NO20074647L - 3,4 dihydro-1H-isoquinolin-2-karboksylsyre-5-ammopyridin-2-yl estere - Google Patents

3,4 dihydro-1H-isoquinolin-2-karboksylsyre-5-ammopyridin-2-yl estere

Info

Publication number
NO20074647L
NO20074647L NO20074647A NO20074647A NO20074647L NO 20074647 L NO20074647 L NO 20074647L NO 20074647 A NO20074647 A NO 20074647A NO 20074647 A NO20074647 A NO 20074647A NO 20074647 L NO20074647 L NO 20074647L
Authority
NO
Norway
Prior art keywords
ammopyridin
isoquinoline
dihydro
esters
carboxylic acid
Prior art date
Application number
NO20074647A
Other languages
English (en)
Inventor
Poul Jacobsen
Johannes Cornelis De Jong
Original Assignee
Novo Nordisk As
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novo Nordisk As filed Critical Novo Nordisk As
Publication of NO20074647L publication Critical patent/NO20074647L/no

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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/472—Non-condensed isoquinolines, e.g. papaverine
    • A61K31/4725—Non-condensed isoquinolines, e.g. papaverine containing further heterocyclic rings
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    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

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Abstract

Nye forbindelser av formel (I), farmasøytiske sammensetninger som omfatter dem og anvendelse derav i behandlingen og/eller forhindringen av sykdommer og lidelser relatert til hormonsensitiv lipase. Mer spesielt er forbindelsene anvendelige for behandlingen og/eller forhindringen av sykdommer og lidelser i hvilke modulering av aktiviteten til hormonsensitiv lipase er fordelaktig.
NO20074647A 2005-02-15 2007-09-12 3,4 dihydro-1H-isoquinolin-2-karboksylsyre-5-ammopyridin-2-yl estere NO20074647L (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DKPA200500222 2005-02-15
DKPA200500295 2005-02-28
PCT/EP2006/050882 WO2006087309A1 (en) 2005-02-15 2006-02-13 3,4-dihydro-1h-isoquinoline-2-carboxylic acid 5-aminopyridin-2-yl esters

Publications (1)

Publication Number Publication Date
NO20074647L true NO20074647L (no) 2007-11-09

Family

ID=36360334

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20074647A NO20074647L (no) 2005-02-15 2007-09-12 3,4 dihydro-1H-isoquinolin-2-karboksylsyre-5-ammopyridin-2-yl estere

Country Status (12)

Country Link
US (1) US20080227792A1 (no)
EP (1) EP1853585A1 (no)
JP (1) JP2008530174A (no)
KR (1) KR20070107000A (no)
AU (1) AU2006215608A1 (no)
BR (1) BRPI0607545A2 (no)
CA (1) CA2596522A1 (no)
IL (1) IL184120A0 (no)
MX (1) MX2007009782A (no)
NO (1) NO20074647L (no)
RU (1) RU2007128987A (no)
WO (1) WO2006087309A1 (no)

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AU2006215608A1 (en) 2006-08-24
WO2006087309A1 (en) 2006-08-24
US20080227792A1 (en) 2008-09-18
RU2007128987A (ru) 2009-03-27
BRPI0607545A2 (pt) 2016-11-01
EP1853585A1 (en) 2007-11-14
JP2008530174A (ja) 2008-08-07
MX2007009782A (es) 2007-08-22
CA2596522A1 (en) 2006-08-24
IL184120A0 (en) 2007-10-31
KR20070107000A (ko) 2007-11-06

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