NO20070686L - 17-Desmetylrapamucin og analoger av det, framgangsmater for framstilling av disse, og bruk av disse som immunosupressanter, antikreft-forbindelser, soppdrepende forbindelser, osv - Google Patents

17-Desmetylrapamucin og analoger av det, framgangsmater for framstilling av disse, og bruk av disse som immunosupressanter, antikreft-forbindelser, soppdrepende forbindelser, osv

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Publication number
NO20070686L
NO20070686L NO20070686A NO20070686A NO20070686L NO 20070686 L NO20070686 L NO 20070686L NO 20070686 A NO20070686 A NO 20070686A NO 20070686 A NO20070686 A NO 20070686A NO 20070686 L NO20070686 L NO 20070686L
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NO
Norway
Prior art keywords
compounds
analogs
diseases
processes
desmethylrapamucine
Prior art date
Application number
NO20070686A
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English (en)
Norwegian (no)
Inventor
Matthew Alan Gregory
Christine Janet Martin
Original Assignee
Biotica Tech Ltd
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Publication date
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Publication of NO20070686L publication Critical patent/NO20070686L/no

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/18—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/436—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having oxygen as a ring hetero atom, e.g. rapamycin
    • A—HUMAN NECESSITIES
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    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/14—Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers

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  • Health & Medical Sciences (AREA)
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  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Immunology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pulmonology (AREA)
  • Oncology (AREA)
  • Dermatology (AREA)
  • Vascular Medicine (AREA)
  • Rheumatology (AREA)
  • Psychology (AREA)
  • Urology & Nephrology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Communicable Diseases (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pain & Pain Management (AREA)
  • Hematology (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Transplantation (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
NO20070686A 2004-08-11 2007-02-06 17-Desmetylrapamucin og analoger av det, framgangsmater for framstilling av disse, og bruk av disse som immunosupressanter, antikreft-forbindelser, soppdrepende forbindelser, osv NO20070686L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0417852.1A GB0417852D0 (en) 2004-08-11 2004-08-11 Production of polyketides and other natural products
PCT/GB2005/003158 WO2006016167A2 (en) 2004-08-11 2005-08-11 17-desmethylrapamycin and analogues thereof, methods for their roduction and their use as immunosupressants, anticancer agents, antifungal agents, etc.

Publications (1)

Publication Number Publication Date
NO20070686L true NO20070686L (no) 2007-04-25

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NO20070686A NO20070686L (no) 2004-08-11 2007-02-06 17-Desmetylrapamucin og analoger av det, framgangsmater for framstilling av disse, og bruk av disse som immunosupressanter, antikreft-forbindelser, soppdrepende forbindelser, osv

Country Status (19)

Country Link
US (1) US7803808B2 (es)
EP (2) EP2029611A2 (es)
JP (1) JP2008509895A (es)
KR (1) KR20070052784A (es)
CN (2) CN101056880A (es)
AU (1) AU2005270989B2 (es)
BR (1) BRPI0514236A (es)
CA (1) CA2575582A1 (es)
CR (1) CR8990A (es)
EC (1) ECSP077303A (es)
GB (1) GB0417852D0 (es)
IL (1) IL181171A0 (es)
MX (1) MX2007001809A (es)
NO (1) NO20070686L (es)
NZ (1) NZ553074A (es)
RU (2) RU2430922C2 (es)
UA (1) UA95895C2 (es)
WO (1) WO2006016167A2 (es)
ZA (1) ZA200701622B (es)

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WO2006016167A3 (en) 2006-04-13
BRPI0514236A (pt) 2008-06-03
US20090253732A1 (en) 2009-10-08
RU2007108772A (ru) 2008-09-20
RU2430922C2 (ru) 2011-10-10
AU2005270989A1 (en) 2006-02-16
US7803808B2 (en) 2010-09-28
ECSP077303A (es) 2007-04-26
NZ553074A (en) 2011-01-28
GB0417852D0 (en) 2004-09-15
ZA200701622B (en) 2008-06-25
EP2471797B1 (en) 2016-02-03
JP2008509895A (ja) 2008-04-03
RU2009140290A (ru) 2011-05-10
IL181171A0 (en) 2007-07-04
CN101056880A (zh) 2007-10-17
EP2029611A2 (en) 2009-03-04
CN101805748A (zh) 2010-08-18
UA95895C2 (ru) 2011-09-26
AU2005270989B2 (en) 2012-04-05
CR8990A (es) 2009-01-14
MX2007001809A (es) 2007-10-08
CA2575582A1 (en) 2006-02-16
KR20070052784A (ko) 2007-05-22

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