NO20082350L - Piperidin-4-YL-pyridazin-3-ylamin derivat som rask dissosiasjon dopamin 2-reseptor antagonister - Google Patents

Piperidin-4-YL-pyridazin-3-ylamin derivat som rask dissosiasjon dopamin 2-reseptor antagonister

Info

Publication number
NO20082350L
NO20082350L NO20082350A NO20082350A NO20082350L NO 20082350 L NO20082350 L NO 20082350L NO 20082350 A NO20082350 A NO 20082350A NO 20082350 A NO20082350 A NO 20082350A NO 20082350 L NO20082350 L NO 20082350L
Authority
NO
Norway
Prior art keywords
receptor antagonists
dopamine
compounds
pyridazin
piperidin
Prior art date
Application number
NO20082350A
Other languages
English (en)
Norwegian (no)
Inventor
Ludo Edmond Josephine Kennis
Marcel Frans Leopold De Bruyn
Xavier Jean Michel Langlois
Yves Emiel Maria Va Roosbroeck
Gregor James Macdonald
Frans Alfons Maria Van Keybus
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of NO20082350L publication Critical patent/NO20082350L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/50—Pyridazines; Hydrogenated pyridazines
    • A61K31/501—Pyridazines; Hydrogenated pyridazines not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Epidemiology (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Psychology (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
NO20082350A 2005-10-26 2008-05-26 Piperidin-4-YL-pyridazin-3-ylamin derivat som rask dissosiasjon dopamin 2-reseptor antagonister NO20082350L (no)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
EP05110028 2005-10-26
EP06100209 2006-01-10
EP06101545 2006-02-10
PCT/EP2006/067696 WO2007048779A1 (en) 2005-10-26 2006-10-24 Piperidin-4-yl-pyridazin-3-ylamine derivatives as fast dissociating dopamine 2 receptor antagonists

Publications (1)

Publication Number Publication Date
NO20082350L true NO20082350L (no) 2008-07-01

Family

ID=35734993

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20082350A NO20082350L (no) 2005-10-26 2008-05-26 Piperidin-4-YL-pyridazin-3-ylamin derivat som rask dissosiasjon dopamin 2-reseptor antagonister

Country Status (34)

Country Link
US (3) US8940743B2 (es)
EP (1) EP1943242B1 (es)
JP (1) JP5140598B2 (es)
KR (1) KR101351910B1 (es)
CN (1) CN101291925B (es)
AP (1) AP2607A (es)
AR (1) AR058151A1 (es)
AT (1) ATE495167T1 (es)
AU (1) AU2006307930B2 (es)
BR (1) BRPI0617787A2 (es)
CA (1) CA2623160C (es)
CR (1) CR10020A (es)
CY (1) CY1111977T1 (es)
DE (1) DE602006019624D1 (es)
DK (1) DK1943242T3 (es)
EA (1) EA015681B1 (es)
EC (1) ECSP088396A (es)
ES (1) ES2359020T3 (es)
GT (1) GT200800033A (es)
HN (1) HN2008000646A (es)
HR (1) HRP20110226T1 (es)
IL (1) IL191016A (es)
JO (1) JO2769B1 (es)
MY (1) MY145609A (es)
NO (1) NO20082350L (es)
NZ (1) NZ566785A (es)
PL (1) PL1943242T3 (es)
PT (1) PT1943242E (es)
RS (1) RS51674B (es)
SI (1) SI1943242T1 (es)
TW (1) TWI399373B (es)
UA (1) UA94058C2 (es)
WO (1) WO2007048779A1 (es)
ZA (1) ZA200803668B (es)

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CA2687931C (en) * 2007-05-31 2016-05-24 Boehringer Ingelheim International Gmbh Ccr2 receptor antagonists and uses thereof
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Also Published As

Publication number Publication date
HK1124317A1 (en) 2009-07-10
HN2008000646A (es) 2011-02-16
NZ566785A (en) 2010-03-26
CY1111977T1 (el) 2015-11-04
CN101291925B (zh) 2013-04-10
US8940743B2 (en) 2015-01-27
GT200800033A (es) 2009-08-20
AP2607A (en) 2013-03-05
ZA200803668B (en) 2009-09-30
CA2623160A1 (en) 2007-05-03
MY145609A (en) 2012-03-15
HRP20110226T1 (hr) 2011-05-31
AP2008004441A0 (en) 2008-04-30
TW200732321A (en) 2007-09-01
EP1943242A1 (en) 2008-07-16
US9751860B2 (en) 2017-09-05
AU2006307930B2 (en) 2011-10-06
PT1943242E (pt) 2011-04-06
IL191016A (en) 2013-10-31
EA200801184A1 (ru) 2008-08-29
ATE495167T1 (de) 2011-01-15
AU2006307930A1 (en) 2007-05-03
US20170022181A1 (en) 2017-01-26
TWI399373B (zh) 2013-06-21
DK1943242T3 (da) 2011-04-26
RS51674B (sr) 2011-10-31
KR20080067658A (ko) 2008-07-21
ECSP088396A (es) 2008-05-30
CR10020A (es) 2009-01-16
ES2359020T3 (es) 2011-05-17
BRPI0617787A2 (pt) 2009-12-01
SI1943242T1 (sl) 2011-05-31
JP5140598B2 (ja) 2013-02-06
EA015681B1 (ru) 2011-10-31
CA2623160C (en) 2013-10-15
EP1943242B1 (en) 2011-01-12
US20080227791A1 (en) 2008-09-18
KR101351910B1 (ko) 2014-01-16
DE602006019624D1 (de) 2011-02-24
JO2769B1 (en) 2014-03-15
JP2009514815A (ja) 2009-04-09
CN101291925A (zh) 2008-10-22
WO2007048779A1 (en) 2007-05-03
US9468640B2 (en) 2016-10-18
PL1943242T3 (pl) 2011-06-30
AR058151A1 (es) 2008-01-23
US20150141432A1 (en) 2015-05-21
UA94058C2 (ru) 2011-04-11

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