MA30267B1 - Derives amides en tant que ligands de canal ionique et compositions pharmaceutiques et procedes d'utilisation de tels derives - Google Patents

Derives amides en tant que ligands de canal ionique et compositions pharmaceutiques et procedes d'utilisation de tels derives

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Publication number
MA30267B1
MA30267B1 MA31218A MA31218A MA30267B1 MA 30267 B1 MA30267 B1 MA 30267B1 MA 31218 A MA31218 A MA 31218A MA 31218 A MA31218 A MA 31218A MA 30267 B1 MA30267 B1 MA 30267B1
Authority
MA
Morocco
Prior art keywords
derivatives
pharmaceutical compositions
methods
ion channel
channel ligands
Prior art date
Application number
MA31218A
Other languages
English (en)
Inventor
Michael G Kelly
Carl J Kaub
John Kincaid
Satyanarayana Janagani
Guoxian Wu
Zhi-Liang Wei
Kiran Sahasrabudhe
Matthew Duncton
Ravindra B Upasani
Yunfeng Fang
Matthew Cox
Original Assignee
Renovis Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Renovis Inc filed Critical Renovis Inc
Publication of MA30267B1 publication Critical patent/MA30267B1/fr

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    • A01N37/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids
    • A01N37/18—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids containing the group —CO—N<, e.g. carboxylic acid amides or imides; Thio analogues thereof
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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems

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  • Chemical & Material Sciences (AREA)
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  • Health & Medical Sciences (AREA)
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  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
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  • Medicinal Chemistry (AREA)
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  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Immunology (AREA)
  • Zoology (AREA)
  • Epidemiology (AREA)
  • Environmental Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Dentistry (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Urology & Nephrology (AREA)
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Abstract

La présente invention concerne des composés de formule (I). Les composés peuvent être préparés sous la forme de compositions pharmaceutiques, et peuvent être utilisés en vue de la prévention et du traitement d'une variété de conditions pathologiques chez des mammifères y compris des humains, comprenant entre autres, la douleur, l'inflammation, la lésion traumatique, et autres.
MA31218A 2006-02-23 2008-09-08 Derives amides en tant que ligands de canal ionique et compositions pharmaceutiques et procedes d'utilisation de tels derives MA30267B1 (fr)

Applications Claiming Priority (12)

Application Number Priority Date Filing Date Title
US77593006P 2006-02-23 2006-02-23
US77605806P 2006-02-23 2006-02-23
US77605606P 2006-02-23 2006-02-23
US77594506P 2006-02-23 2006-02-23
US77610506P 2006-02-23 2006-02-23
US77610606P 2006-02-23 2006-02-23
US77605706P 2006-02-23 2006-02-23
US77606406P 2006-02-23 2006-02-23
US77603306P 2006-02-23 2006-02-23
US77594906P 2006-02-23 2006-02-23
US83999406P 2006-08-24 2006-08-24
US83990306P 2006-08-24 2006-08-24

Publications (1)

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MA30267B1 true MA30267B1 (fr) 2009-03-02

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MA31218A MA30267B1 (fr) 2006-02-23 2008-09-08 Derives amides en tant que ligands de canal ionique et compositions pharmaceutiques et procedes d'utilisation de tels derives

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US (1) US20100004222A1 (fr)
JP (1) JP2009527575A (fr)
KR (1) KR20080098670A (fr)
CA (1) CA2641781A1 (fr)
CO (1) CO6170402A2 (fr)
EA (1) EA200870287A1 (fr)
GB (1) GB2452142A (fr)
IL (1) IL193346A0 (fr)
MA (1) MA30267B1 (fr)
NO (1) NO20083898L (fr)
TN (1) TNSN08328A1 (fr)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE102011014994A1 (de) * 2011-03-23 2012-09-27 Otto Bock Healthcare Gmbh Prothesenfußeinsatz und Prothesenfuß
JP6866583B2 (ja) * 2016-07-05 2021-04-28 Dic株式会社 液晶化合物

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR045979A1 (es) * 2003-04-28 2005-11-23 Astrazeneca Ab Amidas heterociclicas
WO2005046683A1 (fr) * 2003-10-07 2005-05-26 Renovis, Inc. Derives d'amide utilises comme ligands du canal ionique et compositions pharmaceutiques et methodes d'utilisation de ces derives
WO2006006740A1 (fr) * 2004-07-14 2006-01-19 Japan Tobacco Inc. Composé 3-aminobénamide et inhibiteur d'activité à récepteur vanilloïde 1 (vr1)

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KR20080098670A (ko) 2008-11-11
JP2009527575A (ja) 2009-07-30
GB0814753D0 (en) 2008-09-24
IL193346A0 (en) 2009-08-03
NO20083898L (no) 2008-10-30
TNSN08328A1 (en) 2009-12-29
EA200870287A1 (ru) 2009-02-27
CO6170402A2 (es) 2010-06-18
GB2452142A8 (en) 2009-03-18
CA2641781A1 (fr) 2007-09-07
US20100004222A1 (en) 2010-01-07
GB2452142A (en) 2009-02-25

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