing intermediate of fluticasone propionate
CN110317238B (zh) * 2018-03-31 2022-08-09 天津药业研究院股份有限公司 一种糠酸氟替卡松的制备方法
CN116417675A (zh) * 2023-05-16 2023-07-11 珠海冠宇电池股份有限公司 电解液和锂离子电池

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4188385A (en) * 1978-04-05 1980-02-12 Syntex (U.S.A.) Inc. Thioetianic acid derivatives
US4198403A (en) * 1978-04-05 1980-04-15 Syntex (U.S.A.) Inc. 17 Beta-thiocarboxylic acid esters of 4-halo-3-oxoandrost-4-enes
BE887518A (fr) * 1980-02-15 1981-08-13 Glaxo Group Ltd Cartothioates d'androstanes
GB2088877B (en) * 1980-02-15 1984-07-04 Glaxo Group Ltd Androstane 17 carbothioates
US4578221A (en) * 1980-04-23 1986-03-25 Glaxo Group Limited Androstane carbothioic acids
US4578211A (en) * 1983-04-08 1986-03-25 General Electric Company Process for the preparation of rare earth oxyhalide phosphor
JP3091297B2 (ja) * 1992-01-10 2000-09-25 住友製薬株式会社 ピロリジン誘導体およびその製造方法
CN1133643C (zh) * 1995-12-29 2004-01-07 葛兰素集团有限公司 17-β-羧基,羰基硫代以及酰胺雄甾烷衍生物的内酯衍生物
US20020133032A1 (en) * 2000-02-25 2002-09-19 Jufang Barkalow Method for the preparation of fluticasone and related 17beta-carbothioic esters using a novel carbothioic acid synthesis and novel purification methods
GB0017988D0 (en) * 2000-07-21 2000-09-13 Glaxo Group Ltd Novel process
SI1775305T1 (sl) * 2000-08-05 2015-01-30 Glaxo Group Limited S-fluorometil ester 6alfa,9alfa-difluoro-17alfa-((2-furanilkarboksil)oksi)- 11beta-hidroksi-16alfa-metil-3-okso-androst-1,4-dien-17-karbotiojske kisline kot protivnetno sredstvo
JPWO2002085890A1 (ja) * 2001-04-20 2004-08-12 萬有製薬株式会社 ベンズイミダゾロン誘導体

Also Published As

Publication number Publication date
WO2004087731A1 (en) 2004-10-14
AU2004226318B2 (en) 2008-06-05
AU2004226318A1 (en) 2004-10-14
NO20054636D0 (no) 2005-10-10
EP1611149A1 (en) 2006-01-04
CA2530680A1 (en) 2004-10-14
US20070270584A1 (en) 2007-11-22
JP2006522028A (ja) 2006-09-28

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Representative=s name: ONSAGERS AS, POSTBOKS 6963 ST OLAVS PLASS, 0130 OS

FC2A Withdrawal, rejection or dismissal of laid open patent application