NO791592L - Xanthen- og tioxanthenderivater og fremgangsmaate ved fremstilling av disse - Google Patents

Xanthen- og tioxanthenderivater og fremgangsmaate ved fremstilling av disse

Info

Publication number
NO791592L
NO791592L NO791592A NO791592A NO791592L NO 791592 L NO791592 L NO 791592L NO 791592 A NO791592 A NO 791592A NO 791592 A NO791592 A NO 791592A NO 791592 L NO791592 L NO 791592L
Authority
NO
Norway
Prior art keywords
group
groups
effects
formula
carbon atoms
Prior art date
Application number
NO791592A
Other languages
English (en)
Other versions
NO150837B (no
NO150837C (no
Inventor
Niels Lassen
Klaus Peter Bofegesoe
Peter Bregnedal Hansen
Joern Lasse Martin Buus
Allan Johan Bigler
Original Assignee
Kefalas As
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Kefalas As filed Critical Kefalas As
Publication of NO791592L publication Critical patent/NO791592L/no
Publication of NO150837B publication Critical patent/NO150837B/no
Publication of NO150837C publication Critical patent/NO150837C/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D335/00—Heterocyclic compounds containing six-membered rings having one sulfur atom as the only ring hetero atom
    • C07D335/04—Heterocyclic compounds containing six-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D335/10—Dibenzothiopyrans; Hydrogenated dibenzothiopyrans
    • C07D335/12—Thioxanthenes
    • C07D335/14—Thioxanthenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 9
    • C07D335/18—Nitrogen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C309/00—Sulfonic acids; Halides, esters, or anhydrides thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Psychiatry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Neurosurgery (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Saccharide Compounds (AREA)
  • Polymerisation Methods In General (AREA)
  • Inks, Pencil-Leads, Or Crayons (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
NO791592A 1978-05-12 1979-05-11 Analogifremgangsmaate ved fremstilling av terapeutisk aktive xanten- og tioxantenderivater NO150837C (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB1931078 1978-05-12

Publications (3)

Publication Number Publication Date
NO791592L true NO791592L (no) 1979-11-13
NO150837B NO150837B (no) 1984-09-17
NO150837C NO150837C (no) 1985-01-09

Family

ID=10127259

Family Applications (1)

Application Number Title Priority Date Filing Date
NO791592A NO150837C (no) 1978-05-12 1979-05-11 Analogifremgangsmaate ved fremstilling av terapeutisk aktive xanten- og tioxantenderivater

Country Status (14)

Country Link
US (3) US4285956A (no)
EP (1) EP0005607B1 (no)
JP (1) JPS54154772A (no)
AT (1) ATE5141T1 (no)
AU (1) AU522926B2 (no)
CA (1) CA1127648A (no)
DE (1) DE2966344D1 (no)
DK (1) DK190179A (no)
ES (1) ES480468A1 (no)
FI (1) FI791503A7 (no)
IE (1) IE48261B1 (no)
NO (1) NO150837C (no)
NZ (1) NZ190373A (no)
ZA (1) ZA792250B (no)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4356184A (en) * 1980-06-04 1982-10-26 G. D. Searle & Co. Anti-allergic or antihypertensive 1-piperidinylmethyl benzenamines
US4501749A (en) * 1983-10-31 1985-02-26 Merck & Co., Inc. Peripherally selective dopamine antagonists in the treatment of ocular hypertension
US4777177A (en) * 1984-10-19 1988-10-11 Ciba-Geigy Corporation Pesticidal thioxanthen-9-ylidenepiperidines
US5250681A (en) * 1988-06-02 1993-10-05 Ajinomoto Co., Inc. Piperidine derivatives and hypotensives containing the same
US5393890A (en) * 1988-06-02 1995-02-28 Ajinomoto Co., Inc. Piperidine derivatives and hypotensives containing the same
CA2004211A1 (en) * 1988-11-30 1990-05-31 Masataka Syoji Piperidine derivatives and hyportensives containing the same
US7060711B2 (en) * 2001-10-25 2006-06-13 Biofrontera Bioscience Gmbh Derivatives of 4-(thio- or selenoxanthene-9-ylidene)-piperidine or acridine and its use as a selective 5-HT2B receptor antagonist
EP1306376A1 (en) * 2001-10-25 2003-05-02 Biofrontera Pharmaceuticals AG Derivatives of 4-(thio- or selenoxanthene-9-ylidene)-piperidine or acridine and its use as a selective 5-HT2B receptor antagonist
US7589103B2 (en) * 2003-06-27 2009-09-15 Janssen Pharmaceutica N.V. Tricyclic-bridged piperidinylidene derivatives as 8-opioid modulators
EP1910353A1 (en) * 2004-08-05 2008-04-16 Janssen Pharmaceutica N.V. Tricyclic delta- opioid modulators
JP2008525481A (ja) * 2004-12-22 2008-07-17 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ 三環式δ−オピオイド・モジュレーター
JP2008525483A (ja) 2004-12-22 2008-07-17 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ 三環式δ−オピオイド調節剤
ATE432279T1 (de) * 2004-12-22 2009-06-15 Janssen Pharmaceutica Nv Tricyclische delta-opioid-modulatoren
KR20070104380A (ko) * 2005-01-06 2007-10-25 얀센 파마슈티카 엔.브이. 트리사이클릭 δ-오피오이드 조절제
ATE490251T1 (de) * 2005-06-16 2010-12-15 Janssen Pharmaceutica Nv Tricyclische opioidmodulatoren

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3470188A (en) * 1967-01-05 1969-09-30 Smithkline Corp 9-cycloalkyl-lower alkyl-piperidylidene derivatives of xanthenes and thioxanthenes
US3974285A (en) * 1974-04-10 1976-08-10 Merck & Co., Inc. 10,11-Furo-derivatives of cyproheptadine
US4086350A (en) * 1974-11-06 1978-04-25 Smithkline Corporation Pharmaceutical compositions and method of producing anti-psychotic activity without extrapyramidal symptoms
US4031222A (en) * 1975-12-22 1977-06-21 Merck & Co., Inc. Trifluoromethylthio (and sulfonyl) derivatives of cyproheptadine analogs
US4073912A (en) * 1976-10-12 1978-02-14 Smithkline Corporation Piperidylidene derivatives of benzo-fused xanthenes, thioxanthenes and dibenzoxepins and antipsychotic use thereof

Also Published As

Publication number Publication date
EP0005607B1 (en) 1983-10-26
US4275209A (en) 1981-06-23
DK190179A (da) 1979-11-13
JPS54154772A (en) 1979-12-06
AU522926B2 (en) 1982-07-01
IE791105L (en) 1979-11-12
DE2966344D1 (en) 1983-12-01
CA1127648A (en) 1982-07-13
AU4694179A (en) 1979-11-15
IE48261B1 (en) 1984-11-14
NO150837B (no) 1984-09-17
US4309429A (en) 1982-01-05
NZ190373A (en) 1981-12-15
ZA792250B (en) 1980-08-27
US4285956A (en) 1981-08-25
ATE5141T1 (de) 1983-11-15
ES480468A1 (es) 1980-07-01
EP0005607A1 (en) 1979-11-28
NO150837C (no) 1985-01-09
FI791503A7 (fi) 1981-01-01

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