NO20092292L - Ny fremgangsmate for diastereoselektiv produksjon av et kiralt primaert amin pa et stereoid - Google Patents

Ny fremgangsmate for diastereoselektiv produksjon av et kiralt primaert amin pa et stereoid

Info

Publication number
NO20092292L
NO20092292L NO20092292A NO20092292A NO20092292L NO 20092292 L NO20092292 L NO 20092292L NO 20092292 A NO20092292 A NO 20092292A NO 20092292 A NO20092292 A NO 20092292A NO 20092292 L NO20092292 L NO 20092292L
Authority
NO
Norway
Prior art keywords
amine
stereoid
primed
chiral
new method
Prior art date
Application number
NO20092292A
Other languages
English (en)
Other versions
NO342093B1 (no
Inventor
Daniel Bernard
Joelle Bousquet-Frances
Gerard Cazenave
Gilles Oddon
Andre Simonnet
Original Assignee
Sanofi Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of NO20092292L publication Critical patent/NO20092292L/no
Publication of NO342093B1 publication Critical patent/NO342093B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0005—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring the nitrogen atom being directly linked to the cyclopenta(a)hydro phenanthrene skeleton
    • C07J41/0011—Unsubstituted amino radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0005—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring the nitrogen atom being directly linked to the cyclopenta(a)hydro phenanthrene skeleton
    • C07J41/0016—Oximes

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

Foreliggende oppfinnelse angår en diastereoselektiv fremgangsmåte for å oppnå et primært amin på et steroid, som innbefatter reduksjonen av et oksim med litium i ammoniakk ved en lav temperatur i en eter/alkoholblanding.
NO20092292A 2006-12-13 2009-06-15 Ny fremgangsmåte for diastereoselektiv fremstilling av et kiralt, primært amin på et steroid NO342093B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0610853A FR2910002B1 (fr) 2006-12-13 2006-12-13 Nouveau procede pour l'obtention diastereoselective d'une amine primaire chirale sur un steroide
PCT/FR2007/002035 WO2008090272A2 (fr) 2006-12-13 2007-12-11 Nouveau procede pour l'obtention diastereoselective d'une amine primaire chirale sur un steroïde

Publications (2)

Publication Number Publication Date
NO20092292L true NO20092292L (no) 2009-09-09
NO342093B1 NO342093B1 (no) 2018-03-19

Family

ID=38331497

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20092292A NO342093B1 (no) 2006-12-13 2009-06-15 Ny fremgangsmåte for diastereoselektiv fremstilling av et kiralt, primært amin på et steroid

Country Status (31)

Country Link
US (1) US20100069627A1 (no)
EP (1) EP2121724B1 (no)
JP (1) JP2010513252A (no)
KR (1) KR20090086593A (no)
CN (1) CN101558079B (no)
AR (1) AR064297A1 (no)
AT (1) ATE518877T1 (no)
AU (1) AU2007344926B2 (no)
BR (1) BRPI0720206A2 (no)
CA (1) CA2670655C (no)
CL (1) CL2007003621A1 (no)
CY (1) CY1113787T1 (no)
DK (1) DK2121724T3 (no)
EA (1) EA200970568A1 (no)
ES (1) ES2370537T3 (no)
FR (1) FR2910002B1 (no)
HR (1) HRP20110797T1 (no)
MA (1) MA30980B1 (no)
ME (1) ME00926B (no)
MX (1) MX2009006309A (no)
MY (1) MY145902A (no)
NO (1) NO342093B1 (no)
NZ (1) NZ577439A (no)
PL (1) PL2121724T3 (no)
PT (1) PT2121724E (no)
RS (1) RS51993B (no)
SI (1) SI2121724T1 (no)
TW (1) TWI405769B (no)
UY (1) UY30792A1 (no)
WO (1) WO2008090272A2 (no)
ZA (1) ZA200903832B (no)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9533451B2 (en) 2013-03-15 2017-01-03 3D Systems, Inc. Direct writing for additive manufacturing systems

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3035066A (en) * 1961-07-06 1962-05-15 Syntex Sa Quaternary ammonium salts of 3beta, 20beta-diamino-allopregnanes
BE717065A (no) * 1967-06-26 1968-12-24
US3960961A (en) * 1970-08-31 1976-06-01 The Upjohn Company 4'-Fluoro-4-{[4-(phenyl)cyclohexyl]amino}butyrophenones and the salts thereof
JPS4954358A (no) * 1972-09-30 1974-05-27
GB1581234A (en) * 1976-04-05 1980-12-10 Glaxo Operations Ltd 11a - amino - 3a - hydroxysteroids
US4197296A (en) * 1977-03-23 1980-04-08 Glaxo Group Limited Androstanes
AU6119980A (en) * 1979-08-09 1981-02-12 Glaxo Group Limited Benzoxocin derivatives
BR9407866A (pt) * 1993-10-21 1996-10-29 Merck & Co Inc Composto processos para inibiçao de 5 -redufase ou isoenzimas da mesma paratratamento de condiçoes de acne vulgar alopécia androgènica hirsutismo feminino hiperplasia prostática benigna prostatite e para o tratamento e/ou prevençao do cancer da próstata para interrupçao e reversao de alopécia androgènica e promoçao do crescimento de cabelo em um mamifero e para inibiçao de conversao biossintética da testosterona para di-hidro- testosterona em um mamifero e composiçao farmacèutica
US6350738B1 (en) * 1998-03-06 2002-02-26 Brigham Young University Steroid derived antibiotics

Also Published As

Publication number Publication date
CN101558079B (zh) 2013-09-11
KR20090086593A (ko) 2009-08-13
WO2008090272A3 (fr) 2008-11-27
PL2121724T3 (pl) 2011-12-30
WO2008090272A2 (fr) 2008-07-31
NZ577439A (en) 2012-02-24
ZA200903832B (en) 2010-08-25
EA200970568A1 (ru) 2009-10-30
BRPI0720206A2 (pt) 2013-12-31
US20100069627A1 (en) 2010-03-18
CL2007003621A1 (es) 2009-03-27
HK1138287A1 (en) 2010-08-20
RS51993B (sr) 2012-04-30
AU2007344926B2 (en) 2013-03-07
MY145902A (en) 2012-05-15
CA2670655C (fr) 2015-07-14
ME00926B (me) 2012-06-20
SI2121724T1 (sl) 2011-12-30
TWI405769B (zh) 2013-08-21
FR2910002A1 (fr) 2008-06-20
HRP20110797T1 (hr) 2011-11-30
PT2121724E (pt) 2011-11-21
ATE518877T1 (de) 2011-08-15
AU2007344926A1 (en) 2008-07-31
CN101558079A (zh) 2009-10-14
JP2010513252A (ja) 2010-04-30
TW200831526A (en) 2008-08-01
MX2009006309A (es) 2009-08-19
EP2121724A2 (fr) 2009-11-25
ES2370537T3 (es) 2011-12-19
MA30980B1 (fr) 2009-12-01
CA2670655A1 (fr) 2008-07-31
NO342093B1 (no) 2018-03-19
EP2121724B1 (fr) 2011-08-03
DK2121724T3 (da) 2011-11-21
UY30792A1 (es) 2008-07-31
ES2370537T8 (es) 2012-02-13
FR2910002B1 (fr) 2009-01-30
AR064297A1 (es) 2009-03-25
CY1113787T1 (el) 2016-07-27

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