NO20072371L - Kinuklidinderivater og deres anvendelse som muskarine M3-reseptorantagonister - Google Patents

Kinuklidinderivater og deres anvendelse som muskarine M3-reseptorantagonister

Info

Publication number
NO20072371L
NO20072371L NO20072371A NO20072371A NO20072371L NO 20072371 L NO20072371 L NO 20072371L NO 20072371 A NO20072371 A NO 20072371A NO 20072371 A NO20072371 A NO 20072371A NO 20072371 L NO20072371 L NO 20072371L
Authority
NO
Norway
Prior art keywords
muscarinic
kinuclidine
derivatives
receptor antagonists
compounds
Prior art date
Application number
NO20072371A
Other languages
English (en)
Inventor
Neil John Press
Stephen Paul Collingwood
Brian Cox
Urs Baettig
Simon James Watson
Sudhakar Devidasrao Garad
Hyungchul Kim
Dimitris Papoutsakis
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=33515948&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20072371(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of NO20072371L publication Critical patent/NO20072371L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/16—Central respiratory analeptics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Cosmetics (AREA)
  • Hydrogenated Pyridines (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Det beskrives forbindelser med formel (I) i salt- eller zwitterionisk form, der,, Rog Rhar de betydninger som er angitt i beskrivelsen. Forbindelsene er nyttige for behandling av tilstander som medieres av den muskariniske M3 reseptor og særlig infiammatoriske eller obstmktive luftveissykdommer. Farmasøytiske preparater som inneholder forbindelsene og en fremgangsmåte for fremstilling av forbindelsen er også beskrevet.
NO20072371A 2004-11-02 2007-05-08 Kinuklidinderivater og deres anvendelse som muskarine M3-reseptorantagonister NO20072371L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0424284.8A GB0424284D0 (en) 2004-11-02 2004-11-02 Organic compounds
PCT/EP2005/011662 WO2006048225A1 (en) 2004-11-02 2005-10-31 Quinuclidine derivatives and their use as muscarinic m3 receptor antagonists

Publications (1)

Publication Number Publication Date
NO20072371L true NO20072371L (no) 2007-07-12

Family

ID=33515948

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20072371A NO20072371L (no) 2004-11-02 2007-05-08 Kinuklidinderivater og deres anvendelse som muskarine M3-reseptorantagonister

Country Status (33)

Country Link
US (2) US7723356B2 (no)
EP (2) EP2206499A1 (no)
JP (1) JP4950896B2 (no)
KR (1) KR101252307B1 (no)
CN (1) CN101056634B (no)
AR (1) AR054090A1 (no)
AT (1) ATE481099T1 (no)
AU (1) AU2005300710B2 (no)
BR (1) BRPI0517945A (no)
CA (1) CA2583237C (no)
CY (1) CY1110952T1 (no)
DE (1) DE602005023639D1 (no)
DK (1) DK1811999T3 (no)
EC (1) ECSP077424A (no)
ES (1) ES2353142T3 (no)
GB (1) GB0424284D0 (no)
HR (1) HRP20100693T1 (no)
IL (1) IL182695A0 (no)
JO (1) JO2613B1 (no)
MA (1) MA29080B1 (no)
MX (1) MX2007005189A (no)
MY (1) MY145207A (no)
NO (1) NO20072371L (no)
NZ (1) NZ554302A (no)
PE (1) PE20060609A1 (no)
PL (1) PL1811999T3 (no)
PT (1) PT1811999E (no)
RU (1) RU2399620C2 (no)
SI (1) SI1811999T1 (no)
TN (1) TNSN07164A1 (no)
TW (1) TW200628154A (no)
WO (1) WO2006048225A1 (no)
ZA (1) ZA200702772B (no)

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KR20130111968A (ko) * 2010-06-22 2013-10-11 키에시 파르마슈티시 엣스. 피. 에이. 알칼로이드 아미노에스테르 유도체 및 이의 의약 조성물
WO2012034095A1 (en) 2010-09-09 2012-03-15 Irm Llc Compounds and compositions as trk inhibitors
UY33597A (es) 2010-09-09 2012-04-30 Irm Llc Compuestos y composiciones como inhibidores de la trk
BR112013021638A2 (pt) 2011-02-25 2016-08-02 Irm Llc "compostos inibidores de trk, seu uso e composições que os compreendem"
JP2011195593A (ja) * 2011-06-30 2011-10-06 Astrazeneca Ab ムスカリンｍ３受容体アンタゴニストとしてのキヌクリジン誘導体
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US20170065589A1 (en) * 2014-05-06 2017-03-09 Anthony G. Visco Methods of treating or preventing preterm labor
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MY145207A (en) 2012-01-13
US8084463B2 (en) 2011-12-27
KR101252307B1 (ko) 2013-04-08
DK1811999T3 (da) 2010-12-13
PT1811999E (pt) 2010-10-29
TNSN07164A1 (en) 2008-11-21
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US20100168132A1 (en) 2010-07-01
JP4950896B2 (ja) 2012-06-13
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