NO20083898L - Amid-derivativer som ionekanalligander og farmasoytiske sammensetninger og fremgangsmater for bruk derav - Google Patents

Amid-derivativer som ionekanalligander og farmasoytiske sammensetninger og fremgangsmater for bruk derav

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Publication number
NO20083898L
NO20083898L NO20083898A NO20083898A NO20083898L NO 20083898 L NO20083898 L NO 20083898L NO 20083898 A NO20083898 A NO 20083898A NO 20083898 A NO20083898 A NO 20083898A NO 20083898 L NO20083898 L NO 20083898L
Authority
NO
Norway
Prior art keywords
pharmaceutical compositions
methods
ion channel
amide derivatives
channel ligands
Prior art date
Application number
NO20083898A
Other languages
English (en)
Norwegian (no)
Inventor
Matthew Duncton
Kiran Sahasrabudhe
Ravindra B Upasani
Guoxian Wu
Zhi-Liang Wei
Michael G Kelly
Karl J Kaub
John Kincaid
Satyanarayana Janagani
Yunfeng Fang
Matthew Kox
Original Assignee
Renovis Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from PCT/US2007/004912 external-priority patent/WO2007100758A2/fr
Application filed by Renovis Inc filed Critical Renovis Inc
Publication of NO20083898L publication Critical patent/NO20083898L/no

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    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/08—Indoles; Hydrogenated indoles with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to carbon atoms of the hetero ring
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N37/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids
    • A01N37/18—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids containing the group —CO—N<, e.g. carboxylic acid amides or imides; Thio analogues thereof
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    • C07D253/02—Heterocyclic compounds containing six-membered rings having three nitrogen atoms as the only ring hetero atoms, not provided for by group C07D251/00 not condensed with other rings
    • C07D253/06—1,2,4-Triazines
    • C07D253/065—1,2,4-Triazines having three double bonds between ring members or between ring members and non-ring members
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    • C07D215/06—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to the ring carbon atoms having only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, attached to the ring nitrogen atom
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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems

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NO20083898A 2006-02-23 2008-09-11 Amid-derivativer som ionekanalligander og farmasoytiske sammensetninger og fremgangsmater for bruk derav NO20083898L (no)

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US77610606P 2006-02-23 2006-02-23
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US77594506P 2006-02-23 2006-02-23
US77610506P 2006-02-23 2006-02-23
US77593006P 2006-02-23 2006-02-23
US77605706P 2006-02-23 2006-02-23
US77606406P 2006-02-23 2006-02-23
US77603306P 2006-02-23 2006-02-23
US77594906P 2006-02-23 2006-02-23
US83999406P 2006-08-24 2006-08-24
US83990306P 2006-08-24 2006-08-24
PCT/US2007/004912 WO2007100758A2 (fr) 2005-02-28 2007-02-22 Dérivés amides en tant que ligands de canal ionique et compositions pharmaceutiques et procédés d'utilisation de tels dérivés

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WO2005046683A1 (fr) * 2003-10-07 2005-05-26 Renovis, Inc. Derives d'amide utilises comme ligands du canal ionique et compositions pharmaceutiques et methodes d'utilisation de ces derives
WO2006006740A1 (fr) * 2004-07-14 2006-01-19 Japan Tobacco Inc. Composé 3-aminobénamide et inhibiteur d'activité à récepteur vanilloïde 1 (vr1)

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IL193346A0 (en) 2009-08-03
TNSN08328A1 (en) 2009-12-29
EA200870287A1 (ru) 2009-02-27
CO6170402A2 (es) 2010-06-18
GB2452142A8 (en) 2009-03-18
CA2641781A1 (fr) 2007-09-07
US20100004222A1 (en) 2010-01-07
GB2452142A (en) 2009-02-25

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