NO20061424L - Fremgangsmote for fremstillingen av THIP - Google Patents

Fremgangsmote for fremstillingen av THIP

Info

Publication number: NO20061424L
Authority: NO; Norway
Prior art keywords: thip; preparation; alkyl; acid; procedure
Prior art date: 2003-09-05

Application number

NO20061424A

Other languages

English (en)

Norwegian (no)

Inventor

Robert Dancer

Hans Petersen

Michael Bech Somrner

Original Assignee

Lundbeck & Co As H

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2003-09-05

Filing date

2006-03-29

Publication date

2006-03-29

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=58707236&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20061424(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2006-03-29 Application filed by Lundbeck & Co As H filed Critical Lundbeck & Co As H

2006-03-29 Publication of NO20061424L publication Critical patent/NO20061424L/no

Links

ZXRVKCBLGJOCEE-UHFFFAOYSA-N Gaboxadol Chemical compound C1NCCC2=C1ONC2=O ZXRVKCBLGJOCEE-UHFFFAOYSA-N 0.000 title abstract 4
238000000034 method Methods 0.000 title abstract 2
239000002253 acid Substances 0.000 abstract 3
125000004400 (C1-C12) alkyl group Chemical group 0.000 abstract 2
125000003118 aryl group Chemical group 0.000 abstract 2
150000003839 salts Chemical class 0.000 abstract 2
125000004642 (C1-C12) alkoxy group Chemical group 0.000 abstract 1
125000006552 (C3-C8) cycloalkyl group Chemical group 0.000 abstract 1
ZDZDSZQYRBZPNN-UHFFFAOYSA-N 4,5,6,7-tetrahydro-[1,2]oxazolo[5,4-c]pyridin-6-ium-3-olate;hydrochloride Chemical compound Cl.C1NCCC2=C1ONC2=O ZDZDSZQYRBZPNN-UHFFFAOYSA-N 0.000 abstract 1
101100277337 Arabidopsis thaliana DDM1 gene Proteins 0.000 abstract 1
125000002252 acyl group Chemical group 0.000 abstract 1
125000003342 alkenyl group Chemical group 0.000 abstract 1
101150113676 chr1 gene Proteins 0.000 abstract 1
150000001875 compounds Chemical class 0.000 abstract 1
125000000392 cycloalkenyl group Chemical group 0.000 abstract 1
229950004346 gaboxadol Drugs 0.000 abstract 1
229910052500 inorganic mineral Inorganic materials 0.000 abstract 1
239000000543 intermediate Substances 0.000 abstract 1
238000004519 manufacturing process Methods 0.000 abstract 1
239000011707 mineral Substances 0.000 abstract 1
208000019116 sleep disease Diseases 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives

Landscapes

Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Neurosurgery (AREA)
Life Sciences & Earth Sciences (AREA)
Neurology (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Veterinary Medicine (AREA)
Pharmacology & Pharmacy (AREA)
Biomedical Technology (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Anesthesiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Plural Heterocyclic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

NO20061424A 2003-09-05 2006-03-29 Fremgangsmote for fremstillingen av THIP NO20061424L (no)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
US50042203P	2003-09-05	2003-09-05
DKPA200301277		2003-09-05
PCT/DK2004/000579 WO2005023820A1 (en)	2003-09-05	2004-09-01	Method for the manufacture of thip

Publications (1)

Publication Number	Publication Date
NO20061424L true NO20061424L (no)	2006-03-29

Family

ID=58707236

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO20061424A NO20061424L (no)	2003-09-05	2006-03-29	Fremgangsmote for fremstillingen av THIP

Country Status (20)

Country	Link
US (1)	US7371863B2 (sr)
EP (1)	EP1664060A1 (sr)
JP (1)	JP4745233B2 (sr)
KR (1)	KR20060069482A (sr)
CN (2)	CN101497619A (sr)
AR (1)	AR045540A1 (sr)
AU (1)	AU2004270323B2 (sr)
BR (1)	BRPI0413741A (sr)
CA (1)	CA2537840C (sr)
EA (1)	EA200600542A1 (sr)
IL (1)	IL174070A (sr)
IS (1)	IS8333A (sr)
ME (1)	MEP1708A (sr)
MX (1)	MXPA06002434A (sr)
NO (1)	NO20061424L (sr)
NZ (1)	NZ545178A (sr)
RS (1)	RS20060157A (sr)
UA (1)	UA91496C2 (sr)
WO (1)	WO2005023820A1 (sr)
ZA (1)	ZA200602178B (sr)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB0402118D0 (en)	2004-01-30	2004-03-03	Merck Sharp & Dohme	Polymorphic forms of a GABAA agonist
AU2005229493A1 (en) *	2004-04-02	2005-10-13	H. Lundbeck A/S	Treatment of impaired respiratory function with gaboxadol
CN104974175A (zh) *	2014-04-11	2015-10-14	天津药物研究院	一种氨甲基羟异恶唑类似物的制备方法
DK3274331T3 (da)	2015-03-24	2020-03-23	H Lundbeck As	Fremstilling af 4,5,6,7-tetrahydroisozaxolo[5,4-c]pyridin-3-ol
GB2594616A (en)	2018-11-21	2021-11-03	Certego Therapeutics Inc	Gaboxadol for reducing risk of suicide and rapid relief of depression
CN111320577B (zh) *	2018-12-13	2023-06-23	广东东阳光药业有限公司	一种吡啶酰胺的制备方法及其应用
IL298334A (en)	2020-05-20	2023-01-01	Certego Therapeutics Inc	Ring deuterated gaboxadol and its use for the treatment of psychiatric disorders

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DK270378A (da)	1977-06-20	1978-12-21	Krogsgaard Larsen P	Isoxazolderivater
GB2088370B (en) *	1980-11-27	1984-08-01	Kefalas As	Tetrahydroisoxazolopyridine compounds
DE3145473A1 (de) *	1980-11-27	1982-08-26	Kefalas A/S, Koebenhavn-Valby	2-substituierte 4,5,6,7-tetrahydroisoxazolo (5,4-c) pyridin-3-on-verbindungen, verfahren zu ihrer herstellung und diese enthaltende arzneimittel
US4353910A (en) *	1981-11-27	1982-10-12	Kefalas A/S	Derivatives of 4,5,6,7-tetrahydroisoxazolo [5,4-c] pyridine-3-one, pharmaceutical compositions and methods of treatment
DE19525598C2 (de)	1995-07-13	1997-09-25	Max Planck Gesellschaft	Schlafmittel

2004
- 2004-08-30 AR ARP040103118A patent/AR045540A1/es not_active Application Discontinuation
- 2004-09-01 US US10/570,551 patent/US7371863B2/en not_active Expired - Fee Related
- 2004-09-01 MX MXPA06002434A patent/MXPA06002434A/es active IP Right Grant
- 2004-09-01 KR KR1020067004221A patent/KR20060069482A/ko not_active Abandoned
- 2004-09-01 RS YUP-2006/0157A patent/RS20060157A/sr unknown
- 2004-09-01 BR BRPI0413741-8A patent/BRPI0413741A/pt not_active IP Right Cessation
- 2004-09-01 WO PCT/DK2004/000579 patent/WO2005023820A1/en not_active Ceased
- 2004-09-01 CA CA2537840A patent/CA2537840C/en not_active Expired - Fee Related
- 2004-09-01 CN CNA2009100081718A patent/CN101497619A/zh active Pending
- 2004-09-01 CN CNB2004800254248A patent/CN100482668C/zh not_active Expired - Fee Related
- 2004-09-01 EP EP04762799A patent/EP1664060A1/en not_active Withdrawn
- 2004-09-01 UA UAA200603678A patent/UA91496C2/ru unknown
- 2004-09-01 JP JP2006525046A patent/JP4745233B2/ja not_active Expired - Fee Related
- 2004-09-01 ME MEP-17/08A patent/MEP1708A/xx unknown
- 2004-09-01 EA EA200600542A patent/EA200600542A1/ru unknown
- 2004-09-01 NZ NZ545178A patent/NZ545178A/en not_active IP Right Cessation
- 2004-09-01 ZA ZA200602178A patent/ZA200602178B/en unknown
- 2004-09-01 AU AU2004270323A patent/AU2004270323B2/en not_active Ceased
2006
- 2006-02-28 IS IS8333A patent/IS8333A/is unknown
- 2006-03-02 IL IL174070A patent/IL174070A/en not_active IP Right Cessation
- 2006-03-29 NO NO20061424A patent/NO20061424L/no not_active Application Discontinuation

Also Published As

Publication number	Publication date
US7371863B2 (en)	2008-05-13
EA200600542A1 (ru)	2006-08-25
JP2007504179A (ja)	2007-03-01
HK1096398A1 (en)	2007-06-01
EP1664060A1 (en)	2006-06-07
IL174070A0 (en)	2006-08-01
CN1845928A (zh)	2006-10-11
AR045540A1 (es)	2005-11-02
IL174070A (en)	2011-03-31
CA2537840C (en)	2011-10-25
AU2004270323B2 (en)	2010-01-07
NZ545178A (en)	2009-11-27
CN101497619A (zh)	2009-08-05
US20070112198A1 (en)	2007-05-17
CA2537840A1 (en)	2005-03-17
BRPI0413741A (pt)	2006-10-24
KR20060069482A (ko)	2006-06-21
CN100482668C (zh)	2009-04-29
RS20060157A (sr)	2008-06-05
MEP1708A (xx)	2010-02-10
ZA200602178B (en)	2007-07-25
IS8333A (is)	2006-02-28
JP4745233B2 (ja)	2011-08-10
UA91496C2 (en)	2010-08-10
WO2005023820A1 (en)	2005-03-17
AU2004270323A1 (en)	2005-03-17
MXPA06002434A (es)	2006-06-20

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Legal Events

Date	Code	Title	Description
2008-07-14	CREP	Change of representative	Representative=s name: PLOUGMANN & VINGTOFT, POSTBOKS 1003 SENTRUM, 0104
2013-04-22	FC2A	Withdrawal, rejection or dismissal of laid open patent application