NO20061395L - Nye pyridinderivater - Google Patents

Nye pyridinderivater

Info

Publication number
NO20061395L
NO20061395L NO20061395A NO20061395A NO20061395L NO 20061395 L NO20061395 L NO 20061395L NO 20061395 A NO20061395 A NO 20061395A NO 20061395 A NO20061395 A NO 20061395A NO 20061395 L NO20061395 L NO 20061395L
Authority
NO
Norway
Prior art keywords
pyridine derivatives
compounds
new pyridine
preparation
relates
Prior art date
Application number
NO20061395A
Other languages
English (en)
Inventor
Thomas Weller
Martine Clozel
Boris Mathys
Daniel Bur
Claus Mueller
Michael Scherz
Joerg Velker
Original Assignee
Actelion Pharmaceuticals Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Actelion Pharmaceuticals Ltd filed Critical Actelion Pharmaceuticals Ltd
Publication of NO20061395L publication Critical patent/NO20061395L/no

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • A—HUMAN NECESSITIES
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    • A61P5/14—Drugs for disorders of the endocrine system of the thyroid hormones, e.g. T3, T4
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    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
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    • A61P7/04—Antihaemorrhagics; Procoagulants; Haemostatic agents; Antifibrinolytic agents
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    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P9/12—Antihypertensives

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
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  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
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  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Diabetes (AREA)
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  • Hematology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Psychiatry (AREA)
  • Pulmonology (AREA)
  • Pain & Pain Management (AREA)
  • Ophthalmology & Optometry (AREA)
  • Urology & Nephrology (AREA)
  • Endocrinology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Addiction (AREA)
  • Gynecology & Obstetrics (AREA)
  • Communicable Diseases (AREA)
  • Emergency Medicine (AREA)
  • Obesity (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Oncology (AREA)
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  • Gastroenterology & Hepatology (AREA)

Abstract

Oppfinnelsen angår nye pyridinderivater med formel I og beslektede forbindelser og anvendelse av dem som aktive bestanddeler ved fremstilling av farmasøytiske preparater. Oppfinnelsen angår også beslektede aspekter omfattende prosesser for fremstilling av forbindelser, farmasøytiske preparater inneholdende én eller flere av forbindelsene og spesielt anvendelse av dem som nevrohormonelle antagonister, spesielt som urotensin II-inhibitorer.
NO20061395A 2003-09-26 2006-03-27 Nye pyridinderivater NO20061395L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP0310746 2003-09-26
PCT/EP2004/010559 WO2005030209A1 (en) 2003-09-26 2004-09-21 Pyridine derivatives and use thereof as urotensin ii antagonists

Publications (1)

Publication Number Publication Date
NO20061395L true NO20061395L (no) 2006-06-22

Family

ID=34384524

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20061395A NO20061395L (no) 2003-09-26 2006-03-27 Nye pyridinderivater

Country Status (18)

Country Link
US (1) US7750161B2 (no)
EP (1) EP1670470B1 (no)
JP (1) JP4851328B2 (no)
KR (1) KR20070014108A (no)
CN (1) CN1856305B (no)
AR (1) AR045949A1 (no)
AT (1) ATE427748T1 (no)
AU (1) AU2004275488A1 (no)
BR (1) BRPI0414777A (no)
CA (1) CA2540196C (no)
DE (1) DE602004020486D1 (no)
IL (1) IL174497A0 (no)
MX (1) MXPA06003264A (no)
NO (1) NO20061395L (no)
RU (1) RU2006113948A (no)
TW (1) TW200526630A (no)
WO (1) WO2005030209A1 (no)
ZA (1) ZA200602442B (no)

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EP1608319A4 (en) 2003-04-03 2007-02-28 Univ California IMPROVED HEMMER FOR SOLUBLE EPOXY HYDROLASE
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EP1814875A4 (en) 2004-10-20 2010-02-17 Univ California IMPROVED INHIBITORS OF SOLUBLE EPOXY HYDROLASE
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WO2006135694A2 (en) * 2005-06-10 2006-12-21 Acadia Pharmaceuticals Inc. Uii-modulating compounds and their use
AR059826A1 (es) 2006-03-13 2008-04-30 Univ California Inhibidores de urea conformacionalmente restringidos de epoxido hidrolasa soluble
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US8765736B2 (en) * 2007-09-28 2014-07-01 Purdue Pharma L.P. Benzenesulfonamide compounds and the use thereof
KR20100102646A (ko) 2007-12-11 2010-09-24 가부시키가이샤 사이토파스파인더 카르복스아미드 화합물 및 케모카인 수용체 길항제로서의 이의 용도
WO2012054093A2 (en) 2010-01-29 2012-04-26 The Regents Of The University Of California Acyl piperidine inhibitors of soluble epoxide hydrolase

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Also Published As

Publication number Publication date
EP1670470B1 (en) 2009-04-08
BRPI0414777A (pt) 2006-11-21
KR20070014108A (ko) 2007-01-31
EP1670470A1 (en) 2006-06-21
WO2005030209A8 (en) 2006-05-11
JP2007506692A (ja) 2007-03-22
ZA200602442B (en) 2007-09-26
US20070043081A1 (en) 2007-02-22
DE602004020486D1 (de) 2009-05-20
RU2006113948A (ru) 2007-11-10
CA2540196A1 (en) 2005-04-07
MXPA06003264A (es) 2006-06-08
TW200526630A (en) 2005-08-16
US7750161B2 (en) 2010-07-06
JP4851328B2 (ja) 2012-01-11
CN1856305B (zh) 2010-04-28
CN1856305A (zh) 2006-11-01
WO2005030209A1 (en) 2005-04-07
AR045949A1 (es) 2005-11-16
CA2540196C (en) 2012-03-20
IL174497A0 (en) 2006-08-01
AU2004275488A1 (en) 2005-04-07
ATE427748T1 (de) 2009-04-15

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