NO308107B1 - Ikke-solvatert krystallinsk forbindelse, farmasøytisk formulering inneholdende denne samt anvendelse av forbindelsen for fremstilling av et farmasøytisk middel - Google Patents

Ikke-solvatert krystallinsk forbindelse, farmasøytisk formulering inneholdende denne samt anvendelse av forbindelsen for fremstilling av et farmasøytisk middel

Info

Publication number
NO308107B1
NO308107B1 NO953657A NO953657A NO308107B1 NO 308107 B1 NO308107 B1 NO 308107B1 NO 953657 A NO953657 A NO 953657A NO 953657 A NO953657 A NO 953657A NO 308107 B1 NO308107 B1 NO 308107B1
Authority
NO
Norway
Prior art keywords
compound
preparation
formulation containing
pharmaceutical
unsolvated crystalline
Prior art date
Application number
NO953657A
Other languages
English (en)
Norwegian (no)
Other versions
NO953657L (no
NO953657D0 (no
Inventor
Elizabeth Smith Labell
Wayne Douglas Luke
Iii John Mcneill Mcgill
Randal Scot Miller
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26976194&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO308107(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from US08/308,325 external-priority patent/US5629425A/en
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of NO953657D0 publication Critical patent/NO953657D0/no
Publication of NO953657L publication Critical patent/NO953657L/no
Publication of NO308107B1 publication Critical patent/NO308107B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/54—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • C07D333/56—Radicals substituted by oxygen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18—Feminine contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Endocrinology (AREA)
  • Diabetes (AREA)
  • Gynecology & Obstetrics (AREA)
  • Reproductive Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
NO953657A 1994-09-19 1995-09-15 Ikke-solvatert krystallinsk forbindelse, farmasøytisk formulering inneholdende denne samt anvendelse av forbindelsen for fremstilling av et farmasøytisk middel NO308107B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US08/308,325 US5629425A (en) 1994-09-19 1994-09-19 Haloalkyl hemisolvates of 6-hydroxy-2-(4-hydroxyphenyl)-3-[4-piperidinoethoxy)-benzoyl]benzo[b]thiophene
US42791495A 1995-04-26 1995-04-26

Publications (3)

Publication Number Publication Date
NO953657D0 NO953657D0 (no) 1995-09-15
NO953657L NO953657L (no) 1996-03-20
NO308107B1 true NO308107B1 (no) 2000-07-24

Family

ID=26976194

Family Applications (2)

Application Number Title Priority Date Filing Date
NO19953658A NO313996B1 (no) 1994-09-19 1995-09-15 Krystallinsk solvat av forbindelsen 6-hydroksy-2-(4- hydroksyfenyl)-3-[4-(2-piperidinoetoksy)benzoyl]benzo[b]tiofenhydroklorid, fremgangsmåtefor fremstilling av solvatet, og fremgangsmåte for fremstilling av en ikke-solvatisert utgaveav forbind
NO953657A NO308107B1 (no) 1994-09-19 1995-09-15 Ikke-solvatert krystallinsk forbindelse, farmasøytisk formulering inneholdende denne samt anvendelse av forbindelsen for fremstilling av et farmasøytisk middel

Family Applications Before (1)

Application Number Title Priority Date Filing Date
NO19953658A NO313996B1 (no) 1994-09-19 1995-09-15 Krystallinsk solvat av forbindelsen 6-hydroksy-2-(4- hydroksyfenyl)-3-[4-(2-piperidinoetoksy)benzoyl]benzo[b]tiofenhydroklorid, fremgangsmåtefor fremstilling av solvatet, og fremgangsmåte for fremstilling av en ikke-solvatisert utgaveav forbind

Country Status (50)

Country Link
US (4) US6399778B1 (de)
JP (2) JP2860071B2 (de)
KR (2) KR100381346B1 (de)
CN (2) CN1075069C (de)
AP (1) AP754A (de)
AT (2) AT407988B (de)
AU (3) AU691955B2 (de)
BE (2) BE1009626A3 (de)
BG (1) BG62793B1 (de)
BR (2) BR9504059A (de)
CA (2) CA2158400C (de)
CH (3) CH691125A5 (de)
CO (2) CO4410191A1 (de)
CZ (2) CZ292007B6 (de)
DE (3) DE19549755B4 (de)
DK (4) DK175903B1 (de)
EE (1) EE03386B1 (de)
EG (1) EG23763A (de)
ES (2) ES2109882B1 (de)
FI (2) FI121424B (de)
FR (2) FR2732020B1 (de)
GB (2) GB2293602B (de)
GE (1) GEP19991821B (de)
GR (2) GR1002697B (de)
HR (2) HRP950483B1 (de)
HU (2) HU225417B1 (de)
IE (2) IE950722A1 (de)
IL (3) IL115315A (de)
IS (1) IS1788B (de)
IT (2) IT1277601B1 (de)
LU (2) LU88660A1 (de)
LV (2) LV11177B (de)
MY (1) MY116371A (de)
NL (2) NL1001194C2 (de)
NO (2) NO313996B1 (de)
NZ (2) NZ280028A (de)
OA (1) OA10406A (de)
PE (2) PE14796A1 (de)
PL (2) PL187686B1 (de)
PT (2) PT101770B (de)
RO (2) RO115260B1 (de)
RS (2) RS49513B (de)
SE (2) SE520721C2 (de)
SI (2) SI9500293A (de)
SK (1) SK283502B6 (de)
TR (1) TR199501136A2 (de)
TW (1) TW412534B (de)
UA (2) UA44240C2 (de)
UY (1) UY24040A1 (de)
WO (1) WO1996009045A1 (de)

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Also Published As

Publication number Publication date
IL115314A (en) 2000-02-29
DK2797A (da) 1997-01-09
YU61495A (sh) 1998-05-15
FI954402A0 (fi) 1995-09-18
PL187686B1 (pl) 2004-09-30
JP2860071B2 (ja) 1999-02-24
GB2293382B (en) 1998-08-19
DE19534744A1 (de) 1996-03-21
DE19534745A1 (de) 1996-04-04
CZ292007B6 (cs) 2003-07-16
PT101771A (pt) 1996-04-30
CZ290343B6 (cs) 2002-07-17
OA10406A (en) 2001-12-05
US6399778B1 (en) 2002-06-04
ES2129293A1 (es) 1999-06-01
HU225417B1 (en) 2006-11-28
RS49513B (sr) 2006-10-27
NZ280027A (en) 1997-05-26
ES2109882A1 (es) 1998-01-16
NL1001194A1 (nl) 1996-03-19
FI954403A7 (fi) 1996-03-20
AU3173095A (en) 1996-04-04
IL115315A0 (en) 1995-12-31
DK175897B1 (da) 2005-05-30
PT101771B (pt) 1997-04-30
PE32796A1 (es) 1996-08-07
ATA154295A (de) 2000-12-15
BE1009626A3 (fr) 1997-06-03
AT407988B (de) 2001-07-25
FR2732020A1 (fr) 1996-09-27
SE509265C2 (sv) 1998-12-21
EE03386B1 (et) 2001-04-16
CZ240395A3 (en) 1996-04-17
WO1996009045A1 (en) 1996-03-28
GB2293602A (en) 1996-04-03
CN1127253A (zh) 1996-07-24
SE9503214D0 (sv) 1995-09-15
HU9502721D0 (en) 1995-11-28
PT101770A (pt) 1996-04-30
CA2158399A1 (en) 1996-03-20
ITMI951936A1 (it) 1997-03-15
IS4446A (is) 1997-03-18
ITMI951935A1 (it) 1997-03-15
GB9519032D0 (en) 1995-11-15
KR100381346B1 (ko) 2004-04-13
GB9519028D0 (en) 1995-11-15
UA42716C2 (uk) 2001-11-15
SE520721C2 (sv) 2003-08-12
DE19534745B4 (de) 2004-06-09
FI112226B (fi) 2003-11-14
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BG62793B1 (bg) 2000-08-31
HRP950482B1 (en) 2007-04-30
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AU3173195A (en) 1996-04-04
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LV11177B (en) 1996-08-20
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