NO331012B1 - N-sulfonyl-4-metylenamino-3-hydroksy-2-pyridoner som antimikrobielle midler - Google Patents

N-sulfonyl-4-metylenamino-3-hydroksy-2-pyridoner som antimikrobielle midler

Info

Publication number
NO331012B1
NO331012B1 NO20052788A NO20052788A NO331012B1 NO 331012 B1 NO331012 B1 NO 331012B1 NO 20052788 A NO20052788 A NO 20052788A NO 20052788 A NO20052788 A NO 20052788A NO 331012 B1 NO331012 B1 NO 331012B1
Authority
NO
Norway
Prior art keywords
methyleneamino
pyridones
sulfonyl
hydroxy
antimicrobial agents
Prior art date
Application number
NO20052788A
Other languages
English (en)
Norwegian (no)
Other versions
NO20052788L (no
Inventor
Rodney Dean Bush
Namal Chithranga Warshakoon
Original Assignee
Warner Chilcott Co Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Warner Chilcott Co Llc filed Critical Warner Chilcott Co Llc
Publication of NO20052788L publication Critical patent/NO20052788L/no
Publication of NO331012B1 publication Critical patent/NO331012B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/89—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members with hetero atoms directly attached to the ring nitrogen atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
NO20052788A 2002-11-09 2005-06-09 N-sulfonyl-4-metylenamino-3-hydroksy-2-pyridoner som antimikrobielle midler NO331012B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US42507102P 2002-11-09 2002-11-09
PCT/US2003/035623 WO2004043928A2 (fr) 2002-11-09 2003-11-07 N-sulfonyl-4-methylene-amino-3-hydroxy-2-pyridones

Publications (2)

Publication Number Publication Date
NO20052788L NO20052788L (no) 2005-06-09
NO331012B1 true NO331012B1 (no) 2011-09-05

Family

ID=32312927

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20052788A NO331012B1 (no) 2002-11-09 2005-06-09 N-sulfonyl-4-metylenamino-3-hydroksy-2-pyridoner som antimikrobielle midler

Country Status (25)

Country Link
US (3) US6946479B2 (fr)
EP (1) EP1558580B1 (fr)
JP (1) JP4327730B2 (fr)
KR (2) KR20050055793A (fr)
CN (1) CN1708482A (fr)
AT (1) ATE372986T1 (fr)
AU (1) AU2003296045B2 (fr)
BR (1) BR0316086A (fr)
CA (1) CA2502416C (fr)
CO (1) CO5570702A2 (fr)
CY (1) CY1106957T1 (fr)
DE (1) DE60316339T2 (fr)
DK (1) DK1558580T3 (fr)
ES (1) ES2293059T3 (fr)
HR (1) HRP20050517B1 (fr)
IL (1) IL168118A (fr)
MA (1) MA27549A1 (fr)
MX (1) MXPA05004897A (fr)
NO (1) NO331012B1 (fr)
NZ (1) NZ539385A (fr)
PL (1) PL377176A1 (fr)
PT (1) PT1558580E (fr)
RU (1) RU2321584C2 (fr)
WO (1) WO2004043928A2 (fr)
ZA (1) ZA200503682B (fr)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6946479B2 (en) * 2002-11-09 2005-09-20 The Procter & Gamble Company N-sulfonyl-4-methyleneamino-3-hydroxy-2-pyridones
US6930117B2 (en) * 2002-11-09 2005-08-16 The Procter & Gamble Company N-alkyl-4-methyleneamino-3-hydroxy-2-pyridones
US20070275944A1 (en) * 2006-04-05 2007-11-29 The Board Of Trustees Operating Michigan State University Antioxidants and methods of their use
US7622593B2 (en) 2006-06-27 2009-11-24 The Procter & Gamble Company Human protein tyrosine phosphatase inhibitors and methods of use
ES2726946T3 (es) 2009-07-06 2019-10-10 Aerpio Therapeutics Inc Derivados de benzosulfonamida, composiciones de los mismos y su uso en la prevención de la metástasis de las células cancerosas
RS54010B1 (sr) * 2009-11-06 2015-10-30 Aerpio Therapeutics Inc. Inhibitori prolil hidroksilaze
JP6118808B2 (ja) 2011-10-31 2017-04-19 ザ メソジスト ホスピタル リサーチ インスティテュート ヒトグリオームを治療するためのｍａｏ標的化／探索部分を含む化合物
CN103360308A (zh) * 2012-03-28 2013-10-23 孙伟新 1,4-二羟基-6-甲基-2-吡啶酮类化合物及其制备方法和用途
US20150050277A1 (en) 2013-03-15 2015-02-19 Aerpio Therapeutics Inc. Compositions and methods for treating ocular diseases
AU2014233363B2 (en) 2013-03-15 2017-06-29 EyePoint, Inc. Compositions, formulations and methods for treating ocular diseases
US9388135B2 (en) 2014-02-19 2016-07-12 Aerpio Therapeutics, Inc. Process for preparing N-benzyl-3-hydroxy-4-substituted-pyridin-2-(1H)-ones
EP3116503A4 (fr) 2014-03-14 2017-08-23 Aerpio Therapeutics, Inc. Inhibiteurs de hptp-bêta
WO2016022813A1 (fr) 2014-08-07 2016-02-11 Aerpio Therapeutics, Inc. Combinaison d'immunothérapies avec des activateurs de tie -2

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3853900A (en) 1973-09-14 1974-12-10 Searle & Co 4-benzyloxy-2 (1h)-pyridones
US5358949A (en) 1986-03-05 1994-10-25 Otsuka Pharmaceutical Co., Ltd. Carbostyril derivatives and salts thereof and anti-arrhythmic agents containing the carbostyril derivatives
DE4316077A1 (de) 1993-05-13 1994-11-17 Bayer Ag Substituierte Mono- und Bihydridylmethylpyridone
US5817825A (en) * 1994-11-02 1998-10-06 Hoechst Aktiengesellschaft Process for the preparation of 1-hydroxy-2-pyridones
US5789426A (en) 1995-01-20 1998-08-04 Cornell Research Foundation, Inc. Method for the treatment of fibroproliferative disorders by application of inhibitors of protein hydroxylation
US6046219A (en) 1995-01-20 2000-04-04 Cornell Research Foundation, Inc. Method for the treatment of conditions mediated by collagen formation together with cell proliferation by application of inhibitors of protein hydroxylation
US5849587A (en) 1995-06-09 1998-12-15 Cornell Research Foundation, Inc. Method of inhibiting viral replication in eukaryotic cells and of inducing apoptosis of virally-infected cells
US6946479B2 (en) * 2002-11-09 2005-09-20 The Procter & Gamble Company N-sulfonyl-4-methyleneamino-3-hydroxy-2-pyridones

Also Published As

Publication number Publication date
RU2321584C2 (ru) 2008-04-10
AU2003296045B2 (en) 2008-04-03
IL168118A (en) 2011-07-31
CN1708482A (zh) 2005-12-14
WO2004043928A8 (fr) 2005-05-06
WO2004043928A3 (fr) 2004-07-01
US20050256126A1 (en) 2005-11-17
MA27549A1 (fr) 2005-10-03
PL377176A1 (pl) 2006-01-23
US20070238722A1 (en) 2007-10-11
JP4327730B2 (ja) 2009-09-09
EP1558580B1 (fr) 2007-09-12
WO2004043928A2 (fr) 2004-05-27
MXPA05004897A (es) 2005-11-17
CY1106957T1 (el) 2012-09-26
RU2005114490A (ru) 2006-01-20
ZA200503682B (en) 2006-11-29
DE60316339D1 (de) 2007-10-25
ES2293059T3 (es) 2008-03-16
PT1558580E (pt) 2007-12-06
DE60316339T2 (de) 2008-06-05
AU2003296045A1 (en) 2004-06-03
KR20070030334A (ko) 2007-03-15
EP1558580A2 (fr) 2005-08-03
US20040097559A1 (en) 2004-05-20
KR100894237B1 (ko) 2009-04-20
BR0316086A (pt) 2005-09-27
HRP20050517B1 (hr) 2014-03-14
HRP20050517A2 (en) 2005-12-31
NO20052788L (no) 2005-06-09
JP2006513164A (ja) 2006-04-20
DK1558580T3 (da) 2008-01-14
CO5570702A2 (es) 2005-10-31
CA2502416A1 (fr) 2004-05-27
US7247632B2 (en) 2007-07-24
ATE372986T1 (de) 2007-09-15
CA2502416C (fr) 2010-07-20
US6946479B2 (en) 2005-09-20
NZ539385A (en) 2008-02-29
KR20050055793A (ko) 2005-06-13

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