NO20062004L - Forlenget frigjoring farmasoytiske blandinger omfattene aplindor og derivater derav - Google Patents

Forlenget frigjoring farmasoytiske blandinger omfattene aplindor og derivater derav

Info

Publication number
NO20062004L
NO20062004L NO20062004A NO20062004A NO20062004L NO 20062004 L NO20062004 L NO 20062004L NO 20062004 A NO20062004 A NO 20062004A NO 20062004 A NO20062004 A NO 20062004A NO 20062004 L NO20062004 L NO 20062004L
Authority
NO
Norway
Prior art keywords
aplindor
derivatives
pharmaceutical compositions
compositions include
release pharmaceutical
Prior art date
Application number
NO20062004A
Other languages
English (en)
Inventor
Wendy Ann Dulin
Eric J Benjamin
Yanning Lin
Kai Zhuang
Original Assignee
Wyeth Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34572826&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20062004(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Wyeth Corp filed Critical Wyeth Corp
Publication of NO20062004L publication Critical patent/NO20062004L/no

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/407—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Neurology (AREA)
  • Organic Chemistry (AREA)
  • Biomedical Technology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Psychiatry (AREA)
  • Psychology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Foreliggende oppfinnelse tilveiebringer kontroUert frigjøring doseringsformuleringer av forbindelser med Formel (I): (CH2)¿¿z eUer farmasøytisk akseptable salter derav og spesielt, aplindor. Doseringsformene er anvendelige, bl. a. for å redusere bivfrkninger fra adminisfrering av slike forbindelser.
NO20062004A 2003-10-29 2006-05-04 Forlenget frigjoring farmasoytiske blandinger omfattene aplindor og derivater derav NO20062004L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US51531503P 2003-10-29 2003-10-29
PCT/US2004/036013 WO2005044262A1 (en) 2003-10-29 2004-10-28 Sustained release pharmaceutical compositions comprising aplindore and derivatives thereof

Publications (1)

Publication Number Publication Date
NO20062004L true NO20062004L (no) 2006-07-07

Family

ID=34572826

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20062004A NO20062004L (no) 2003-10-29 2006-05-04 Forlenget frigjoring farmasoytiske blandinger omfattene aplindor og derivater derav

Country Status (21)

Country Link
US (5) US20050095292A1 (no)
EP (1) EP1675583B1 (no)
JP (1) JP5547865B2 (no)
KR (1) KR101409724B1 (no)
CN (2) CN1874767A (no)
AR (1) AR046222A1 (no)
AU (1) AU2004286855B2 (no)
BR (1) BRPI0415953B8 (no)
CA (1) CA2543045C (no)
ES (1) ES2405404T3 (no)
GT (1) GT200400218A (no)
IL (1) IL174958A (no)
MX (1) MXPA06004752A (no)
NO (1) NO20062004L (no)
PA (1) PA8616201A1 (no)
PE (1) PE20050484A1 (no)
RU (1) RU2376988C2 (no)
SG (1) SG147450A1 (no)
TW (1) TW200517106A (no)
WO (1) WO2005044262A1 (no)
ZA (1) ZA200603409B (no)

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US8858993B2 (en) * 2005-07-25 2014-10-14 Metrics, Inc. Coated tablet with zero-order or near zero-order release kinetics
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US20070134322A1 (en) * 2005-12-14 2007-06-14 Forest Laboratories, Inc. Modified and pulsatile release pharmaceutical formulations of escitalopram
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JP5657565B2 (ja) * 2008-12-22 2015-01-21 ノバルティス アーゲー Ｓ１ｐ受容体アゴニストの投与レジメン
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EP2468264A1 (en) * 2010-12-27 2012-06-27 Laboratorios Liconsa, S.A. Oral pharmaceutical tablet for controled release of mesalazine and process for obtaining it
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US10980747B2 (en) * 2017-11-27 2021-04-20 Shin-Etsu Chemical Co., Ltd. Composition for solid preparation, solid preparation, and method for producing the same
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KR102408292B1 (ko) * 2018-09-28 2022-06-10 카루나 세러퓨틱스 인코포레이티드 무스카린성 수용체 활성화에 의해 개선된 장애의 치료를 위한 조성물 및 방법
TWI841545B (zh) * 2018-12-12 2024-05-11 日商田邊三菱製藥股份有限公司 耐胃性控制釋放經口劑型
CN113559074B (zh) * 2020-06-28 2023-04-21 海创药业股份有限公司 一种喹啉类化合物缓释片及其制备方法
CN116549406B (zh) * 2023-05-23 2023-12-19 北京丰科睿泰医药科技有限公司 一种盐酸曲唑酮缓释片剂
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Also Published As

Publication number Publication date
JP5547865B2 (ja) 2014-07-16
ES2405404T3 (es) 2013-05-31
US11179369B2 (en) 2021-11-23
BRPI0415953A (pt) 2007-01-02
AR046222A1 (es) 2005-11-30
US20230061743A1 (en) 2023-03-02
TW200517106A (en) 2005-06-01
US20200138781A1 (en) 2020-05-07
US20050095292A1 (en) 2005-05-05
RU2376988C2 (ru) 2009-12-27
PA8616201A1 (es) 2005-05-24
CA2543045A1 (en) 2005-05-19
US20180193311A1 (en) 2018-07-12
US10292966B2 (en) 2019-05-21
MXPA06004752A (es) 2006-07-05
RU2006118321A (ru) 2007-12-10
US20180344695A1 (en) 2018-12-06
EP1675583B1 (en) 2013-02-27
CN102335116A (zh) 2012-02-01
SG147450A1 (en) 2008-11-28
US10463648B2 (en) 2019-11-05
KR101409724B1 (ko) 2014-06-19
AU2004286855B2 (en) 2011-04-21
GT200400218A (es) 2005-06-06
IL174958A0 (en) 2008-04-13
JP2007509970A (ja) 2007-04-19
AU2004286855A1 (en) 2005-05-19
CN1874767A (zh) 2006-12-06
WO2005044262A1 (en) 2005-05-19
PE20050484A1 (es) 2005-10-13
BRPI0415953B1 (pt) 2018-12-26
ZA200603409B (en) 2010-10-27
IL174958A (en) 2012-08-30
HK1089394A1 (en) 2006-12-01
EP1675583A1 (en) 2006-07-05
CA2543045C (en) 2013-12-17
KR20060110281A (ko) 2006-10-24
BRPI0415953B8 (pt) 2021-05-25

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