NO314499B1 - Fremgangsmåte for å oppnå enantiomerer av cis-olirtin - Google Patents

Fremgangsmåte for å oppnå enantiomerer av cis-olirtin Download PDF

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Publication number
NO314499B1
NO314499B1 NO20000560A NO20000560A NO314499B1 NO 314499 B1 NO314499 B1 NO 314499B1 NO 20000560 A NO20000560 A NO 20000560A NO 20000560 A NO20000560 A NO 20000560A NO 314499 B1 NO314499 B1 NO 314499B1
Authority
NO
Norway
Prior art keywords
pyrazol
ketone
methyl
phenyl
chiral
Prior art date
Application number
NO20000560A
Other languages
English (en)
Norwegian (no)
Other versions
NO20000560D0 (no
NO20000560L (no
Inventor
Antoni Torrens-Jover
Jordi Frigola-Constansa
Original Assignee
Esteve Labor Dr
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Esteve Labor Dr filed Critical Esteve Labor Dr
Publication of NO20000560D0 publication Critical patent/NO20000560D0/no
Publication of NO20000560L publication Critical patent/NO20000560L/no
Publication of NO314499B1 publication Critical patent/NO314499B1/no

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
NO20000560A 1997-08-04 2000-02-03 Fremgangsmåte for å oppnå enantiomerer av cis-olirtin NO314499B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
ES009701728A ES2130083B1 (es) 1997-08-04 1997-08-04 Procedimiento para la obtencion de los enantiomeros de cizolirtina.
PCT/ES1998/000223 WO1999007684A1 (es) 1997-08-04 1998-07-31 Procedimiento para la obtencion de los enantiomeros de cizolirtina

Publications (3)

Publication Number Publication Date
NO20000560D0 NO20000560D0 (no) 2000-02-03
NO20000560L NO20000560L (no) 2000-03-29
NO314499B1 true NO314499B1 (no) 2003-03-31

Family

ID=8300306

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20000560A NO314499B1 (no) 1997-08-04 2000-02-03 Fremgangsmåte for å oppnå enantiomerer av cis-olirtin

Country Status (12)

Country Link
US (1) US6118009A (de)
EP (1) EP1029852B1 (de)
JP (1) JP2001512718A (de)
AT (1) ATE227272T1 (de)
AU (1) AU8442698A (de)
CA (1) CA2299447C (de)
DE (1) DE69809282T2 (de)
DK (1) DK1029852T3 (de)
ES (2) ES2130083B1 (de)
NO (1) NO314499B1 (de)
PT (1) PT1029852E (de)
WO (1) WO1999007684A1 (de)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20040142929A1 (en) * 2001-07-06 2004-07-22 Ramon Merce-Vidal Derivatives of aryl (or heteroaryl) azolylcarbinoles for the treatment of urinary incontinence
TW200533657A (en) * 2004-02-17 2005-10-16 Esteve Labor Dr Substituted pyrazoline compounds, their preparation and use as medicaments
JP2007531785A (ja) * 2004-04-05 2007-11-08 ラボラトリオス・デル・デエレ・エステベ・エセ・ア 活性物質組合せ物
ES2244326B1 (es) * 2004-04-05 2007-02-16 Laboratorios Del Dr. Esteve, S.A. Combinacion de substancias activas.
EP1584335A3 (de) * 2004-04-05 2006-02-22 Laboratorios Del Dr. Esteve, S.A. Zusammensetzung aus Aktiva mit einer Carbinolverbindung und einem Opioid
US20060040924A1 (en) * 2004-06-22 2006-02-23 Laboratorios Dr. Esteve S.A. Derivatives of aryl (or heteroaryl) azolylcarbinols for the treatment of renal colic
EP1671953A1 (de) * 2004-12-17 2006-06-21 Laboratorios Del Dr. Esteve, S.A. Verfahren zur Herstellung von Cizolirtine und dessen Enantiomeren
WO2006063861A1 (en) * 2004-12-17 2006-06-22 Laboratorios Del Dr. Esteve, S.A. Process for obtaining cizolirtine and its enantiomers
EP1671968A1 (de) * 2004-12-17 2006-06-21 Laboratorios Del Dr. Esteve, S.A. Verfahren zur Herstellung von Enantiomeren von Thienylazolylalkoxyethanamines
US7897589B2 (en) * 2005-07-15 2011-03-01 Laboratorios Del Dr. Esteve, S.A. Substituted pyrazoline compounds, their preparation and use as medicaments
EP1743892A1 (de) * 2005-07-15 2007-01-17 Laboratorios del Dr. Esteve S.A. Substituierte Pyrazolin Verbindungen, deren Herstellung und Verwendung als Medikament
EP1743890A1 (de) * 2005-07-15 2007-01-17 Laboratorios Del Dr. Esteve, S.A. 4,5-Dihydro-1H-Pyrazol-Derivative, Verfahren zur Herstellung und ihre Verwendung als Medikamente.
EP1757587A1 (de) * 2005-07-15 2007-02-28 Laboratorios Del Dr. Esteve, S.A. Substituierte Pyrazolinderivate, ihre Herstellung und Verwendung als Arzneimittel
EP1820502A1 (de) 2006-02-10 2007-08-22 Laboratorios Del Dr. Esteve, S.A. Wirkstoffzusammensetzungen enthaltend Azolycarbinolderivate
EP2151234A1 (de) * 2008-07-28 2010-02-10 Laboratorios Del. Dr. Esteve, S.A. Pharmazeutische Formulierung mit einer CB1-Rezeptorverbindung in einer festen Lösung und/oder festen Dispersion
US20100291151A1 (en) * 2009-04-21 2010-11-18 Auspex Pharmaceuticals, Inc. 1-methylpyrazole modulators of substance p, calcitonin gene-related peptide, adrenergic receptor, and/or 5-ht receptor
DE102010056283A1 (de) 2010-12-24 2012-06-28 Volkswagen Ag Wärmeübertragungssystem
CN108558695A (zh) * 2018-05-15 2018-09-21 浙江华贝药业有限责任公司 2，2，2-三氟-n-[(1s，4s)-4-羟基四氢萘-1-基]-乙酰胺制备方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4943635A (en) * 1987-08-27 1990-07-24 President & Fellows Of Harvard College Enantioselective reduction of ketones
CA2134096C (en) * 1992-05-14 1997-11-25 George J. Quallich Enantioselective oxazaborolidine catalysts
US5442118A (en) * 1994-04-22 1995-08-15 Sepracor, Inc. Asymmetric synthesis of (R)- and (S)-arylethanolamines from iminoketones

Also Published As

Publication number Publication date
NO20000560D0 (no) 2000-02-03
EP1029852A1 (de) 2000-08-23
DE69809282T2 (de) 2003-09-11
WO1999007684A1 (es) 1999-02-18
DE69809282D1 (de) 2002-12-12
AU8442698A (en) 1999-03-01
NO20000560L (no) 2000-03-29
ES2187044T3 (es) 2003-05-16
EP1029852B1 (de) 2002-11-06
US6118009A (en) 2000-09-12
CA2299447C (en) 2007-05-29
DK1029852T3 (da) 2003-02-24
ES2130083B1 (es) 2000-01-16
ES2130083A1 (es) 1999-06-16
JP2001512718A (ja) 2001-08-28
PT1029852E (pt) 2003-03-31
CA2299447A1 (en) 1999-02-18
ATE227272T1 (de) 2002-11-15

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