NO20072454L - Pyridinderivater, fremstillingen og den terapeutiske anvendelse derav - Google Patents

Pyridinderivater, fremstillingen og den terapeutiske anvendelse derav

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Publication number
NO20072454L
NO20072454L NO20072454A NO20072454A NO20072454L NO 20072454 L NO20072454 L NO 20072454L NO 20072454 A NO20072454 A NO 20072454A NO 20072454 A NO20072454 A NO 20072454A NO 20072454 L NO20072454 L NO 20072454L
Authority
NO
Norway
Prior art keywords
preparation
therapeutic use
pyridine derivatives
group
substituted
Prior art date
Application number
NO20072454A
Other languages
English (en)
Inventor
Christian Congy
Francis Barth
Murielle Rinaldi-Carmona
Philippe Pointeau
Lionel Barre
Original Assignee
Sanofi Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of NO20072454L publication Critical patent/NO20072454L/no

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    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
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Abstract

Oppfinnelsen er relatert til forbindelser av formel (1), hvor Z er en N(R1)XR2, N(R1)COOR'2 eller OCON(R1)R'2 gruppe; X er en -CO-, -SO2-, -CON(R10)- eller -CSN(R10)-; R1 er et hydrogenatom eller en (Cl-C4)alkylgruppe; R2 er en (C3-C10)alkylgruppe, en (C3-C12) karboksyklisk ikke-aromatisk radikal, en heterocyklisk radikal, en ikke-substituert eller substituert fenyl og en (C1-C2) alkylen substituert ved en eller to like eller forskjellige substituenter; R3 er et hydrogenatom, eller en (Cl-C4) alkyl, cyano, (Cl-C4) alkoksymetyl eller hydroksymetyl gruppe. Den oppfunnede fremgangsmåten kan bli benyttet for å fremstille og terapeutisk benytte nevnte forbindelser.
NO20072454A 2004-10-18 2007-05-14 Pyridinderivater, fremstillingen og den terapeutiske anvendelse derav NO20072454L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0411030A FR2876691B1 (fr) 2004-10-18 2004-10-18 Derives de pyridine, leur preparation, leur application en therapeutique
PCT/FR2005/002566 WO2006042955A1 (fr) 2004-10-18 2005-10-17 Derives de pyridine, leur preparation, leur application en therapeutique

Publications (1)

Publication Number Publication Date
NO20072454L true NO20072454L (no) 2007-05-14

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FR2899899A1 (fr) * 2006-04-14 2007-10-19 Sanofi Aventis Sa Derives d'aminomethyl pyridine, leur preparation et leur application en therapeutique
TW200815438A (en) * 2006-06-13 2008-04-01 Bayer Schering Pharma Ag Substituted pyrazolopyridines and salts thereof, pharmaceutical compositions comprising same, methods of preparing same and uses of same
US7781593B2 (en) 2006-09-14 2010-08-24 Hoffmann-La Roche Inc. 5-phenyl-nicotinamide derivatives
FR2922209B1 (fr) 2007-10-12 2010-06-11 Sanofi Aventis 5,6-DIARYLES PYRIDINES SUBSTITUES EN POSITION 2 et 3, LEUR PREPARATION ET LEUR APPLICATION EN THERAPEUTIQUE.
ES2459468T3 (es) 2009-05-15 2014-05-09 Novartis Ag Arilpiridinas como inhibidores de aldosterona sintasa
EP3495348A4 (en) 2016-07-29 2020-01-22 Toray Industries, Inc. GUANIDINE DERIVATIVE AND ITS USE FOR MEDICAL PURPOSES
WO2018159650A1 (ja) * 2017-02-28 2018-09-07 東レ株式会社 グアニジン誘導体及びその医薬用途

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FR2198737B1 (no) * 1972-09-13 1975-11-28 Serdex
US5686470A (en) * 1995-02-10 1997-11-11 Weier; Richard M. 2, 3-substituted pyridines for the treatment of inflammation
WO2002055502A1 (en) * 2001-01-02 2002-07-18 Fujisawa Pharmaceutical Co., Ltd. Pyridine derivatives useful as cyclooxygenase inhibitor
EP1492784A4 (en) * 2002-03-28 2006-03-29 Merck & Co Inc SUBSTITUTED 2,3-DIPHENYLPYRIDINES
FR2838439B1 (fr) * 2002-04-11 2005-05-20 Sanofi Synthelabo Derives de terphenyle, leur preparation, les compositions pharmaceutqiues en contenant
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CN101039912A (zh) 2007-09-19
WO2006042955A1 (fr) 2006-04-27
EA200700891A1 (ru) 2007-08-31
KR20070063008A (ko) 2007-06-18
UY29163A1 (es) 2006-04-28
MX2007004482A (es) 2007-06-13
CA2582778A1 (fr) 2006-04-27
IL182385A0 (en) 2007-07-24
TNSN07114A1 (fr) 2008-06-02
FR2876691B1 (fr) 2006-12-29
EP1805143A1 (fr) 2007-07-11
BRPI0516926A (pt) 2008-09-23
PE20060584A1 (es) 2006-08-18
ECSP077400A (es) 2007-05-30
AR051221A1 (es) 2006-12-27
MA29016B1 (fr) 2007-11-01
TW200628450A (en) 2006-08-16
JP2008516934A (ja) 2008-05-22
AU2005296959A1 (en) 2006-04-27
FR2876691A1 (fr) 2006-04-21
US20080021070A1 (en) 2008-01-24

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