NO20054740L - Farmasoytiske sammensetninger av CETP inhibitorer - Google Patents

Farmasoytiske sammensetninger av CETP inhibitorer

Info

Publication number
NO20054740L
NO20054740L NO20054740A NO20054740A NO20054740L NO 20054740 L NO20054740 L NO 20054740L NO 20054740 A NO20054740 A NO 20054740A NO 20054740 A NO20054740 A NO 20054740A NO 20054740 L NO20054740 L NO 20054740L
Authority
NO
Norway
Prior art keywords
pharmaceutical compositions
cetp inhibitors
inhibitor
cept
administration
Prior art date
Application number
NO20054740A
Other languages
English (en)
Other versions
NO336891B1 (no
NO20054740D0 (no
Inventor
Masaki Sunami
Takanori Serigano
Original Assignee
Japan Tobacco Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=33033290&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20054740(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Japan Tobacco Inc filed Critical Japan Tobacco Inc
Publication of NO20054740D0 publication Critical patent/NO20054740D0/no
Publication of NO20054740L publication Critical patent/NO20054740L/no
Publication of NO336891B1 publication Critical patent/NO336891B1/no

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C235/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms
    • C07C235/70—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups and doubly-bound oxygen atoms bound to the same carbon skeleton
    • C07C235/82—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups and doubly-bound oxygen atoms bound to the same carbon skeleton with the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a ring other than a six-membered aromatic ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/095—Sulfur, selenium, or tellurium compounds, e.g. thiols
    • A61K31/10—Sulfides; Sulfoxides; Sulfones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A61K31/167—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the nitrogen of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/265—Esters, e.g. nitroglycerine, selenocyanates of carbonic, thiocarbonic, or thiocarboxylic acids, e.g. thioacetic acid, xanthogenic acid, trithiocarbonic acid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Diabetes (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Emergency Medicine (AREA)
  • Hematology (AREA)
  • Cardiology (AREA)
  • Obesity (AREA)
  • Pain & Pain Management (AREA)
  • Endocrinology (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)
  • Steroid Compounds (AREA)

Abstract

Det tilveiebringes farmasøytiske preparater omfattende en kolesterylester overføringsprotein (CETP) inhibitor og et vannuoppløselig, konsentrasjonsøkende additiv, som viser forbedret biotilgjengelighet. Det beskrives videre metoder for behandling av kardiovaskulære lidelser omfattende administrering av det farmasøytiske preparat omfattende en CETP-inhibitor.
NO20054740A 2003-03-17 2005-10-14 Farmasøytiske sammensetninger av CETP inhibitorer NO336891B1 (no)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US45529303P 2003-03-17 2003-03-17
US46052103P 2003-04-04 2003-04-04
US47720203P 2003-06-10 2003-06-10
US49364903P 2003-08-08 2003-08-08
PCT/JP2004/003585 WO2004082593A2 (en) 2003-03-17 2004-03-17 Pharmaceutical compositions of cetp inhibitors

Publications (3)

Publication Number Publication Date
NO20054740D0 NO20054740D0 (no) 2005-10-14
NO20054740L true NO20054740L (no) 2005-12-13
NO336891B1 NO336891B1 (no) 2015-11-23

Family

ID=33033290

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20054740A NO336891B1 (no) 2003-03-17 2005-10-14 Farmasøytiske sammensetninger av CETP inhibitorer

Country Status (20)

Country Link
US (2) US20040225018A1 (no)
EP (2) EP2289507A1 (no)
JP (2) JP5546715B2 (no)
KR (2) KR20080008440A (no)
AT (1) ATE534381T1 (no)
AU (1) AU2004222434B2 (no)
BR (1) BRPI0408466B8 (no)
CA (1) CA2519432C (no)
CO (1) CO5640101A2 (no)
CY (1) CY1112324T1 (no)
DK (1) DK1603553T3 (no)
ES (1) ES2377121T3 (no)
IL (1) IL170749A (no)
MX (1) MXPA05009848A (no)
NO (1) NO336891B1 (no)
NZ (1) NZ542852A (no)
PL (1) PL1603553T3 (no)
PT (1) PT1603553E (no)
SI (1) SI1603553T1 (no)
WO (1) WO2004082593A2 (no)

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US7393652B2 (en) 2000-05-10 2008-07-01 The Trustees Of Columbia University In The City Of New York Methods for identifying a chemical compound that directly enhances binding of FKBP12.6 to PKA-phosphorylated type 2 ryanodine receptor (RyR2)
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US8710045B2 (en) 2004-01-22 2014-04-29 The Trustees Of Columbia University In The City Of New York Agents for preventing and treating disorders involving modulation of the ryanodine receptors
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CN101378731B (zh) 2006-02-09 2014-03-05 默沙东公司 Cetp抑制剂的聚合物制剂
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BR112013014291A2 (pt) * 2010-12-08 2016-09-20 Hoffmann La Roche formulação lipossômica de calcetrapib
CN103391769A (zh) * 2011-02-17 2013-11-13 霍夫曼-拉罗奇有限公司 通过热熔挤出使活性药物成分从过冷液体状态受控结晶的方法
BR112016013923A2 (pt) * 2013-12-19 2017-08-08 Hoffmann La Roche Modulador de cetp para o uso no tratamento de enfermidade ocular
JP2021534236A (ja) * 2018-08-09 2021-12-09 ダルコア ファーマ ユーケー リミテッド，レザーヘッド，ツーク ブランチ 新規発症２型糖尿病の発生遅延並びに２型糖尿病の進行緩徐化及び治療の方法
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CO5640101A2 (es) 2006-05-31
AU2004222434B2 (en) 2010-06-03
KR20050110019A (ko) 2005-11-22
IL170749A0 (en) 2009-02-11
EP1603553A2 (en) 2005-12-14
BRPI0408466B1 (pt) 2018-11-21
US20140243414A1 (en) 2014-08-28
EP1603553B1 (en) 2011-11-23
ATE534381T1 (de) 2011-12-15
JP2006520808A (ja) 2006-09-14
NZ542852A (en) 2008-09-26
ES2377121T9 (es) 2012-08-21
ES2377121T3 (es) 2012-03-22
BRPI0408466A (pt) 2006-04-04
KR100857759B1 (ko) 2008-09-09
BRPI0408466B8 (pt) 2021-05-25
JP5546715B2 (ja) 2014-07-09
NO336891B1 (no) 2015-11-23
NO20054740D0 (no) 2005-10-14
PL1603553T3 (pl) 2012-04-30
SI1603553T1 (sl) 2012-03-30
JP2011052006A (ja) 2011-03-17
EP1603553B9 (en) 2012-06-20
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CA2519432A1 (en) 2004-09-30
MXPA05009848A (es) 2005-12-06
AU2004222434A1 (en) 2004-09-30
US20040225018A1 (en) 2004-11-11
HK1084882A1 (en) 2006-08-11
WO2004082593A3 (en) 2005-02-24
IL170749A (en) 2012-08-30
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DK1603553T3 (da) 2012-01-30
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