NO20074763L - (1,5-difenyl-1H-pyrazol-3-yl)oksadiazolderivater, fremgangsmate ved fremstilling derav og anvendelse av samme i terapi - Google Patents

(1,5-difenyl-1H-pyrazol-3-yl)oksadiazolderivater, fremgangsmate ved fremstilling derav og anvendelse av samme i terapi

Info

Publication number: NO20074763L
Authority: NO; Norway
Prior art keywords: pyrazol; diphenyl; therapy; preparation; same
Prior art date: 2005-02-21

Application number

NO20074763A

Other languages

English (en)

Norwegian (no)

Inventor

Christian Congy

Patrick Gueule

Francis Barth

Murielle Rinaldi-Carmona

Didier Van Broeck

Original Assignee

Sanofi Aventis

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2005-02-21

Filing date

2007-09-18

Publication date

2007-11-16

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=35079215&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20074763(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2007-09-18 Application filed by Sanofi Aventis filed Critical Sanofi Aventis

2007-11-16 Publication of NO20074763L publication Critical patent/NO20074763L/no

Links

UPWOUOHVXSRHDB-UHFFFAOYSA-N 4-(1,5-diphenylpyrazol-3-yl)oxadiazole Chemical class O1N=NC(C2=NN(C(C=3C=CC=CC=3)=C2)C=2C=CC=CC=2)=C1 UPWOUOHVXSRHDB-UHFFFAOYSA-N 0.000 title 1
238000000034 method Methods 0.000 title 1
238000002560 therapeutic procedure Methods 0.000 title 1
125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 2
125000000217 alkyl group Chemical group 0.000 abstract 1
150000001875 compounds Chemical class 0.000 abstract 1
125000004093 cyano group Chemical group *C#N 0.000 abstract 1
150000004677 hydrates Chemical class 0.000 abstract 1
239000000203 mixture Substances 0.000 abstract 1
239000012453 solvate Substances 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4245—Oxadiazoles
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Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Pharmacology & Pharmacy (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Engineering & Computer Science (AREA)
Chemical Kinetics & Catalysis (AREA)
Bioinformatics & Cheminformatics (AREA)
Neurosurgery (AREA)
Neurology (AREA)
Biomedical Technology (AREA)
Diabetes (AREA)
Pain & Pain Management (AREA)
Psychiatry (AREA)
Physical Education & Sports Medicine (AREA)
Rheumatology (AREA)
Endocrinology (AREA)
Addiction (AREA)
Cardiology (AREA)
Orthopedic Medicine & Surgery (AREA)
Hematology (AREA)
Urology & Nephrology (AREA)
Immunology (AREA)
Heart & Thoracic Surgery (AREA)
Obesity (AREA)
Vascular Medicine (AREA)
Reproductive Health (AREA)
Ophthalmology & Optometry (AREA)
Pulmonology (AREA)
Oncology (AREA)
Hospice & Palliative Care (AREA)
Communicable Diseases (AREA)
Child & Adolescent Psychology (AREA)

NO20074763A 2005-02-21 2007-09-18 (1,5-difenyl-1H-pyrazol-3-yl)oksadiazolderivater, fremgangsmate ved fremstilling derav og anvendelse av samme i terapi NO20074763L (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
FR0501860A FR2882365B1 (fr)	2005-02-21	2005-02-21	Derives de 2-(1,5-diphenyl-1h-pyrazol-3-yl)-1,3,4-oxadiazole leur preparation et leur application en therapeutique
PCT/FR2006/000368 WO2006087480A1 (fr)	2005-02-21	2006-02-17	DERIVES DE (l,5-DIPHENYL-lH-PYRAZOL-3-YL)OXADIAZOLE, LEUR PREPARATION ET LEUR APPLICATION EN THERAPEUTIQUE

Publications (1)

Publication Number	Publication Date
NO20074763L true NO20074763L (no)	2007-11-16

Family

ID=35079215

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO20074763A NO20074763L (no)	2005-02-21	2007-09-18	(1,5-difenyl-1H-pyrazol-3-yl)oksadiazolderivater, fremgangsmate ved fremstilling derav og anvendelse av samme i terapi

Country Status (25)

Country	Link
US (1)	US7632852B2 (pt)
EP (1)	EP1853595A1 (pt)
JP (1)	JP4812778B2 (pt)
KR (1)	KR20070107053A (pt)
CN (1)	CN101119990A (pt)
AR (1)	AR055560A1 (pt)
AU (1)	AU2006215443A1 (pt)
BR (1)	BRPI0606845A2 (pt)
CA (1)	CA2597359A1 (pt)
DO (1)	DOP2006000045A (pt)
EA (1)	EA200701779A1 (pt)
FR (1)	FR2882365B1 (pt)
GT (1)	GT200600082A (pt)
IL (1)	IL185163A0 (pt)
MA (1)	MA29261B1 (pt)
MX (1)	MX2007009994A (pt)
NO (1)	NO20074763L (pt)
NZ (1)	NZ560790A (pt)
PA (1)	PA8663901A1 (pt)
PE (1)	PE20061038A1 (pt)
SV (1)	SV2007002422A (pt)
TW (1)	TW200640916A (pt)
UY (1)	UY29388A1 (pt)
WO (1)	WO2006087480A1 (pt)
ZA (1)	ZA200706953B (pt)

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AU2007283113A1 (en)	2006-08-08	2008-02-14	Sanofi-Aventis	Arylaminoaryl-alkyl-substituted imidazolidine-2,4-diones, processes for preparing them, medicaments comprising these compounds, and their use
WO2008039023A1 (en) *	2006-09-29	2008-04-03	Green Cross Corporation	Heteroaryl-pyrazole derivatives as cannabinoid cb1 receptor antagonists
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EP2025674A1 (de)	2007-08-15	2009-02-18	sanofi-aventis	Substituierte Tetrahydronaphthaline, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel
WO2009078498A1 (en) *	2007-12-17	2009-06-25	Green Cross Corporation	Biarylpyrazole 4-carboxamides as cannabinoid cb1 receptor ligands
UY31968A (es)	2008-07-09	2010-01-29	Sanofi Aventis	Nuevos derivados heterocíclicos, sus procesos para su preparación, y sus usos terapéuticos
WO2010035915A1 (en) *	2008-09-25	2010-04-01	Green Cross Corporation	Sulfur containing pyrazole-heterocycle derivatives as cannabinoid cb1 receptor antagonists
WO2010068601A1 (en)	2008-12-08	2010-06-17	Sanofi-Aventis	A crystalline heteroaromatic fluoroglycoside hydrate, processes for making, methods of use and pharmaceutical compositions thereof
KR20120060207A (ko)	2009-08-26	2012-06-11	사노피	신규한 결정성 헤테로방향족 플루오로글리코시드 수화물, 이들 화합물을 포함하는 약제 및 이들의 용도
EP2582709B1 (de)	2010-06-18	2018-01-24	Sanofi	Azolopyridin-3-on-derivate als inhibitoren von lipasen und phospholipasen
EP2683704B1 (de)	2011-03-08	2014-12-17	Sanofi	Verzweigte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung
US8710050B2 (en)	2011-03-08	2014-04-29	Sanofi	Di and tri- substituted oxathiazine derivatives, method for the production, method for the production thereof, use thereof as medicine and drug containing said derivatives and use thereof
US8871758B2 (en)	2011-03-08	2014-10-28	Sanofi	Tetrasubstituted oxathiazine derivatives, method for producing them, their use as medicine and drug containing said derivatives and the use thereof
EP2766349B1 (de)	2011-03-08	2016-06-01	Sanofi	Mit carbozyklen oder heterozyklen substituierte oxathiazinderivate, verfahren zu deren herstellung, diese verbindungen enthaltende arzneimittel und deren verwendung
US8828994B2 (en)	2011-03-08	2014-09-09	Sanofi	Di- and tri-substituted oxathiazine derivatives, method for the production thereof, use thereof as medicine and drug containing said derivatives and use thereof
CN109651350B (zh) *	2019-01-11	2022-05-24	贵州大学	一类杂环取代的1,3,4-噁(噻)二唑类化合物及其制备方法和用途
CN109942567B (zh) *	2019-04-30	2023-04-07	贵州大学	一种1,3,4-噁(噻)二唑基的咪唑类化合物及其制备方法和用途

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MXPA05004115A (es) *	2002-10-18	2005-06-22	Pfizer Prod Inc	Ligandos del receptor cannabionoide y usos de los mismos.
BR0316332A (pt) *	2002-12-02	2005-09-27	Astellas Pharma Inc	Composto pirazólico, composição farmacêutica e agente analgésico contendo o mesmo, processo para sua preparação e seu uso e pacote comercial
FR2856683A1 (fr) *	2003-06-25	2004-12-31	Sanofi Synthelabo	Derives de 4-cyanopyrazole-3-carboxamide, leur preparation et leur application en therapeutique

2005
- 2005-02-21 FR FR0501860A patent/FR2882365B1/fr not_active Expired - Fee Related
2006
- 2006-02-17 ZA ZA200706953A patent/ZA200706953B/xx unknown
- 2006-02-17 JP JP2007555667A patent/JP4812778B2/ja not_active Expired - Fee Related
- 2006-02-17 WO PCT/FR2006/000368 patent/WO2006087480A1/fr not_active Ceased
- 2006-02-17 PE PE2006000202A patent/PE20061038A1/es not_active Application Discontinuation
- 2006-02-17 CA CA002597359A patent/CA2597359A1/fr not_active Abandoned
- 2006-02-17 BR BRPI0606845-6A patent/BRPI0606845A2/pt not_active IP Right Cessation
- 2006-02-17 EP EP06709338A patent/EP1853595A1/fr not_active Withdrawn
- 2006-02-17 KR KR1020077019014A patent/KR20070107053A/ko not_active Withdrawn
- 2006-02-17 CN CNA2006800049844A patent/CN101119990A/zh active Pending
- 2006-02-17 EA EA200701779A patent/EA200701779A1/ru unknown
- 2006-02-17 AU AU2006215443A patent/AU2006215443A1/en not_active Abandoned
- 2006-02-17 MX MX2007009994A patent/MX2007009994A/es not_active Application Discontinuation
- 2006-02-17 NZ NZ560790A patent/NZ560790A/en unknown
- 2006-02-20 TW TW095105632A patent/TW200640916A/zh unknown
- 2006-02-20 DO DO2006000045A patent/DOP2006000045A/es unknown
- 2006-02-20 GT GT200600082A patent/GT200600082A/es unknown
- 2006-02-21 UY UY29388A patent/UY29388A1/es not_active Application Discontinuation
- 2006-02-21 PA PA20068663901A patent/PA8663901A1/es unknown
- 2006-02-21 SV SV2006002422A patent/SV2007002422A/es unknown
- 2006-02-21 AR ARP060100610A patent/AR055560A1/es unknown
2007
- 2007-08-08 US US11/835,670 patent/US7632852B2/en not_active Expired - Fee Related
- 2007-08-09 IL IL185163A patent/IL185163A0/en unknown
- 2007-08-23 MA MA30157A patent/MA29261B1/fr unknown
- 2007-09-18 NO NO20074763A patent/NO20074763L/no not_active Application Discontinuation

Also Published As

Publication number	Publication date
JP2008530188A (ja)	2008-08-07
MX2007009994A (es)	2007-10-10
FR2882365B1 (fr)	2007-09-07
PE20061038A1 (es)	2006-11-24
DOP2006000045A (es)	2006-11-15
SV2007002422A (es)	2007-01-17
AR055560A1 (es)	2007-08-22
BRPI0606845A2 (pt)	2009-07-21
WO2006087480A1 (fr)	2006-08-24
US7632852B2 (en)	2009-12-15
AU2006215443A1 (en)	2006-08-24
US20080039510A1 (en)	2008-02-14
CN101119990A (zh)	2008-02-06
EA200701779A1 (ru)	2008-02-28
EP1853595A1 (fr)	2007-11-14
NZ560790A (en)	2009-08-28
FR2882365A1 (fr)	2006-08-25
UY29388A1 (es)	2006-10-02
PA8663901A1 (es)	2006-12-07
JP4812778B2 (ja)	2011-11-09
TW200640916A (en)	2006-12-01
KR20070107053A (ko)	2007-11-06
CA2597359A1 (fr)	2006-08-24
ZA200706953B (en)	2009-03-25
IL185163A0 (en)	2007-12-03
MA29261B1 (fr)	2008-02-01
GT200600082A (es)	2006-10-19

Legal Events

Date	Code	Title	Description
2011-09-26	FC2A	Withdrawal, rejection or dismissal of laid open patent application

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