NO20084659L - Ko-krystall av C-glucosidderivat og L-prolin - Google Patents

Ko-krystall av C-glucosidderivat og L-prolin

Info

Publication number
NO20084659L
NO20084659L NO20084659A NO20084659A NO20084659L NO 20084659 L NO20084659 L NO 20084659L NO 20084659 A NO20084659 A NO 20084659A NO 20084659 A NO20084659 A NO 20084659A NO 20084659 L NO20084659 L NO 20084659L
Authority
NO
Norway
Prior art keywords
crystal
proline
glucoside derivative
glucoside
derivative
Prior art date
Application number
NO20084659A
Other languages
English (en)
Norwegian (no)
Inventor
Kenichi Onda
Daisuke Sasuga
Ryota Shiraki
Masakazu Imamura
Keita Nakanishi
Masamichi Yuda
Original Assignee
Astellas Pharma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38563736&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20084659(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astellas Pharma Inc filed Critical Astellas Pharma Inc
Publication of NO20084659L publication Critical patent/NO20084659L/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D407/00Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00
    • C07D407/02Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings
    • C07D407/10Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings linked by a carbon chain containing aromatic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D207/00Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/16Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/38Heterocyclic compounds having sulfur as a ring hetero atom
    • A61K31/381Heterocyclic compounds having sulfur as a ring hetero atom having five-membered rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/48Drugs for disorders of the endocrine system of the pancreatic hormones
    • A61P5/50Drugs for disorders of the endocrine system of the pancreatic hormones for increasing or potentiating the activity of insulin
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/10Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Diabetes (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • Obesity (AREA)
  • Emergency Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicinal Preparation (AREA)
NO20084659A 2006-04-05 2008-11-04 Ko-krystall av C-glucosidderivat og L-prolin NO20084659L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2006103711 2006-04-05
PCT/JP2007/057597 WO2007114475A1 (ja) 2006-04-05 2007-04-04 C-グリコシド誘導体とl-プロリンとの共結晶

Publications (1)

Publication Number Publication Date
NO20084659L true NO20084659L (no) 2009-01-02

Family

ID=38563736

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20084659A NO20084659L (no) 2006-04-05 2008-11-04 Ko-krystall av C-glucosidderivat og L-prolin

Country Status (15)

Country Link
US (1) US8097592B2 (de)
EP (1) EP2009010A4 (de)
JP (1) JP5210154B2 (de)
KR (2) KR20120025001A (de)
CN (1) CN101443328B (de)
AU (1) AU2007232763B2 (de)
BR (1) BRPI0710581A2 (de)
CA (1) CA2649022C (de)
IL (1) IL194512A0 (de)
MX (1) MX2008012705A (de)
NO (1) NO20084659L (de)
RU (1) RU2408595C2 (de)
TW (1) TWI370818B (de)
WO (1) WO2007114475A1 (de)
ZA (1) ZA200809201B (de)

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WO2008075736A1 (ja) 2006-12-21 2008-06-26 Astellas Pharma Inc. C-グリコシド誘導体の製造方法及びその合成中間体
UA101004C2 (en) 2007-12-13 2013-02-25 Теракос, Инк. Derivatives of benzylphenylcyclohexane and use thereof
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JP2024525981A (ja) 2021-07-28 2024-07-12 ベーリンガー インゲルハイム フェトメディカ ゲーエムベーハー ヒト以外の哺乳動物における腎疾患の予防及び/又は治療のためのsglt-2阻害剤の使用
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TW202446389A (zh) 2023-04-24 2024-12-01 荷蘭商新阿姆斯特丹製藥公司 非晶形奧比特拉(obicetrapib)與sglt2抑制劑之組合
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Also Published As

Publication number Publication date
TW200811152A (en) 2008-03-01
KR101243039B1 (ko) 2013-03-20
CA2649022C (en) 2012-05-29
BRPI0710581A2 (pt) 2011-08-16
RU2008143362A (ru) 2010-05-10
EP2009010A4 (de) 2012-06-13
AU2007232763A1 (en) 2007-10-11
MX2008012705A (es) 2008-10-15
CN101443328B (zh) 2012-07-25
CN101443328A (zh) 2009-05-27
KR20090015912A (ko) 2009-02-12
TWI370818B (en) 2012-08-21
ZA200809201B (en) 2009-12-30
EP2009010A1 (de) 2008-12-31
JPWO2007114475A1 (ja) 2009-08-20
US20090143316A1 (en) 2009-06-04
KR20120025001A (ko) 2012-03-14
IL194512A0 (en) 2009-08-03
JP5210154B2 (ja) 2013-06-12
US8097592B2 (en) 2012-01-17
CA2649022A1 (en) 2007-10-11
WO2007114475A1 (ja) 2007-10-11
AU2007232763B2 (en) 2011-07-28
RU2408595C2 (ru) 2011-01-10

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