NO853859L - Triazolikinazolin-forbindelser. - Google Patents

Triazolikinazolin-forbindelser.

Info

Publication number
NO853859L
NO853859L NO853859A NO853859A NO853859L NO 853859 L NO853859 L NO 853859L NO 853859 A NO853859 A NO 853859A NO 853859 A NO853859 A NO 853859A NO 853859 L NO853859 L NO 853859L
Authority
NO
Norway
Prior art keywords
lower alkyl
formula
compound
stands
acid
Prior art date
Application number
NO853859A
Other languages
English (en)
Norwegian (no)
Inventor
John E Francis
Karl O Gelotte
Original Assignee
Ciba Geigy Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy Ag filed Critical Ciba Geigy Ag
Publication of NO853859L publication Critical patent/NO853859L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
NO853859A 1984-10-01 1985-09-30 Triazolikinazolin-forbindelser. NO853859L (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US65583184A 1984-10-01 1984-10-01

Publications (1)

Publication Number Publication Date
NO853859L true NO853859L (no) 1986-04-02

Family

ID=24630556

Family Applications (1)

Application Number Title Priority Date Filing Date
NO853859A NO853859L (no) 1984-10-01 1985-09-30 Triazolikinazolin-forbindelser.

Country Status (13)

Country Link
EP (1) EP0181282A1 (fr)
JP (1) JPS61165386A (fr)
AU (1) AU4813285A (fr)
DD (1) DD236931A5 (fr)
DK (1) DK442385A (fr)
ES (4) ES8707732A1 (fr)
FI (1) FI853736L (fr)
GR (1) GR852343B (fr)
HU (1) HU194566B (fr)
IL (1) IL76528A0 (fr)
NO (1) NO853859L (fr)
PT (1) PT81225B (fr)
ZA (1) ZA857529B (fr)

Families Citing this family (28)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3677445D1 (de) * 1985-09-30 1991-03-14 Ciba Geigy Ag 2-substituierte-e-kondensierte(1,5-c)-pyrimidine, pharmazeutische zubereitungen und ihre verwendung.
US4831013A (en) * 1986-03-20 1989-05-16 Ciba-Geigy Corporation 2-substituted-e-fused-[1,2,4]triazolo[1,5-c]pyrimidines, pharmaceutical compositions, and uses thereof
DE3781080T2 (de) * 1986-09-30 1992-12-24 Ciba Geigy Ag 2-substituierte-e-kondensierte(1,2,4)triazolo-(1,5-c)pyrimidine, pharmazeutische zubereitungen und ihre verwendung.
HU198484B (en) * 1986-11-05 1989-10-30 Egyt Gyogyszervegyeszeti Gyar Process for producing new condensed cyclic triazolo/1,5-a/pyrimidine derivatives
US4780464A (en) * 1986-12-08 1988-10-25 Warner-Lambert Company (1,2,4)triazolo(4,3-a)quinoxaline-4-amines
CA1331178C (fr) * 1988-02-05 1994-08-02 James J. Wade Triazolo ¬1,5-c| pyrimido ¬1,4| azines utilisees comme bronchodilatateurs
US5338743A (en) * 1988-06-06 1994-08-16 Fujisawa Pharmaceutical Co., Ltd. New use of the adenosine antagonist
US5095015A (en) * 1990-07-24 1992-03-10 Neurogen Corporation Certain azacycloalkyl imidazopyrimidines; a new class of gaba brain receptor ligands
US5185446A (en) * 1990-09-04 1993-02-09 Neurogen Corporation Certain cycloalkyl imidazopyrimidines; a new class of gaba brainreceptor ligands
US5744602A (en) * 1990-10-31 1998-04-28 Neurogen Corporation Certain imidazoquinoxalines; a new class of GABA brain receptor ligands
US5130430A (en) * 1990-10-31 1992-07-14 Neurogen Corporation 2-substituted imidazoquinoxaline diones, a new class of gaba brain receptor ligands
US5182386A (en) * 1991-08-27 1993-01-26 Neurogen Corporation Certain imidazoquinoxalinones; a new class of gaba brain receptor ligands
US5182290A (en) * 1991-08-27 1993-01-26 Neurogen Corporation Certain oxazoloquinolinones; a new class of GABA brain receptor ligands
US5243049A (en) * 1992-01-22 1993-09-07 Neurogen Corporation Certain pyrroloquinolinones: a new class of GABA brain receptor ligands
US5266698A (en) * 1992-04-30 1993-11-30 Neurogen Corporation Certain aryl and cycloalkyl fused imidazopyrazinediones; a new class of GABA brain receptor ligands
US5306819A (en) * 1992-08-27 1994-04-26 Neurogen Corporation Certain aryl a cycloalkyl fused imidazopyrazinols; and new class of GABA brain receptor ligands
DE4241564A1 (de) * 1992-12-10 1994-06-16 Basf Ag Triazolochinazoline zur Behandlung zentralnervöser Erkrankungen
ES2165393T3 (es) * 1993-07-27 2002-03-16 Kyowa Hakko Kogyo Kk Remedio contra la enfermedad de parkinson.
US5792766A (en) 1996-03-13 1998-08-11 Neurogen Corporation Imidazo 1,5-c! quinazolines; a new class of GABA brain receptor ligands
US5955465A (en) * 1996-03-22 1999-09-21 Neurogen Corporation 1,2,4-triazolo 4,3-c!quinazolin-3-ones and 1,2,4-triazolo 4,3-c!quinazolin-3-thiones
US5677309A (en) * 1996-03-22 1997-10-14 Neurogen Corporation 1,2,4-triazolo 4,3-c! quinazolin-3-ones and 1,2,4-triazolo 4,3-c!quinazolin-3-thiones; a new class of GABA brain receptor ligands
AU1130700A (en) * 1998-10-23 2000-05-15 Dow Agrosciences Llc Insecticidal 1-(substituted pyridyl)-1,2,4-triazoles
AU2013277294C1 (en) 2012-06-18 2018-02-08 Dart Neuroscience (Cayman) Ltd Substituted thiophene- and furan-fused azolopyrimidine-5-(6h)-one compounds
WO2014101113A1 (fr) * 2012-12-28 2014-07-03 Merck Sharp & Dohme Corp. Composés de 7-méthoxy-[1,2,4]triazolo[1,5-c]quinazoline-5-amine à substitution pipérazine présentant des propriétés d'antagoniste d'a2a
WO2014101120A1 (fr) 2012-12-28 2014-07-03 Merck Sharp & Dohme Corp. Composés de 7-méthoxy-[1,2,4]triazolo[1,5-c]quinazoline-5-amine à substitution hétérobicyclo présentant des propriétés d'antagoniste d'a2a
WO2017008205A1 (fr) 2015-07-10 2017-01-19 Merck Sharp & Dohme Corp. Composés d'aminoquinazoline substitués a titre d'antagonistes du récepteur a2a
JP6420400B2 (ja) * 2017-04-12 2018-11-07 ダート・ニューロサイエンス・（ケイマン）・リミテッド 置換ピリジンアゾロピリミジン−５−（６ｈ）−オン化合物
GB2575490A (en) * 2018-07-12 2020-01-15 Recordati Ind Chimica E Farmaceutica Spa P2X3 receptor antagonists

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4252945A (en) * 1979-07-11 1981-02-24 E. R. Squibb & Sons, Inc. Process for preparing pyrazolo[1,5-c]-quinazoline derivatives and novel intermediates
DE3146599A1 (de) * 1981-11-25 1983-07-07 Basf Ag, 6700 Ludwigshafen Neue triazolochinazoline, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische zubereitungen

Also Published As

Publication number Publication date
AU4813285A (en) 1986-04-10
ES557118A0 (es) 1988-01-01
HUT38941A (en) 1986-07-28
ES557119A0 (es) 1988-05-16
DK442385D0 (da) 1985-09-30
ES557120A0 (es) 1988-05-16
FI853736A7 (fi) 1986-04-02
EP0181282A1 (fr) 1986-05-14
ZA857529B (en) 1986-05-28
JPS61165386A (ja) 1986-07-26
IL76528A0 (en) 1986-01-31
DK442385A (da) 1986-04-02
ES8802387A1 (es) 1988-05-16
DD236931A5 (de) 1986-06-25
GR852343B (fr) 1986-01-28
ES8707732A1 (es) 1987-08-16
ES557117A0 (es) 1987-08-16
ES8801277A1 (es) 1988-01-01
ES8802386A1 (es) 1988-05-16
HU194566B (en) 1988-02-29
FI853736A0 (fi) 1985-09-27
FI853736L (fi) 1986-04-02
PT81225B (en) 1987-07-15
PT81225A (en) 1985-10-01

Similar Documents

Publication Publication Date Title
NO853859L (no) Triazolikinazolin-forbindelser.
US4713383A (en) Triazoloquinazoline compounds, and their methods of preparation, pharmaceutical compositions, and uses
EP1507780B1 (fr) Composes de pyrazolo-pyrimidine aniline utiles comme inhibiteurs de kinase.
AU2004235907B2 (en) Fused pyrimidine derivatives with CRF activity
RU2229299C2 (ru) Применение диазепинов для приготовления лекарственных средств, предназначенных для лечения патологических состояний или заболеваний, связанных с действием одного из рецепторов соматостатина
US7741332B2 (en) Fused ring heterocycles as potassium channel modulators
CA2288910C (fr) Pyrazolopyrimidinones pour des dysfonctions sexuelles
CA1288097C (fr) Compositions pharmaceutiques de type 2-substituant-anneau e condense-(1,2,4) triazolo (1,5c) pyrimidines, et leurs utilisations
AU8027187A (en) 2-substituted-E-fused-(1,2,4)triazolo(1,5-C)pyrimidines pharmaceutical compositions
US20050143398A1 (en) Phenyl-aniline substituted bicyclic compounds useful as kinase inhibitors
US20080269238A1 (en) Thiazolopyrimidine Derivative
AU2005321946A1 (en) Enzyme modulators and treatments
SK281077B6 (sk) Heterocyklické zlúčeniny, spôsob ich prípravy, farmaceutický prostriedok a použitie
AU2012296529A1 (en) Heteroaryl sodium channel inhibitors
BR122017002951A2 (pt) amidas heterocíclicas como inibidores de quinases
EP4117784B1 (fr) Composés modulateurs de gpr52
MX2014008158A (es) Compuestos de piridazina-amida.
EP2083816A2 (fr) Composés d'amide hétérocyclique utiles comme inhibiteurs de kinase
EP0807633A2 (fr) (5,6)-Pyrimidin-4-ones condensées à hétéroaryle, substituées en 2,3
CA3122623A1 (fr) Composes d'halogenoallylamine et leur utilisation
AU689468B2 (en) Imidazopyridine
US4831013A (en) 2-substituted-e-fused-[1,2,4]triazolo[1,5-c]pyrimidines, pharmaceutical compositions, and uses thereof
WO2001044250A1 (fr) 1,2,3-TRIAZOLO[1,5-a]QUINAZOLINES SUBSTITUE NOOTROPE
JP5324785B2 (ja) 複素環アミド化合物及びその用途
JPS62135475A (ja) ２−置換−ｅ−融合−〔１，２，４〕トリアゾロ−〔１，５−Ｃ〕ピリミジン