NO320022B1 - Kontrollert frigjorende farmasoytisk preparat med tilidinmesylat som virkestoff - Google Patents

Kontrollert frigjorende farmasoytisk preparat med tilidinmesylat som virkestoff Download PDF

Info

Publication number: NO320022B1
Authority: NO; Norway
Prior art keywords: tilidine; controlled release; pharmaceutical preparation; oral administration; active ingredient
Prior art date: 1998-12-23

Application number

NO20013060A

Other languages

English (en)

Norwegian (no)

Other versions

NO20013060L (no

NO20013060D0 (no

Inventor

Richard Hirsch

Martin Wesseling

Thomas Struengmann

Original Assignee

Hexal Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1998-12-23

Filing date

2001-06-20

Publication date

2005-10-10

2001-06-20 Application filed by Hexal Ag filed Critical Hexal Ag

2001-06-20 Publication of NO20013060L publication Critical patent/NO20013060L/no

2001-06-20 Publication of NO20013060D0 publication Critical patent/NO20013060D0/no

2005-10-10 Publication of NO320022B1 publication Critical patent/NO320022B1/no

Links

229960001402 tilidine Drugs 0.000 title claims abstract description 65
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AFVFQIVMOAPDHO-UHFFFAOYSA-N Methanesulfonic acid Chemical compound CS(O)(=O)=O AFVFQIVMOAPDHO-UHFFFAOYSA-N 0.000 title claims abstract description 48
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Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
- A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
- A61K31/216—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acids having aromatic rings, e.g. benactizyne, clofibrate
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Epidemiology (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Emergency Medicine (AREA)
Pain & Pain Management (AREA)
Organic Chemistry (AREA)
Molecular Biology (AREA)
Biophysics (AREA)
General Chemical & Material Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Neurosurgery (AREA)
Neurology (AREA)
Biomedical Technology (AREA)
Engineering & Computer Science (AREA)
Rheumatology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicinal Preparation (AREA)
Steroid Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

NO20013060A 1998-12-23 2001-06-20 Kontrollert frigjorende farmasoytisk preparat med tilidinmesylat som virkestoff NO320022B1 (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
DE19859636A DE19859636A1 (de)	1998-12-23	1998-12-23	Kontrolliert freisetzende pharmazeutische Zusammensetzung mit Tilidinmesylat als Wirkstoff
PCT/EP1999/010381 WO2000038656A1 (de)	1998-12-23	1999-12-23	Kontrolliert freisetzende pharmazeutische zusammensetzung mit tilidinmesylat als wirkstoff

Publications (3)

Publication Number	Publication Date
NO20013060L NO20013060L (no)	2001-06-20
NO20013060D0 NO20013060D0 (no)	2001-06-20
NO320022B1 true NO320022B1 (no)	2005-10-10

Family

ID=7892368

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO20013060A NO320022B1 (no)	1998-12-23	2001-06-20	Kontrollert frigjorende farmasoytisk preparat med tilidinmesylat som virkestoff

Country Status (21)

Country	Link
US (1)	US6579536B1 (cs)
EP (1)	EP1140031B1 (cs)
JP (1)	JP2002533381A (cs)
AT (1)	ATE252377T1 (cs)
AU (1)	AU770293B2 (cs)
BR (1)	BR9916575A (cs)
CA (1)	CA2355891A1 (cs)
CZ (1)	CZ301628B6 (cs)
DE (2)	DE19859636A1 (cs)
DK (1)	DK1140031T3 (cs)
ES (1)	ES2207334T3 (cs)
HU (1)	HUP0104647A3 (cs)
MX (1)	MXPA01006493A (cs)
NO (1)	NO320022B1 (cs)
NZ (1)	NZ512079A (cs)
PL (1)	PL199024B1 (cs)
PT (1)	PT1140031E (cs)
SK (1)	SK284901B6 (cs)
TR (1)	TR200101864T2 (cs)
WO (1)	WO2000038656A1 (cs)
ZA (1)	ZA200105040B (cs)

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TR200001942T2 (tr)	1997-12-22	2000-11-21	Euro-Celtique, S.A.	Opioid agonist/antagonist kombinasyonlar
US6375957B1 (en)	1997-12-22	2002-04-23	Euro-Celtique, S.A.	Opioid agonist/opioid antagonist/acetaminophen combinations
CA2400578C (en) *	2000-02-08	2007-01-02	Euro-Celtique, S.A.	Controlled-release compositions containing opioid agonist and antagonist
SI2283842T1 (sl) *	2000-02-08	2015-07-31	Euro-Celtique S.A.	Oralne formulacije opioidnih agonistov, varne pred zlorabo
EP1387673B1 (en)	2001-05-11	2010-12-29	Endo Pharmaceuticals Inc.	Abuse-resistant controlled-release opioid dosage form
LT2425821T (lt)	2002-04-05	2017-07-25	Euro-Celtique S.A.	Farmacinis preparatas, turintis oksikodono ir naloksono
JP4563642B2 (ja) *	2002-05-31	2010-10-13	ワトソンラボラトリーズ、インコーポレイテッド	医薬製剤
DE10233108A1 (de) *	2002-07-20	2004-01-29	Krewel Meuselbach Gmbh	Retardiertes Schmerzmittel enthaltend Tilidin und ein Lichtschutzmittel
DE10250081A1 (de) *	2002-10-25	2004-05-13	Boehringer Ingelheim Vetmedica Gmbh	Wasserlösliche Meloxicam Granulate
EP1479381A1 (en) *	2003-05-19	2004-11-24	Euro-Celtique S.A.	Pharmaceutical dosage form comprising a solid solution
EP1604666A1 (en)	2004-06-08	2005-12-14	Euro-Celtique S.A.	Opioids for the treatment of the Chronic Obstructive Pulmonary Disease (COPD)
WO2006009403A1 (en) *	2004-07-22	2006-01-26	Amorepacific Corporation	Sustained-release preparations containing topiramate and the producing method thereof
EP1702558A1 (en)	2005-02-28	2006-09-20	Euro-Celtique S.A.	Method and device for the assessment of bowel function
US20070048373A1 (en) *	2005-08-30	2007-03-01	Cima Labs Inc.	Dried milled granulate and methods
EP2168945A1 (en) *	2008-09-26	2010-03-31	Hexal Ag	Crystalline forms of Tilidine Mesylate
WO2010099508A1 (en)	2009-02-26	2010-09-02	Theraquest Biosciences, Inc.	Extended release oral pharmaceutical compositions of 3-hydroxy-n-methylmorphinan and method of use
PL2405915T3 (pl)	2009-03-10	2019-05-31	Euro Celtique Sa	Kompozycje farmaceutyczne o natychmiastowym uwalnianiu zawierające oksykodon i nalokson
KR20160034352A (ko)	2013-07-23	2016-03-29	유로-셀티큐 에스.에이.	장내 세균총이상을 초래하고/하거나 장내 박테리아 전위에 대한 위험을 증가시키는 질환과 통증으로 인해 고통받고 있는 환자에서 통증을 치료하는데 사용하기 위한 옥시코돈과 날록손의 조합물
BR112017005574A2 (pt)	2014-09-19	2017-12-12	Procter & Gamble	formas de dosagem de liberação pulsada de fenilefrina
US10278930B2 (en)	2017-03-16	2019-05-07	The Procter & Gamble Company	Method for relieving sinus congestion

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* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
LU71847A1 (cs) *	1975-02-14	1977-01-05
KR100310041B1 (ko) *	1992-10-26	2002-04-24	괴데케악티엔게젤샤프트	틸리딘이수소오르토포스페이트,그제조방법및이를함유한의약제제
US5965161A (en) *	1994-11-04	1999-10-12	Euro-Celtique, S.A.	Extruded multi-particulates
DE19710008A1 (de)	1997-03-12	1998-09-17	Basf Ag	Feste, mindestens zweiphasige Zubereitungsformen eines Opioid-Analgeticums mit verzögerter Freisetzung
DE19981795T1 (de) *	1998-04-28	2001-05-10	Russinsky Ltd	Tilidinmesylat, Verfahren zu dessen Herstellung und pharmazeutische Zusammensetzung davon

1998
- 1998-12-23 DE DE19859636A patent/DE19859636A1/de not_active Ceased
1999
- 1999-12-23 BR BR9916575-9A patent/BR9916575A/pt not_active IP Right Cessation
- 1999-12-23 AU AU22862/00A patent/AU770293B2/en not_active Ceased
- 1999-12-23 MX MXPA01006493A patent/MXPA01006493A/es not_active Application Discontinuation
- 1999-12-23 ES ES99967009T patent/ES2207334T3/es not_active Expired - Lifetime
- 1999-12-23 PT PT99967009T patent/PT1140031E/pt unknown
- 1999-12-23 PL PL348419A patent/PL199024B1/pl not_active IP Right Cessation
- 1999-12-23 AT AT99967009T patent/ATE252377T1/de active
- 1999-12-23 DE DE59907481T patent/DE59907481D1/de not_active Expired - Lifetime
- 1999-12-23 EP EP99967009A patent/EP1140031B1/de not_active Expired - Lifetime
- 1999-12-23 HU HU0104647A patent/HUP0104647A3/hu unknown
- 1999-12-23 US US09/869,033 patent/US6579536B1/en not_active Expired - Fee Related
- 1999-12-23 JP JP2000590610A patent/JP2002533381A/ja active Pending
- 1999-12-23 DK DK99967009T patent/DK1140031T3/da active
- 1999-12-23 SK SK892-2001A patent/SK284901B6/sk unknown
- 1999-12-23 CZ CZ20012167A patent/CZ301628B6/cs not_active IP Right Cessation
- 1999-12-23 WO PCT/EP1999/010381 patent/WO2000038656A1/de not_active Ceased
- 1999-12-23 NZ NZ512079A patent/NZ512079A/en unknown
- 1999-12-23 TR TR2001/01864T patent/TR200101864T2/xx unknown
- 1999-12-23 CA CA002355891A patent/CA2355891A1/en not_active Abandoned
2001
- 2001-06-20 ZA ZA200105040A patent/ZA200105040B/en unknown
- 2001-06-20 NO NO20013060A patent/NO320022B1/no not_active IP Right Cessation

Also Published As

Publication number	Publication date
CZ301628B6 (cs)	2010-05-05
ATE252377T1 (de)	2003-11-15
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CN103002882B (zh)	2016-03-02	不含活性剂之颗粒及包含其之片剂的制备
US10179130B2 (en)	2019-01-15	Controlled release hydrocodone formulations
HK1039273B (en)	2004-03-12	Sustained-release pharmaceutical preparation containing tilidine mesylate as active ingredient
KR20210039876A (ko)	2021-04-12	옥시코돈 및 날록손을 포함하는 서방성 제제