NO20055925L - Ny fremgangsmate for fremstilling av melagatran - Google Patents

Ny fremgangsmate for fremstilling av melagatran

Info

Publication number: NO20055925L
Authority: NO; Norway
Prior art keywords: melagatran; preparation; new process; formula; compound
Prior art date: 2003-06-25

Application number

NO20055925A

Other languages

English (en)

Norwegian (no)

Inventor

Marcus Grehn

Tibor Musil

Magnus Sjogren

Original Assignee

Astrazeneca Ab

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2003-06-25

Filing date

2005-12-13

Publication date

2006-01-19

2005-12-13 Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab

2006-01-19 Publication of NO20055925L publication Critical patent/NO20055925L/no

Links

DKWNMCUOEDMMIN-PKOBYXMFSA-N melagatran Chemical compound C1=CC(C(=N)N)=CC=C1CNC(=O)[C@H]1N(C(=O)[C@H](NCC(O)=O)C2CCCCC2)CC1 DKWNMCUOEDMMIN-PKOBYXMFSA-N 0.000 title abstract 2
229960002137 melagatran Drugs 0.000 title abstract 2
238000000034 method Methods 0.000 title abstract 2
125000000217 alkyl group Chemical group 0.000 abstract 1
125000001797 benzyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])* 0.000 abstract 1
150000001875 compounds Chemical class 0.000 abstract 1
230000007062 hydrolysis Effects 0.000 abstract 1
238000006460 hydrolysis reaction Methods 0.000 abstract 1
LMBFAGIMSUYTBN-MPZNNTNKSA-N teixobactin Chemical compound C([C@H](C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H](CCC(N)=O)C(=O)N[C@H]([C@@H](C)CC)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H]1C(N[C@@H](C)C(=O)N[C@@H](C[C@@H]2NC(=N)NC2)C(=O)N[C@H](C(=O)O[C@H]1C)[C@@H](C)CC)=O)NC)C1=CC=CC=C1 LMBFAGIMSUYTBN-MPZNNTNKSA-N 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06008—Dipeptides with the first amino acid being neutral
- C07K5/06078—Dipeptides with the first amino acid being neutral and aromatic or cycloaliphatic
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Molecular Biology (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Biophysics (AREA)
General Health & Medical Sciences (AREA)
Genetics & Genomics (AREA)
Medicinal Chemistry (AREA)
Health & Medical Sciences (AREA)
Biochemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Plural Heterocyclic Compounds (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Peptides Or Proteins (AREA)

NO20055925A 2003-06-25 2005-12-13 Ny fremgangsmate for fremstilling av melagatran NO20055925L (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
SE0301879A SE0301879D0 (sv)	2003-06-25	2003-06-25	New process
PCT/SE2004/001016 WO2004113364A1 (en)	2003-06-25	2004-06-23	New process for the production of melagatran

Publications (1)

Publication Number	Publication Date
NO20055925L true NO20055925L (no)	2006-01-19

Family

ID=27656614

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO20055925A NO20055925L (no)	2003-06-25	2005-12-13	Ny fremgangsmate for fremstilling av melagatran

Country Status (14)

Country	Link
US (1)	US20060178312A1 (pt)
EP (1)	EP1641814A1 (pt)
JP (1)	JP2007536197A (pt)
KR (1)	KR20060025569A (pt)
CN (1)	CN1809585A (pt)
AU (1)	AU2004249658B2 (pt)
BR (1)	BRPI0411769A (pt)
CA (1)	CA2528930A1 (pt)
IL (1)	IL172287A0 (pt)
MX (1)	MXPA05013944A (pt)
NO (1)	NO20055925L (pt)
SE (1)	SE0301879D0 (pt)
WO (1)	WO2004113364A1 (pt)
ZA (1)	ZA200510102B (pt)

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
SE9301916D0 (sv) *	1993-06-03	1993-06-03	Ab Astra	New peptides derivatives
TWI238827B (en) *	1995-12-21	2005-09-01	Astrazeneca Ab	Prodrugs of thrombin inhibitors

2003
- 2003-06-25 SE SE0301879A patent/SE0301879D0/xx unknown
2004
- 2004-06-23 JP JP2006517053A patent/JP2007536197A/ja active Pending
- 2004-06-23 CN CNA2004800175458A patent/CN1809585A/zh active Pending
- 2004-06-23 BR BRPI0411769-7A patent/BRPI0411769A/pt not_active IP Right Cessation
- 2004-06-23 WO PCT/SE2004/001016 patent/WO2004113364A1/en not_active Ceased
- 2004-06-23 AU AU2004249658A patent/AU2004249658B2/en not_active Ceased
- 2004-06-23 MX MXPA05013944A patent/MXPA05013944A/es unknown
- 2004-06-23 CA CA002528930A patent/CA2528930A1/en not_active Abandoned
- 2004-06-23 KR KR1020057024865A patent/KR20060025569A/ko not_active Withdrawn
- 2004-06-23 EP EP04749054A patent/EP1641814A1/en not_active Withdrawn
- 2004-06-23 US US10/561,944 patent/US20060178312A1/en not_active Abandoned
2005
- 2005-11-30 IL IL172287A patent/IL172287A0/en unknown
- 2005-12-12 ZA ZA200510102A patent/ZA200510102B/xx unknown
- 2005-12-13 NO NO20055925A patent/NO20055925L/no not_active Application Discontinuation

Also Published As

Publication number	Publication date
AU2004249658B2 (en)	2007-02-01
KR20060025569A (ko)	2006-03-21
ZA200510102B (en)	2006-11-29
JP2007536197A (ja)	2007-12-13
IL172287A0 (en)	2006-04-10
AU2004249658A1 (en)	2004-12-29
MXPA05013944A (es)	2006-02-24
US20060178312A1 (en)	2006-08-10
WO2004113364A1 (en)	2004-12-29
BRPI0411769A (pt)	2006-08-08
SE0301879D0 (sv)	2003-06-25
CA2528930A1 (en)	2004-12-29
CN1809585A (zh)	2006-07-26
EP1641814A1 (en)	2006-04-05

Similar Documents

Publication	Publication Date	Title
AU2009258040A8 (en)	2014-04-24	Compounds and method for reducing uric acid
EA200970172A1 (ru)	2009-08-28	Пролекарство соединения амида коричной кислоты
MXPA05006907A (es)	2006-01-11	Compuestos diazoicos cationicos, composiciones que los contienen como colorante directo, procedimiento de coloracion de fibras queratinicas y dispositivo.
EG25480A (en)	2012-01-15	Method for preparation of optionally 2-substituted1,6-dihydro-6-oxo-4-pyrimidinecarboxylic acids
MX2007004215A (es)	2007-12-12	Proceso para la sintesis de 4-(3-metansulfonilfenil)-1-n- propilpiperidina.
WO2009095933A3 (en)	2011-06-30	Improved and novel process for the preparation of bosentan
WO2009066735A1 (ja)	2009-05-28	２－アザアダマンタン類の製造方法
NO20040388L (no)	2004-01-29	Fremgangsmåte for fremstilling av beraprost og salter derav, samt forbindelser som er mellomprodukter i fremgangsmåten
NO20023126L (no)	2002-06-27	Fremgangsmåte for fremstilling av citalopram
NO20092076L (no)	2009-08-17	Ny fremgangsmate for fremstilling av 4,4'-(1-metyl-1,2-etandiyl)-bis-(2,6-piperazindion)
UA106191C2 (ru)	2014-08-11	Способ получения транс-1-((1r,3s)-6-хлор-3-фенилиндан-1-ил)-3,3-диметилпиперазина
ATE441627T1 (de)	2009-09-15	Verfahren zur herstellung von valsartan
WO2007057225A3 (en)	2007-07-26	Process for making montelukast and intermediates therefor
MXPA04000046A (es)	2004-05-21	Proceso para la preparacion de las formas enantiomericas de los derivados de acido 2-(2,5-dioxoimidazolidin-1-il)-acetico 2-sustituidos.
NO20055925L (no)	2006-01-19	Ny fremgangsmate for fremstilling av melagatran
TW200719889A (en)	2007-06-01	Amino acid derivatives
EE05136B1 (et)	2009-02-16	Asendatud imidasopridiinhendite valmistamise meetod
FI20030026A0 (fi)	2003-01-08	Menetelmä substituoitujen imidatsolijohdannaisten valmistamiseksi ja menetelmässä käytettäviä välituotteita
MEP1708A (xx)	2010-02-10	Postupak proizvodnje thip-a
ATE519739T1 (de)	2011-08-15	Neuartiges verfahren zur herstellung von sulphonylpyrrolen als hdac-hemmer
NO20063112L (no)	2006-09-05	Forbedret syntese av 2-substituerte adenosiner
WO2007057767A3 (en)	2007-08-30	Amino acid derivatives
TW200801016A (en)	2008-01-01	Thienopyridine-2-carboxamide derivatives
WO2007025696A3 (en)	2007-05-18	Process for making substituted piperazinyl compounds
WO2005066174A3 (en)	2006-01-12	Process for the preparation of carbapenem compounds

Legal Events

Date	Code	Title	Description
2010-01-25	FC2A	Withdrawal, rejection or dismissal of laid open patent application